ATE174917T1 - Pyrazolo(1,5-a>pyrimidinderivate und sie enthaltende antiinflammatorische mittel - Google Patents

Pyrazolo(1,5-a>pyrimidinderivate und sie enthaltende antiinflammatorische mittel

Info

Publication number
ATE174917T1
ATE174917T1 AT91913666T AT91913666T ATE174917T1 AT E174917 T1 ATE174917 T1 AT E174917T1 AT 91913666 T AT91913666 T AT 91913666T AT 91913666 T AT91913666 T AT 91913666T AT E174917 T1 ATE174917 T1 AT E174917T1
Authority
AT
Austria
Prior art keywords
lower alkyl
substituted
hydroxy
phenyl
hydrogen
Prior art date
Application number
AT91913666T
Other languages
German (de)
English (en)
Inventor
Makoto Inoue
Kinji Hashimoto
Toshiko Kuwahara
Matsushige-Cho
Yukio Sugimoto
Takuji Uesako
Toshiaki Funato
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Application granted granted Critical
Publication of ATE174917T1 publication Critical patent/ATE174917T1/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pain & Pain Management (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
AT91913666T 1991-04-22 1991-08-06 Pyrazolo(1,5-a>pyrimidinderivate und sie enthaltende antiinflammatorische mittel ATE174917T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP9070791 1991-04-22

Publications (1)

Publication Number Publication Date
ATE174917T1 true ATE174917T1 (de) 1999-01-15

Family

ID=14006001

Family Applications (1)

Application Number Title Priority Date Filing Date
AT91913666T ATE174917T1 (de) 1991-04-22 1991-08-06 Pyrazolo(1,5-a>pyrimidinderivate und sie enthaltende antiinflammatorische mittel

Country Status (12)

Country Link
US (1) US5688949A (env)
EP (1) EP0591528B1 (env)
JP (1) JPH0570353A (env)
KR (1) KR100191774B1 (env)
AT (1) ATE174917T1 (env)
AU (1) AU651986B2 (env)
CA (1) CA2107479C (env)
DE (1) DE69130683T2 (env)
DK (1) DK0591528T3 (env)
ES (1) ES2126573T3 (env)
TW (1) TW221434B (env)
WO (1) WO1992018504A1 (env)

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US7642266B2 (en) * 2005-10-06 2010-01-05 Schering Corporation Substituted pyrazolo[1,5-a]pyrimidines as protein kinase inhibitors
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EP2398500B1 (en) 2009-02-20 2019-03-13 2-BBB Medicines B.V. Glutathione-based drug delivery system
ES2942923T3 (es) 2009-05-06 2023-06-07 Laboratory Skin Care Inc Composiciones de administración dérmica que comprenden complejos de agente activo-partículas de fosfato de calcio y métodos de uso de las mismas
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KR101483834B1 (ko) * 2009-12-23 2015-01-16 카트호리이케 유니버시타이트 로이펜 항바이러스 화합물
US8927562B2 (en) * 2010-09-28 2015-01-06 Merck Sharp & Dohme Corp. Fused tricyclic inhibitors of mammalian target of rapamycin
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates
BR112013011737A2 (pt) 2010-11-15 2016-08-09 Univ Leuven Kath composto, uso de um composto composição farmacêutica, e, método de tratamento ou prevenção de uma infecção por hiv
US8633198B1 (en) 2011-09-20 2014-01-21 Nant Holdings Ip, Llc Small molecule inhibitors of influenza A RNA-dependent RNA polymerase
WO2015088516A1 (en) * 2013-12-11 2015-06-18 Nant Holdings Ip, Llc Small molecule inhibitors of influenza a rna-dependent rna polymerase
AU2015208205B2 (en) * 2014-01-22 2019-12-05 Curovir Ab Pyrazolo[1,5-a]pyrimidines as antiviral compounds
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DE102018201598A1 (de) 2018-02-02 2019-08-08 Beiersdorf Ag Stabile Wundheilsalbe
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Also Published As

Publication number Publication date
CA2107479C (en) 1997-12-16
ES2126573T3 (es) 1999-04-01
JPH0570353A (ja) 1993-03-23
AU8295891A (en) 1992-11-17
DE69130683T2 (de) 1999-05-06
DE69130683D1 (de) 1999-02-04
EP0591528B1 (en) 1998-12-23
AU651986B2 (en) 1994-08-11
CA2107479A1 (en) 1992-10-23
EP0591528A4 (en) 1995-02-15
US5688949A (en) 1997-11-18
DK0591528T3 (da) 1999-08-23
EP0591528A1 (en) 1994-04-13
KR100191774B1 (ko) 1999-06-15
TW221434B (env) 1994-03-01
WO1992018504A1 (en) 1992-10-29

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Legal Events

Date Code Title Description
UEP Publication of translation of european patent specification
REN Ceased due to non-payment of the annual fee