AT393508B - Verfahren zur herstellung von carboxyalkyldipeptiden - Google Patents

Verfahren zur herstellung von carboxyalkyldipeptiden Download PDF

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Publication number
AT393508B
AT393508B AT2012/83A AT201283A AT393508B AT 393508 B AT393508 B AT 393508B AT 2012/83 A AT2012/83 A AT 2012/83A AT 201283 A AT201283 A AT 201283A AT 393508 B AT393508 B AT 393508B
Authority
AT
Austria
Prior art keywords
formula
compound
dipeptide
meanings given
preparation
Prior art date
Application number
AT2012/83A
Other languages
German (de)
English (en)
Other versions
ATA201283A (de
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27011123&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AT393508(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of ATA201283A publication Critical patent/ATA201283A/de
Application granted granted Critical
Publication of AT393508B publication Critical patent/AT393508B/de

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
    • C07K5/06052—Val-amino acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06026—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atom, i.e. Gly or Ala
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
    • C07K5/06043—Leu-amino acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06078—Dipeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06086—Dipeptides with the first amino acid being basic
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S530/00—Chemistry: natural resins or derivatives; peptides or proteins; lignins or reaction products thereof
    • Y10S530/80—Antihypertensive peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
AT2012/83A 1982-06-07 1983-06-01 Verfahren zur herstellung von carboxyalkyldipeptiden AT393508B (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38574582A 1982-06-07 1982-06-07
US06/462,727 US4442030A (en) 1982-06-07 1983-01-31 Process for preparing carboxyalkyl dipeptides

Publications (2)

Publication Number Publication Date
ATA201283A ATA201283A (de) 1991-04-15
AT393508B true AT393508B (de) 1991-11-11

Family

ID=27011123

Family Applications (1)

Application Number Title Priority Date Filing Date
AT2012/83A AT393508B (de) 1982-06-07 1983-06-01 Verfahren zur herstellung von carboxyalkyldipeptiden

Country Status (7)

Country Link
US (1) US4442030A (OSRAM)
KR (1) KR910001720B1 (OSRAM)
AT (1) AT393508B (OSRAM)
ES (2) ES8502082A1 (OSRAM)
GR (1) GR78282B (OSRAM)
NO (1) NO166231C (OSRAM)
PT (2) PT76790B (OSRAM)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4746676A (en) * 1984-09-12 1988-05-24 Rorer Pharmaceutical Corporation Carboxyalkyl dipeptide compounds
TW533196B (en) * 1998-09-23 2003-05-21 Merck & Co Inc Improved stereoselective process for ENALAPRIL

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0012401A1 (en) * 1978-12-11 1980-06-25 Merck & Co. Inc. Carboxyalkyl dipeptide derivatives, process for preparing them and pharmaceutical composition containing them

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0012401A1 (en) * 1978-12-11 1980-06-25 Merck & Co. Inc. Carboxyalkyl dipeptide derivatives, process for preparing them and pharmaceutical composition containing them

Also Published As

Publication number Publication date
NO166231B (no) 1991-03-11
ATA201283A (de) 1991-04-15
ES522753A0 (es) 1984-12-16
ES8506264A1 (es) 1985-07-01
KR840005079A (ko) 1984-11-03
PT76790B (en) 1986-04-09
PT76790A (en) 1983-07-01
KR910001720B1 (ko) 1991-03-22
ES535853A0 (es) 1985-07-01
PT76790B1 (pt) 1996-09-30
US4442030A (en) 1984-04-10
NO166231C (no) 1991-06-19
ES8502082A1 (es) 1984-12-16
NO832036L (no) 1983-12-08
GR78282B (OSRAM) 1984-09-26

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