AT351547B - METHOD FOR PRODUCING NEW THIENO- (1,5) -BENZODIAZEPINES AND THEIR ACID ADDITION SALTS - Google Patents
METHOD FOR PRODUCING NEW THIENO- (1,5) -BENZODIAZEPINES AND THEIR ACID ADDITION SALTSInfo
- Publication number
- AT351547B AT351547B AT898275A AT898275A AT351547B AT 351547 B AT351547 B AT 351547B AT 898275 A AT898275 A AT 898275A AT 898275 A AT898275 A AT 898275A AT 351547 B AT351547 B AT 351547B
- Authority
- AT
- Austria
- Prior art keywords
- benzodiazepines
- acid addition
- addition salts
- producing new
- new thieno
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
- C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB51240/74A GB1533235A (en) | 1974-11-26 | 1974-11-26 | Benzodiazepine derivatives |
Publications (2)
Publication Number | Publication Date |
---|---|
ATA898275A ATA898275A (en) | 1979-01-15 |
AT351547B true AT351547B (en) | 1979-07-25 |
Family
ID=10459213
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT898275A AT351547B (en) | 1974-11-26 | 1975-11-26 | METHOD FOR PRODUCING NEW THIENO- (1,5) -BENZODIAZEPINES AND THEIR ACID ADDITION SALTS |
Country Status (30)
Country | Link |
---|---|
JP (1) | JPS6044314B2 (en) |
AR (1) | AR221203A1 (en) |
AT (1) | AT351547B (en) |
AU (1) | AU506340B2 (en) |
BE (1) | BE835932A (en) |
BG (1) | BG29573A3 (en) |
CA (1) | CA1075687A (en) |
CH (2) | CH613454A5 (en) |
CS (1) | CS236753B2 (en) |
DD (1) | DD123343A5 (en) |
DE (1) | DE2552403C2 (en) |
DK (1) | DK146887C (en) |
ES (1) | ES443011A1 (en) |
FR (1) | FR2292479A1 (en) |
GB (1) | GB1533235A (en) |
HK (1) | HK58681A (en) |
HU (1) | HU172493B (en) |
IE (1) | IE42564B1 (en) |
IL (1) | IL48502A (en) |
KE (1) | KE3163A (en) |
MY (1) | MY8200149A (en) |
NL (1) | NL186088C (en) |
NZ (1) | NZ179335A (en) |
PH (2) | PH11669A (en) |
PL (1) | PL100135B1 (en) |
RO (1) | RO69912A (en) |
SE (2) | SE421209B (en) |
SU (2) | SU629879A3 (en) |
YU (1) | YU298375A (en) |
ZA (1) | ZA757344B (en) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL62792A (en) * | 1980-05-07 | 1985-02-28 | Byk Gulden Lomberg Chem Fab | Acylated dihydrothienodiazepinone compounds,process for their preparation,and medicaments containing them |
GB8819059D0 (en) * | 1988-08-11 | 1988-09-14 | Lilly Industries Ltd | Benzodiazepine compounds & their use as pharmaceuticals |
GB9009229D0 (en) * | 1990-04-25 | 1990-06-20 | Lilly Industries Ltd | Pharmaceutical compounds |
DE69329887T2 (en) * | 1992-05-29 | 2001-05-23 | Lilly Co Eli | Thienobenzodiazepine derivatives for the treatment of disorders of the central nervous system |
CA2234641A1 (en) * | 1995-11-01 | 1997-05-09 | Merck & Co., Inc. | Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases |
US6043358A (en) | 1995-11-01 | 2000-03-28 | Merck & Co., Inc. | Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases |
CN1268949A (en) | 1997-09-02 | 2000-10-04 | 吉富制药株式会社 | Fused thiophene compounds and medical use thereof |
PL199016B1 (en) * | 2002-06-20 | 2008-08-29 | Adamed Sp Z Oo | Method of manufacture of alanzapine, new derivative of n-demethyl olanzapine and method of manufacture of new derivative of n-demethyl olanzapine |
SI21270A (en) | 2002-07-15 | 2004-02-29 | Krka, Tovarna Zdravil, D.D., Novo Mesto | Crystal forms of olanzapine and procedures for their preparation |
DE10301923B3 (en) * | 2003-01-17 | 2004-09-16 | Krka Tovarna Zdravil, D.D. | Process and intermediates for the production of olanzapine |
EP1711503A1 (en) * | 2004-01-27 | 2006-10-18 | Synthon B.V. | Synthesis of olanzapine and intermediates thereof |
AR048272A1 (en) | 2004-03-18 | 2006-04-12 | Lek Pharmaceuticals | SYNTHESIS OF 2 METHYL - 4- (4- METHYL -1- PIPERAZINIL) - 10 H- TIENO (2,3-B) (1,5) BENZODIAZEPIN AND ITS SALTS, METHODS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING IT AND ITS USE IN THE MANUFACTURE OF MEDICINES FOR THE TREATMENT OF MENTAL DISEASES. |
JP5025469B2 (en) * | 2004-06-30 | 2012-09-12 | アサーシス, インク. | Substituted azepine derivatives as serotonin receptor modulators |
EP2292624A1 (en) | 2009-07-20 | 2011-03-09 | LEK Pharmaceuticals d.d. | Process for the purification of olanzapine |
-
1974
- 1974-11-25 SU SU742191705A patent/SU629879A3/en active
- 1974-11-26 GB GB51240/74A patent/GB1533235A/en not_active Expired
-
1975
- 1975-11-20 IL IL48502A patent/IL48502A/en unknown
- 1975-11-20 DK DK524175A patent/DK146887C/en active
- 1975-11-20 CA CA240,082A patent/CA1075687A/en not_active Expired
- 1975-11-21 PH PH17788A patent/PH11669A/en unknown
- 1975-11-21 AU AU86858/75A patent/AU506340B2/en not_active Expired
- 1975-11-22 DE DE2552403A patent/DE2552403C2/en not_active Expired
- 1975-11-24 SE SE7513185A patent/SE421209B/en not_active IP Right Cessation
- 1975-11-24 NZ NZ179335A patent/NZ179335A/en unknown
- 1975-11-24 CH CH1517275A patent/CH613454A5/en not_active IP Right Cessation
- 1975-11-24 ZA ZA757344A patent/ZA757344B/en unknown
- 1975-11-24 CH CH604478A patent/CH613455A5/en not_active IP Right Cessation
- 1975-11-25 AR AR261340A patent/AR221203A1/en active
- 1975-11-25 JP JP50141080A patent/JPS6044314B2/en not_active Expired
- 1975-11-25 RO RO7584018A patent/RO69912A/en unknown
- 1975-11-25 BE BE6045266A patent/BE835932A/en not_active IP Right Cessation
- 1975-11-25 YU YU02983/75A patent/YU298375A/en unknown
- 1975-11-25 IE IE2565/75A patent/IE42564B1/en unknown
- 1975-11-25 DD DD189666A patent/DD123343A5/xx unknown
- 1975-11-25 FR FR7535900A patent/FR2292479A1/en active Granted
- 1975-11-26 PL PL1975184991A patent/PL100135B1/en unknown
- 1975-11-26 BG BG7531601A patent/BG29573A3/en unknown
- 1975-11-26 HU HU75LI00000284A patent/HU172493B/en unknown
- 1975-11-26 CS CS757991A patent/CS236753B2/en unknown
- 1975-11-26 ES ES443011A patent/ES443011A1/en not_active Expired
- 1975-11-26 AT AT898275A patent/AT351547B/en not_active IP Right Cessation
- 1975-11-26 NL NLAANVRAGE7513833,A patent/NL186088C/en not_active IP Right Cessation
-
1976
- 1976-10-07 SU SU762406250A patent/SU626702A3/en active
-
1977
- 1977-02-22 PH PH19480A patent/PH24534A/en unknown
-
1978
- 1978-11-27 SE SE7812194A patent/SE429045B/en not_active IP Right Cessation
-
1981
- 1981-09-24 KE KE3163A patent/KE3163A/en unknown
- 1981-11-26 HK HK586/81A patent/HK58681A/en unknown
-
1982
- 1982-12-30 MY MY149/82A patent/MY8200149A/en unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ELA | Expired due to lapse of time |