AR075472A1 - Proceso para la preparacion de benzonorbornenos - Google Patents

Proceso para la preparacion de benzonorbornenos

Info

Publication number
AR075472A1
AR075472A1 ARP090104114A ARP090104114A AR075472A1 AR 075472 A1 AR075472 A1 AR 075472A1 AR P090104114 A ARP090104114 A AR P090104114A AR P090104114 A ARP090104114 A AR P090104114A AR 075472 A1 AR075472 A1 AR 075472A1
Authority
AR
Argentina
Prior art keywords
compound
formula
chlorine
preparation
reacting
Prior art date
Application number
ARP090104114A
Other languages
English (en)
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP08018721A external-priority patent/EP2181981A1/en
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of AR075472A1 publication Critical patent/AR075472A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/30Preparation of compounds containing amino groups bound to a carbon skeleton by reduction of nitrogen-to-oxygen or nitrogen-to-nitrogen bonds
    • C07C209/32Preparation of compounds containing amino groups bound to a carbon skeleton by reduction of nitrogen-to-oxygen or nitrogen-to-nitrogen bonds by reduction of nitro groups
    • C07C209/36Preparation of compounds containing amino groups bound to a carbon skeleton by reduction of nitrogen-to-oxygen or nitrogen-to-nitrogen bonds by reduction of nitro groups by reduction of nitro groups bound to carbon atoms of six-membered aromatic rings in presence of hydrogen-containing gases and a catalyst
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00Preparation of halogenated hydrocarbons
    • C07C17/26Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/32Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by introduction of halogenated alkyl groups into ring compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/27Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00Preparation of halogenated hydrocarbons
    • C07C17/23Preparation of halogenated hydrocarbons by dehalogenation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00Preparation of halogenated hydrocarbons
    • C07C17/25Preparation of halogenated hydrocarbons by splitting-off hydrogen halides from halogenated hydrocarbons
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00Preparation of halogenated hydrocarbons
    • C07C17/26Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00Preparation of halogenated hydrocarbons
    • C07C17/26Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/263Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions
    • C07C17/266Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions of hydrocarbons and halogenated hydrocarbons
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C201/00Preparation of esters of nitric or nitrous acid or of compounds containing nitro or nitroso groups bound to a carbon skeleton
    • C07C201/06Preparation of nitro compounds
    • C07C201/12Preparation of nitro compounds by reactions not involving the formation of nitro groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/06Compounds containing nitro groups bound to a carbon skeleton having nitro groups bound to carbon atoms of six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/07Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms
    • C07C205/11Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms having nitro groups bound to carbon atoms of six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/07Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms
    • C07C205/11Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms having nitro groups bound to carbon atoms of six-membered aromatic rings
    • C07C205/12Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by halogen atoms having nitro groups bound to carbon atoms of six-membered aromatic rings the six-membered aromatic ring or a condensed ring system containing that ring being substituted by halogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/30Preparation of compounds containing amino groups bound to a carbon skeleton by reduction of nitrogen-to-oxygen or nitrogen-to-nitrogen bonds
    • C07C209/32Preparation of compounds containing amino groups bound to a carbon skeleton by reduction of nitrogen-to-oxygen or nitrogen-to-nitrogen bonds by reduction of nitro groups
    • C07C209/36Preparation of compounds containing amino groups bound to a carbon skeleton by reduction of nitrogen-to-oxygen or nitrogen-to-nitrogen bonds by reduction of nitro groups by reduction of nitro groups bound to carbon atoms of six-membered aromatic rings in presence of hydrogen-containing gases and a catalyst
    • C07C209/365Preparation of compounds containing amino groups bound to a carbon skeleton by reduction of nitrogen-to-oxygen or nitrogen-to-nitrogen bonds by reduction of nitro groups by reduction of nitro groups bound to carbon atoms of six-membered aromatic rings in presence of hydrogen-containing gases and a catalyst by reduction with preservation of halogen-atoms in compounds containing nitro groups and halogen atoms bound to the same carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00Compounds containing amino groups bound to a carbon skeleton
    • C07C211/43Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/57Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton
    • C07C211/61Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton with at least one of the condensed ring systems formed by three or more rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C22/00Cyclic compounds containing halogen atoms bound to an acyclic carbon atom
    • C07C22/02Cyclic compounds containing halogen atoms bound to an acyclic carbon atom having unsaturation in the rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C22/00Cyclic compounds containing halogen atoms bound to an acyclic carbon atom
    • C07C22/02Cyclic compounds containing halogen atoms bound to an acyclic carbon atom having unsaturation in the rings
    • C07C22/04Cyclic compounds containing halogen atoms bound to an acyclic carbon atom having unsaturation in the rings containing six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C23/00Compounds containing at least one halogen atom bound to a ring other than a six-membered aromatic ring
    • C07C23/02Monocyclic halogenated hydrocarbons
    • C07C23/08Monocyclic halogenated hydrocarbons with a five-membered ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/06Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/10Systems containing only non-condensed rings with a five-membered ring the ring being unsaturated
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00Systems containing at least three condensed rings
    • C07C2603/56Ring systems containing bridged rings
    • C07C2603/58Ring systems containing bridged rings containing three rings
    • C07C2603/60Ring systems containing bridged rings containing three rings containing at least one ring with less than six members
    • C07C2603/66Ring systems containing bridged rings containing three rings containing at least one ring with less than six members containing five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Emergency Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Saccharide Compounds (AREA)

Abstract

La presente solicitud se refiere a un proceso novedoso para la preparacion de 9-diclorometilen-1,2,3,4-tetrahidro-1,4-metano-naftalen-5-ilamina, proceso que comprende: a) hacer reaccionar ciclopentadieno en presencia de un iniciador de radicales y CXCl3, donde X es cloro o bromo, para obtener un compuesto de formula (2), aa) hacer reaccionar ciclopentadieno con CXCl3, donde X es cloro, en presencia de un catalizador metálico para obtener un compuesto de formula (2) donde X es cloro, b) hacer reaccionar el compuesto de formula (2) con una base en presencia de un solvente apropiado para obtener el compuesto de formula (3); c) y convertir el compuesto de formula (3) en presencia de 1,2-deshidro-6- nitrobenceno para obtener el compuesto de formula (4) y d) hidrogenar el compuesto de formula (4) en presencia de un catalizador metálico.
ARP090104114A 2008-10-27 2009-10-26 Proceso para la preparacion de benzonorbornenos AR075472A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08018721A EP2181981A1 (en) 2008-10-27 2008-10-27 Process for the preparation of benzonorbornenes
EP09161388 2009-05-28

Publications (1)

Publication Number Publication Date
AR075472A1 true AR075472A1 (es) 2011-04-06

Family

ID=41175685

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP090104114A AR075472A1 (es) 2008-10-27 2009-10-26 Proceso para la preparacion de benzonorbornenos

Country Status (24)

Country Link
US (3) US9115043B2 (es)
EP (1) EP2349975B1 (es)
JP (1) JP5406302B2 (es)
KR (1) KR101596814B1 (es)
CN (2) CN103319305B (es)
AR (1) AR075472A1 (es)
AU (1) AU2009309884B2 (es)
BR (1) BRPI0920833B1 (es)
CA (1) CA2739656C (es)
CO (1) CO6361987A2 (es)
CR (1) CR20110208A (es)
EA (1) EA019039B1 (es)
EC (1) ECSP11011004A (es)
EG (1) EG26332A (es)
ES (1) ES2431818T3 (es)
GE (1) GEP20135747B (es)
IL (1) IL211975A (es)
MX (1) MX2011003758A (es)
MY (1) MY150841A (es)
NZ (1) NZ591977A (es)
TW (1) TWI438176B (es)
UY (1) UY32195A (es)
WO (1) WO2010049228A1 (es)
ZA (1) ZA201102453B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2453919T3 (es) * 2010-04-20 2014-04-08 Syngenta Participations Ag Proceso para preparar amidas de ácidos carboxílicos pirazólicos
EP2433922A1 (en) * 2010-08-25 2012-03-28 Syngenta Participations AG Process for the preparation of dichlorofulvene
TWI510472B (zh) 2012-02-15 2015-12-01 Syngenta Participations Ag 立體選擇性製備吡唑羧醯胺之方法
JP7220151B2 (ja) 2017-08-28 2023-02-09 株式会社日本ファインケム ピラゾール-4-カルボキサミド誘導体の製造方法
CN111454157B (zh) * 2020-05-14 2022-07-22 利民化学有限责任公司 一种3-硝基苯炔的制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH07291876A (ja) * 1994-03-03 1995-11-07 Ricoh Co Ltd シクロペンタジエン化合物及びそれを含有する電子写真感光体
JP4294129B2 (ja) * 1998-11-04 2009-07-08 旭化成ケミカルズ株式会社 シクロアルケンの塩素化法
CN101979374A (zh) * 2005-09-16 2011-02-23 先正达参股股份有限公司 酰胺的制备方法
PT1940813E (pt) * 2005-10-25 2011-01-20 Syngenta Participations Ag Derivados de amidas heterocíclicas úteis como microbicidas
EP2316814A1 (en) 2005-12-12 2011-05-04 Syngenta Participations AG Process for preparation of halogen substituted benzonorbornenes derivatives
CA2842787C (en) * 2007-04-25 2016-03-22 Syngenta Participations Ag Fungicidal compositions comprising a 3-substituted 1-methyl-1h-pyrazole-4-carboxylic acid (9-dihalomethylidene-benzonorbornene-5-yl) amide and a second fungicide

Also Published As

Publication number Publication date
CN102197016B (zh) 2013-12-18
CA2739656C (en) 2016-08-16
EP2349975B1 (en) 2013-07-31
AU2009309884B2 (en) 2013-08-29
US9115043B2 (en) 2015-08-25
EG26332A (en) 2013-08-19
MY150841A (en) 2014-02-28
ECSP11011004A (es) 2011-05-31
AU2009309884A1 (en) 2010-05-06
CR20110208A (es) 2011-05-11
JP2012506842A (ja) 2012-03-22
US20180016211A1 (en) 2018-01-18
US9878970B1 (en) 2018-01-30
GEP20135747B (en) 2013-02-11
KR20110074982A (ko) 2011-07-05
TWI438176B (zh) 2014-05-21
IL211975A0 (en) 2011-06-30
CN103319305B (zh) 2015-04-08
TW201016642A (en) 2010-05-01
WO2010049228A1 (en) 2010-05-06
ES2431818T3 (es) 2013-11-28
ZA201102453B (en) 2011-12-28
CN102197016A (zh) 2011-09-21
CN103319305A (zh) 2013-09-25
CA2739656A1 (en) 2010-05-06
US20150141712A1 (en) 2015-05-21
UY32195A (es) 2010-05-31
KR101596814B1 (ko) 2016-02-23
US20110207958A1 (en) 2011-08-25
JP5406302B2 (ja) 2014-02-05
EA019039B1 (ru) 2013-12-30
EP2349975A1 (en) 2011-08-03
EA201100665A1 (ru) 2011-12-30
CO6361987A2 (es) 2012-01-20
MX2011003758A (es) 2011-04-27
BRPI0920833A2 (pt) 2015-12-22
BRPI0920833B1 (pt) 2018-02-06
US9796646B2 (en) 2017-10-24
IL211975A (en) 2015-06-30
NZ591977A (en) 2012-08-31

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