UY33340A - Proceso para la preparación de amidas de ácido pirazol carboxílico - Google Patents

Proceso para la preparación de amidas de ácido pirazol carboxílico

Info

Publication number
UY33340A
UY33340A UY0001033340A UY33340A UY33340A UY 33340 A UY33340 A UY 33340A UY 0001033340 A UY0001033340 A UY 0001033340A UY 33340 A UY33340 A UY 33340A UY 33340 A UY33340 A UY 33340A
Authority
UY
Uruguay
Prior art keywords
preparation
amidas
pirazol
formula
carboxyl acid
Prior art date
Application number
UY0001033340A
Other languages
English (en)
Inventor
Trah Stephan
Vettiger Thomas
Rommel Michael
Dumeunier Raphael
Schleth Florian
Original Assignee
Syngenta Participations Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag filed Critical Syngenta Participations Ag
Publication of UY33340A publication Critical patent/UY33340A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/23—Preparation of halogenated hydrocarbons by dehalogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/26—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/30—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by a Diels-Alder synthesis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/04—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups
    • C07C209/06—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms
    • C07C209/10—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms with formation of amino groups bound to carbon atoms of six-membered aromatic rings or from amines having nitrogen atoms bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/24—Halogenated aromatic hydrocarbons with unsaturated side chains
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C29/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
    • C07C29/132—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C35/00—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C07C35/48—Halogenated derivatives
    • C07C35/52—Alcohols with a condensed ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/27—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation
    • C07C45/29—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation of hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/12—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
    • C07D303/16—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by esterified hydroxyl radicals
    • C07D303/17—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by esterified hydroxyl radicals containing oxirane rings condensed with carbocyclic ring systems having three or more relevant rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/56—Ring systems containing bridged rings
    • C07C2603/58—Ring systems containing bridged rings containing three rings
    • C07C2603/60—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members
    • C07C2603/66—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members containing five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Epoxy Compounds (AREA)
  • Catalysts (AREA)

Abstract

La invención se refiere a la preparación del compuesto I proceso que comprende los siguientes pasos a) hacer reaccionar un compuesto de la fórmula II donde X es cloro o bromo, con una especie organometálica en una atmósfera inerte para obtener un halobencino de la fórmula X hacer reaccionar el halobencino de la fórmula X así formando con ciclopentadieno para obtener III y luego de una serie de pasos intermedios, se llega, según se describe en la memoria descriptiva, a obtener el compuesto de la fórmula I.
UY0001033340A 2010-04-20 2011-04-15 Proceso para la preparación de amidas de ácido pirazol carboxílico UY33340A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP10160438 2010-04-20

Publications (1)

Publication Number Publication Date
UY33340A true UY33340A (es) 2011-12-01

Family

ID=44072655

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001033340A UY33340A (es) 2010-04-20 2011-04-15 Proceso para la preparación de amidas de ácido pirazol carboxílico

Country Status (12)

Country Link
US (1) US8519152B2 (es)
EP (1) EP2560959B1 (es)
JP (1) JP5684896B2 (es)
CN (1) CN102906072B (es)
AR (1) AR080922A1 (es)
BR (1) BR112012026631B1 (es)
ES (1) ES2513540T3 (es)
IL (1) IL222398A (es)
MX (1) MX2012012005A (es)
TW (1) TWI428325B (es)
UY (1) UY33340A (es)
WO (1) WO2011131545A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112012026456B1 (pt) * 2010-04-20 2017-06-27 Syngenta Participations Ag Process for the preparation of carboxylic pyrazole acid amides
TWI534126B (zh) * 2011-01-25 2016-05-21 先正達合夥公司 用於製備吡唑羧酸醯胺之方法
GB201403438D0 (en) 2014-02-27 2014-04-16 Syngenta Participations Ag Polymorphs
WO2024017788A1 (en) 2022-07-22 2024-01-25 Syngenta Crop Protection Ag Solid form of a heterocyclic amide derivative

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH075487B2 (ja) 1985-11-14 1995-01-25 住友化学工業株式会社 １―ブロモ―２―クロロ―４―フルオロベンゼンの製造法
US5093347A (en) 1991-01-28 1992-03-03 Monsanto Company 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use
US7223879B2 (en) 1998-07-10 2007-05-29 Massachusetts Institute Of Technology Ligands for metals and improved metal-catalyzed processes based thereon
CN101296913B (zh) 2005-10-25 2013-02-13 先正达参股股份有限公司 用作杀微生物剂的杂环酰胺衍生物
WO2007124907A2 (en) 2006-04-27 2007-11-08 Syngenta Participations Ag Heterocyclyl-carboxylic acid (benzonorbornene-5-yl)amide derivatives as fungicides for agrochemical use
EP2076123B1 (en) 2006-10-25 2011-06-01 Syngenta Limited Process for the production of substituted bromobenzenes
CN102264705A (zh) * 2008-12-24 2011-11-30 辛根塔有限公司 制备芳基酰胺的方法

Also Published As

Publication number Publication date
TW201204704A (en) 2012-02-01
JP2013525317A (ja) 2013-06-20
US20130035496A1 (en) 2013-02-07
EP2560959A1 (en) 2013-02-27
BR112012026631B1 (pt) 2017-07-25
EP2560959B1 (en) 2014-08-20
JP5684896B2 (ja) 2015-03-18
CN102906072A (zh) 2013-01-30
IL222398A (en) 2017-01-31
MX2012012005A (es) 2012-12-17
CN102906072B (zh) 2014-07-02
AR080922A1 (es) 2012-05-16
BR112012026631A2 (pt) 2015-09-15
WO2011131545A1 (en) 2011-10-27
TWI428325B (zh) 2014-03-01
US8519152B2 (en) 2013-08-27
ES2513540T3 (es) 2014-10-27

Similar Documents

Publication Publication Date Title
CO2017013709A2 (es) Lactamas bicíclicas.
EP2966706A3 (en) Organic electroluminescent materials and devices
AR092278A1 (es) Proceso de obtencion de derivados n-acilicos de bifenil-alanina e intermediarios relacionados
CR20140231A (es) Derivados de ácido benzotiazol-6-il acético y su uso para tratar una infección por vih
CU24410B1 (es) Benzimidazol-2-aminas como inhibidores de midh1
WO2016017919A3 (ko) 헤테로고리를 포함하는 축합 플루오렌 유도체
GT201200230A (es) Inhibidores del virus de la hepatitis c
CR20200276A (es) Sulfamoilarilamidas y su uso como medicamentos para el tratamientos de la hepatitis b (divisional exp. 2015-0059)
UA114087C2 (xx) Похідні піридину
EP2666768A3 (en) Condensed-cyclic compound and organic light-emitting diode comprising the same
WO2010114263A3 (en) Novel organic electroluminescent compounds and organic electroluminescent device using the same
UY33339A (es) Proceso para la preparación de amidas de ácido pirazol carboxílico
WO2014058232A3 (ko) 스파이로형 유기 재료 및 이를 이용한 유기 전기발광 소자
AR112787A2 (es) Compuestos 1,5-difenil-penta-1,4-dien-3-ona
WO2015150234A8 (en) Silyl-benzimidazolo[1,2-a]benzimidazole as host for organic light emitting diodes
WO2010114262A3 (en) Novel organic electroluminescent compounds and organic electroluminescent device using the same
UY33340A (es) Proceso para la preparación de amidas de ácido pirazol carboxílico
EP2772955A3 (en) Organic light emitting diode device
UY33341A (es) Proceso para la preparación de amidas de ácido pirazol carboxílico
MX2017008045A (es) Composiciones de polímero parcialmente fluorado curables.
AR085052A1 (es) Metodos para producir un compuesto profarmaco inhibidor de la union al vih e intermediarios
CY1118945T1 (el) Μεθοδος και ενδιαμεσα για την παρασκευη πρεγκαμπαλινης
AR117002A2 (es) Proceso para la preparación de inhibidores de quinasa c-fms
CY1114493T1 (el) Διαδικασια για την παρασκευη μιας ενωσης χρησιμης ως αναστολεα της tafia
WO2012093861A3 (ko) 유기 화합물 및 이를 이용한 유기 전계 발광 소자

Legal Events

Date Code Title Description
110 Patent granted

Effective date: 20210405