AR067084A1 - Dispersion solida que contiene revaprazan y procedimiento para la preparacion de la misma. composicion farmaceutica. - Google Patents
Dispersion solida que contiene revaprazan y procedimiento para la preparacion de la misma. composicion farmaceutica.Info
- Publication number
- AR067084A1 AR067084A1 ARP080102637A ARP080102637A AR067084A1 AR 067084 A1 AR067084 A1 AR 067084A1 AR P080102637 A ARP080102637 A AR P080102637A AR P080102637 A ARP080102637 A AR P080102637A AR 067084 A1 AR067084 A1 AR 067084A1
- Authority
- AR
- Argentina
- Prior art keywords
- solid dispersion
- pharmaceutical composition
- revapraze
- procedure
- preparation
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1635—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1617—Organic compounds, e.g. phospholipids, fats
- A61K9/1623—Sugars or sugar alcohols, e.g. lactose; Derivatives thereof; Homeopathic globules
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
Landscapes
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Inorganic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Una dispersion solida en la cual las partículas de revaprazán son modificadas en la superficie con un polímero soluble en agua, un sacárido soluble en agua, un tensioactivo, o una mezcla de los mismos, y un procedimiento para preparar la misma. La presente provee también una composicion farmacéutica que contiene la dispersion solida y un procedimiento para preparar la composicion farmacéutica. Reivindicacion 5: La dispersion solida de acuerdo con la reivindicacion 1, caracterizada porque las partículas de revaprazán son modificadas en la superficie con polivinilpirrolidona, éster de ácido graso de sacarosa y aceite de ricino hidrogenado o natural glicolado polioxietileno.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR20060132722 | 2006-12-22 | ||
KR1020070135270A KR100954828B1 (ko) | 2006-12-22 | 2007-12-21 | 레바프라잔 함유 고체분산체 및 그의 제조방법 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR067084A1 true AR067084A1 (es) | 2009-09-30 |
Family
ID=39562674
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP080102637A AR067084A1 (es) | 2006-12-22 | 2008-06-20 | Dispersion solida que contiene revaprazan y procedimiento para la preparacion de la misma. composicion farmaceutica. |
Country Status (20)
Country | Link |
---|---|
US (1) | US8663658B2 (es) |
EP (1) | EP2101737B1 (es) |
JP (1) | JP5484910B2 (es) |
KR (1) | KR100954828B1 (es) |
CN (1) | CN101600419B (es) |
AR (1) | AR067084A1 (es) |
AU (1) | AU2007339080B2 (es) |
BR (1) | BRPI0720472A2 (es) |
CA (1) | CA2673536A1 (es) |
ES (1) | ES2496166T3 (es) |
HK (1) | HK1138517A1 (es) |
MX (1) | MX2009006105A (es) |
MY (1) | MY146557A (es) |
PA (1) | PA8784701A1 (es) |
PE (1) | PE20090424A1 (es) |
RU (1) | RU2461382C2 (es) |
SA (1) | SA08290368B1 (es) |
TW (1) | TW200927124A (es) |
WO (1) | WO2008078922A1 (es) |
ZA (1) | ZA200905094B (es) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2673536A1 (en) | 2006-12-22 | 2008-07-03 | Yuhan Corporation | Revaprazan-containing solid dispersion and process for the preparation thereof |
CN101874775B (zh) * | 2010-05-31 | 2013-03-13 | 沈阳药科大学 | 盐酸瑞伐拉赞纳米混悬剂及其制备方法 |
KR101739816B1 (ko) * | 2010-12-01 | 2017-05-25 | 주식회사유한양행 | 레바프라잔 또는 그의 염을 함유하는 주사용 액제 조성물 또는 주사용 건조 분말 |
KR101739815B1 (ko) * | 2010-12-01 | 2017-05-26 | 주식회사유한양행 | 레바프라잔 또는 그의 염을 함유하는 주사용 액제 조성물 |
KR101730865B1 (ko) * | 2011-02-11 | 2017-04-27 | 주식회사유한양행 | 레바프라잔-함유 나노입자를 포함하는 경구투여용 약학 조성물 및 그의 제조방법 |
KR101739818B1 (ko) * | 2011-05-20 | 2017-05-26 | 주식회사유한양행 | 레바프라잔 또는 그의 염을 함유하는 현탁액 형태의 경구투여용 약학 조성물 |
KR101739820B1 (ko) * | 2012-03-28 | 2017-05-25 | 주식회사유한양행 | 레바프라잔 또는 그의 염을 함유하는 비수성 액체 형태의 경구투여용 약학 조성물 |
WO2015175505A1 (en) * | 2014-05-15 | 2015-11-19 | Lundbeck Llc | Tetrabenazine modified release formulation |
CN106456556A (zh) * | 2014-06-18 | 2017-02-22 | 豪夫迈·罗氏有限公司 | 包含非离子性表面活性剂的新型药物组合物 |
CN104825410A (zh) * | 2015-05-04 | 2015-08-12 | 海南海力制药有限公司 | 一种盐酸瑞伐拉赞片及其制备方法 |
CN105288636B (zh) * | 2015-12-11 | 2019-05-07 | 北京科莱博医药开发有限责任公司 | 增溶体系、固体分散体及药物制剂 |
WO2017106130A1 (en) * | 2015-12-16 | 2017-06-22 | Merck Sharp & Dohme Corp. | Process for preparing pharmaceutical compositions |
CN105687150B (zh) * | 2016-03-15 | 2019-12-10 | 常州市第四制药厂有限公司 | 一种盐酸瑞伐拉赞组合物及制备方法 |
CN106361721A (zh) * | 2016-08-31 | 2017-02-01 | 佛山市弘泰药物研发有限公司 | 一种盐酸瑞伐拉赞胶囊及其制备方法 |
PT110585B (pt) * | 2018-02-22 | 2021-04-22 | Hovione Farmaciencia Sa | Processo de produção contínua de partículas compreendendo secagem por atomização com preparação contínua da solução de atomização |
JPWO2020261619A1 (es) | 2019-06-26 | 2020-12-30 | ||
EP3989940A1 (en) | 2019-06-26 | 2022-05-04 | Ricoh Company, Ltd. | Instantly soluble particle and method for producing the same |
Family Cites Families (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH05255125A (ja) | 1992-02-29 | 1993-10-05 | Upjohn Co:The | 徐放性製剤およびその製法 |
KR0157075B1 (ko) * | 1994-08-13 | 1998-11-16 | 김태훈 | 신규의 피리미딘 유도체 및 그의 제조방법 |
ES2201112T3 (es) * | 1994-08-13 | 2004-03-16 | Yuhan Corporation | Nuevos derivados de pirimidina y procedimientos para su preparacion. |
EP0834314B1 (en) * | 1995-06-12 | 2003-01-15 | Ono Pharmaceutical Co., Ltd. | Granules containing pranlukast, process for producing the granules, and method of lowering cohesiveness of pranlukast |
US5955475A (en) * | 1997-06-30 | 1999-09-21 | Endo Pharmaceuticals Inc. | Process for manufacturing paroxetine solid dispersions |
IT1294760B1 (it) * | 1997-09-03 | 1999-04-12 | Jagotec Ag | Procedimento per la preparazione di compresse farmaceutiche in grado di cedere,secondo schemi predeterminabili, principi attivi poco |
EP1227797B1 (en) * | 1999-11-12 | 2005-01-12 | Abbott Laboratories | Solid dispersion pharmaceutical formulations |
AU782469B2 (en) * | 1999-12-23 | 2005-08-04 | Mayne Pharma International Pty Ltd | Improved pharmaceutical compositions for poorly soluble drugs |
HUP0303700A3 (en) * | 2000-07-17 | 2006-07-28 | Astellas Pharma Inc Chuo Ku | Pharmaceutical composition improved in peroral absorbability |
US8206741B2 (en) * | 2001-06-01 | 2012-06-26 | Pozen Inc. | Pharmaceutical compositions for the coordinated delivery of NSAIDs |
EP1275377B1 (en) * | 2001-07-11 | 2003-06-18 | Apr Applied Pharma Research S.A. | Granulates containing liposoluble substances and process of preparation thereof |
KR20040081123A (ko) * | 2002-01-11 | 2004-09-20 | 다케다 야쿠힌 고교 가부시키가이샤 | 쿠마린 유도체, 이의 제조 방법 및 용도 |
ES2280835T3 (es) * | 2002-12-19 | 2007-09-16 | Pharmacia Corporation | Formulacion no higroscopica que comprende un farmaco higroscopico. |
US20050096365A1 (en) * | 2003-11-03 | 2005-05-05 | David Fikstad | Pharmaceutical compositions with synchronized solubilizer release |
CN100563658C (zh) * | 2003-11-14 | 2009-12-02 | 味之素株式会社 | 苯丙氨酸衍生物的固体分散体或固体分散体医药制剂 |
WO2006046623A1 (ja) * | 2004-10-25 | 2006-05-04 | Japan Tobacco Inc. | 溶解性及び安定性の改善された固形製剤及びその製造方法 |
US20060165797A1 (en) | 2005-01-12 | 2006-07-27 | Pozen Inc. | Dosage form for treating gastrointestinal disorders |
WO2007070164A1 (en) * | 2005-10-19 | 2007-06-21 | The Curators Of The University Of Missouri | Pharmaceutical composition comprising a proton pump inhibitor, a buffering agent and an anti-h. pylori active substance and methods of using same |
US7776873B2 (en) | 2005-12-01 | 2010-08-17 | Yuhan Corporation | Method for treating damage to gastric mucosa |
CA2673536A1 (en) | 2006-12-22 | 2008-07-03 | Yuhan Corporation | Revaprazan-containing solid dispersion and process for the preparation thereof |
-
2007
- 2007-12-21 CA CA002673536A patent/CA2673536A1/en not_active Abandoned
- 2007-12-21 RU RU2009128206/15A patent/RU2461382C2/ru not_active IP Right Cessation
- 2007-12-21 JP JP2009542655A patent/JP5484910B2/ja not_active Expired - Fee Related
- 2007-12-21 US US12/520,037 patent/US8663658B2/en not_active Expired - Fee Related
- 2007-12-21 CN CN2007800475422A patent/CN101600419B/zh active Active
- 2007-12-21 WO PCT/KR2007/006738 patent/WO2008078922A1/en active Application Filing
- 2007-12-21 AU AU2007339080A patent/AU2007339080B2/en not_active Ceased
- 2007-12-21 EP EP07851703.4A patent/EP2101737B1/en not_active Not-in-force
- 2007-12-21 BR BRPI0720472-8A patent/BRPI0720472A2/pt not_active IP Right Cessation
- 2007-12-21 ES ES07851703.4T patent/ES2496166T3/es active Active
- 2007-12-21 KR KR1020070135270A patent/KR100954828B1/ko active IP Right Grant
- 2007-12-21 ZA ZA200905094A patent/ZA200905094B/xx unknown
- 2007-12-21 MX MX2009006105A patent/MX2009006105A/es unknown
- 2007-12-21 MY MYPI20092582A patent/MY146557A/en unknown
-
2008
- 2008-06-13 PA PA20088784701A patent/PA8784701A1/es unknown
- 2008-06-18 SA SA8290368A patent/SA08290368B1/ar unknown
- 2008-06-20 AR ARP080102637A patent/AR067084A1/es not_active Application Discontinuation
- 2008-06-20 TW TW097123092A patent/TW200927124A/zh unknown
- 2008-06-20 PE PE2008001062A patent/PE20090424A1/es not_active Application Discontinuation
-
2010
- 2010-05-28 HK HK10105215.6A patent/HK1138517A1/xx unknown
Also Published As
Publication number | Publication date |
---|---|
AU2007339080B2 (en) | 2012-09-27 |
US8663658B2 (en) | 2014-03-04 |
BRPI0720472A2 (pt) | 2014-01-14 |
KR20080059083A (ko) | 2008-06-26 |
CA2673536A1 (en) | 2008-07-03 |
JP2010513474A (ja) | 2010-04-30 |
WO2008078922A1 (en) | 2008-07-03 |
EP2101737A4 (en) | 2013-05-01 |
HK1138517A1 (en) | 2010-08-27 |
CN101600419A (zh) | 2009-12-09 |
US20100041688A1 (en) | 2010-02-18 |
JP5484910B2 (ja) | 2014-05-07 |
RU2009128206A (ru) | 2011-01-27 |
KR100954828B1 (ko) | 2010-04-27 |
PA8784701A1 (es) | 2009-07-23 |
EP2101737A1 (en) | 2009-09-23 |
CN101600419B (zh) | 2012-05-09 |
PE20090424A1 (es) | 2009-05-15 |
RU2461382C2 (ru) | 2012-09-20 |
ES2496166T3 (es) | 2014-09-18 |
ZA200905094B (en) | 2010-09-29 |
SA08290368B1 (ar) | 2011-10-08 |
MY146557A (en) | 2012-08-30 |
TW200927124A (en) | 2009-07-01 |
MX2009006105A (es) | 2009-06-18 |
EP2101737B1 (en) | 2014-06-18 |
AU2007339080A1 (en) | 2008-07-03 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Abandonment or withdrawal |