AR054626A1 - Derivados de quinolina como agentes antibacterianos - Google Patents

Derivados de quinolina como agentes antibacterianos

Info

Publication number
AR054626A1
AR054626A1 ARP060102787A ARP060102787A AR054626A1 AR 054626 A1 AR054626 A1 AR 054626A1 AR P060102787 A ARP060102787 A AR P060102787A AR P060102787 A ARP060102787 A AR P060102787A AR 054626 A1 AR054626 A1 AR 054626A1
Authority
AR
Argentina
Prior art keywords
alkyl
alkyloxy
hydroxy
hydrocarbon radical
halo
Prior art date
Application number
ARP060102787A
Other languages
English (en)
Spanish (es)
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34940244&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR054626(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of AR054626A1 publication Critical patent/AR054626A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/04Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to the ring carbon atoms
    • C07D215/06Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to the ring carbon atoms having only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to the ring nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/12Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • C07D215/22Oxygen atoms attached in position 2 or 4
    • C07D215/227Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ARP060102787A 2005-06-28 2006-06-28 Derivados de quinolina como agentes antibacterianos AR054626A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05105762 2005-06-28

Publications (1)

Publication Number Publication Date
AR054626A1 true AR054626A1 (es) 2007-07-04

Family

ID=34940244

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP060102787A AR054626A1 (es) 2005-06-28 2006-06-28 Derivados de quinolina como agentes antibacterianos

Country Status (31)

Country Link
US (1) US8841321B2 (enExample)
EP (1) EP1898914B1 (enExample)
JP (1) JP5193858B2 (enExample)
KR (1) KR101329585B1 (enExample)
CN (1) CN101247811B (enExample)
AP (1) AP2386A (enExample)
AR (1) AR054626A1 (enExample)
AU (1) AU2006263883B2 (enExample)
BR (1) BRPI0612498A8 (enExample)
CA (1) CA2612619C (enExample)
CY (1) CY1113579T1 (enExample)
DK (1) DK1898914T3 (enExample)
EA (1) EA014423B1 (enExample)
ES (1) ES2393203T3 (enExample)
HR (1) HRP20120912T1 (enExample)
IL (1) IL188393A0 (enExample)
JO (1) JO2752B1 (enExample)
ME (1) ME01484B (enExample)
MX (1) MX2008000081A (enExample)
MY (1) MY153291A (enExample)
NO (1) NO342701B1 (enExample)
NZ (1) NZ564379A (enExample)
PA (1) PA8683801A1 (enExample)
PL (1) PL1898914T3 (enExample)
PT (1) PT1898914E (enExample)
RS (1) RS52517B (enExample)
SI (1) SI1898914T1 (enExample)
TW (1) TWI387457B (enExample)
UA (1) UA92175C2 (enExample)
WO (1) WO2007000435A1 (enExample)
ZA (1) ZA200711165B (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO2970B1 (en) 2006-12-06 2016-03-15 جانسين فارماسوتيكا ان. في Quinoline antibacterial derivatives
JO2683B1 (en) * 2006-12-06 2013-03-03 جانسين فارماسوتيكا ان. في Quinoline antibacterial derivatives
CN104254527B (zh) 2012-04-27 2017-05-31 詹森药业有限公司 抗菌的喹啉衍生物
AU2013254670B2 (en) 2012-04-27 2017-03-30 Janssen Pharmaceutica Nv Antibacterial quinoline derivatives
EP3237383B1 (en) 2014-12-23 2019-12-04 Albemarle Corporation One-step process for the synthesis of alkylated metyrapone analogs
CN106928139B (zh) * 2017-05-08 2019-06-25 福建省微生物研究所 一种贝达喹啉杂质的合成方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19937116A1 (de) * 1999-08-06 2001-02-08 Bayer Ag Moxifloxacin Kochsalzformulierung
DK2301544T3 (da) 2002-07-25 2013-01-02 Janssen Pharmaceutica Nv Quinolinderivater som mellemprodukter til mykobakterielle inhibitorer
SI1675852T1 (sl) 2003-09-22 2009-06-30 Janssen Pharmaceutica Nv 7-amino alkilidenil-heterociklični kinoloni in naftiridoni
EP1753427B1 (en) * 2004-05-28 2008-04-02 Janssen Pharmaceutica N.V. Use of substituted quinoline derivatives for the treatment of drug resistant mycobacterial diseases
EE05394B1 (et) * 2004-12-24 2011-04-15 Janssen Pharmaceutica N.V. Kinoliinihendid kasutamiseks latentse tuberkuloosi ravis
DK1898909T3 (en) 2005-06-28 2017-02-06 Janssen Pharmaceutica Nv QUINOLIN DERIVATIVES AS ANTIBACTERIAL AGENTS

Also Published As

Publication number Publication date
CY1113579T1 (el) 2016-06-22
SI1898914T1 (sl) 2013-01-31
HRP20120912T1 (hr) 2012-12-31
PA8683801A1 (es) 2007-01-17
EA014423B1 (ru) 2010-12-30
US20100048585A1 (en) 2010-02-25
BRPI0612498A8 (pt) 2018-01-02
KR20080021156A (ko) 2008-03-06
IL188393A0 (en) 2008-08-07
US8841321B2 (en) 2014-09-23
ME01484B (me) 2014-04-20
MY153291A (en) 2015-01-29
NZ564379A (en) 2010-11-26
ES2393203T3 (es) 2012-12-19
KR101329585B1 (ko) 2013-11-15
JP2008543964A (ja) 2008-12-04
AU2006263883B2 (en) 2012-12-13
TW200740437A (en) 2007-11-01
ZA200711165B (en) 2011-05-25
JP5193858B2 (ja) 2013-05-08
CA2612619C (en) 2015-12-01
AP2386A (en) 2012-03-23
RS52517B (sr) 2013-04-30
DK1898914T3 (da) 2012-11-26
MX2008000081A (es) 2008-03-24
EP1898914A1 (en) 2008-03-19
NO20080501L (no) 2008-02-28
BRPI0612498A2 (pt) 2010-11-23
PT1898914E (pt) 2012-11-20
UA92175C2 (ru) 2010-10-11
EP1898914B1 (en) 2012-08-15
CN101247811B (zh) 2013-01-02
CA2612619A1 (en) 2007-01-04
NO342701B1 (no) 2018-07-09
HK1122730A1 (en) 2009-05-29
EA200800154A1 (ru) 2008-10-30
WO2007000435A1 (en) 2007-01-04
CN101247811A (zh) 2008-08-20
PL1898914T3 (pl) 2013-01-31
JO2752B1 (en) 2014-03-15
TWI387457B (zh) 2013-03-01
AU2006263883A1 (en) 2007-01-04

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