AR046966A1 - Esteroides con un perfil androgenico y progestagenico mixto - Google Patents

Esteroides con un perfil androgenico y progestagenico mixto

Info

Publication number
AR046966A1
AR046966A1 ARP040104787A ARP040104787A AR046966A1 AR 046966 A1 AR046966 A1 AR 046966A1 AR P040104787 A ARP040104787 A AR P040104787A AR P040104787 A ARP040104787 A AR P040104787A AR 046966 A1 AR046966 A1 AR 046966A1
Authority
AR
Argentina
Prior art keywords
steroids
progestagenic
profile
androgenic
mixed
Prior art date
Application number
ARP040104787A
Other languages
English (en)
Inventor
Der Louw Jaap Van
Dirk Leysen
Arij Jan Grootenhuis
Gooijer Marcel Evert De
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Publication of AR046966A1 publication Critical patent/AR046966A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • C07J63/008—Expansion of ring D by one atom, e.g. D homo steroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16—Masculine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26—Androgens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/34—Gestagens

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

La presente se refiere a esteroides con un perfil androgénico y progestagénico mixto, composicion farmacéutica que los comprende y usos. Reivindicacion 1: Un compuesto de formula (1) donde: R1 es O, o NOR con R siendo H, alquil C1-6 o acil C1-6, R2 es metil o etil, y R3 es H o acil C1-15.
ARP040104787A 2003-12-22 2004-12-20 Esteroides con un perfil androgenico y progestagenico mixto AR046966A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP03104898 2003-12-22

Publications (1)

Publication Number Publication Date
AR046966A1 true AR046966A1 (es) 2006-01-04

Family

ID=34707282

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP040104787A AR046966A1 (es) 2003-12-22 2004-12-20 Esteroides con un perfil androgenico y progestagenico mixto

Country Status (30)

Country Link
US (1) US7582622B2 (es)
EP (1) EP1720895B1 (es)
JP (1) JP2007515455A (es)
KR (1) KR20060123484A (es)
CN (1) CN1898258B (es)
AR (1) AR046966A1 (es)
AT (1) ATE373674T1 (es)
AU (1) AU2004303524A1 (es)
BR (1) BRPI0417781A (es)
CA (1) CA2549148A1 (es)
CY (1) CY1106935T1 (es)
DE (1) DE602004009107T2 (es)
DK (1) DK1720895T3 (es)
EC (1) ECSP066666A (es)
ES (1) ES2294569T3 (es)
HR (1) HRP20070492T3 (es)
IL (1) IL175890A0 (es)
IS (1) IS8488A (es)
MX (1) MXPA06007195A (es)
NO (1) NO20062585L (es)
NZ (1) NZ547772A (es)
PE (1) PE20050677A1 (es)
PL (1) PL1720895T3 (es)
PT (1) PT1720895E (es)
RU (1) RU2357972C2 (es)
SI (1) SI1720895T1 (es)
TW (1) TW200521134A (es)
UA (1) UA84037C2 (es)
WO (1) WO2005061528A2 (es)
ZA (1) ZA200604976B (es)

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3959322A (en) * 1960-09-22 1976-05-25 Herchel Smith Synthesis of 13-alkyl-gon-4-ones
FR1434172A (fr) 1963-12-24 1966-04-08 Ciba Geigy Procédé de préparation de nouvelles oestrones substituées
NL125069C (es) * 1963-12-24
US4412993A (en) * 1980-01-25 1983-11-01 The Upjohn Company Method of treating pseudopregnancy, galactorrhea and mastitis in mammals
US4788218A (en) * 1984-05-21 1988-11-29 Sri International 17 a β-hydroxy-7 α-methyl-d-homo-19-norandrost-4,16-diene-3-one and the 17-esters thereof: methods of preparation and uses
EP0182808A1 (en) * 1984-05-21 1986-06-04 Sri International 17 a?$g(b)-HYDROXY-7$g(a)-METHYL-D-HOMO-19-NORANDROST-4,16-DIENE-3-ONE AND THE 17-ESTERS THEREOF: METHODS OF PREPARATION AND USES
TR200003743T2 (tr) 1998-06-19 2001-07-23 Akzo Nobel N.V. Testosteron türevi.
WO2000053619A1 (en) 1999-03-08 2000-09-14 Akzo Nobel N.V. 14.beta., 17-alpha-hydroxymethylandrostane derivatives as androgens
EP1212345B1 (en) 1999-04-06 2003-08-06 Akzo Nobel N.V. Orally active 7-alpha-alkyl androgens
TW548277B (en) 1999-07-16 2003-08-21 Akzo Nobel Nv Orally active androgens

Also Published As

Publication number Publication date
HRP20070492T3 (en) 2007-12-31
DE602004009107D1 (de) 2007-10-31
ES2294569T3 (es) 2008-04-01
BRPI0417781A (pt) 2007-03-20
RU2006126632A (ru) 2008-01-27
CN1898258A (zh) 2007-01-17
ECSP066666A (es) 2006-10-25
MXPA06007195A (es) 2006-09-04
ATE373674T1 (de) 2007-10-15
NO20062585L (no) 2006-09-20
IL175890A0 (en) 2006-10-05
TW200521134A (en) 2005-07-01
CY1106935T1 (el) 2012-09-26
PL1720895T3 (pl) 2008-02-29
WO2005061528A2 (en) 2005-07-07
US7582622B2 (en) 2009-09-01
EP1720895B1 (en) 2007-09-19
SI1720895T1 (sl) 2007-12-31
CN1898258B (zh) 2010-06-16
IS8488A (is) 2006-05-26
KR20060123484A (ko) 2006-12-01
PT1720895E (pt) 2007-10-09
PE20050677A1 (es) 2005-10-04
US20070155836A1 (en) 2007-07-05
RU2357972C2 (ru) 2009-06-10
DE602004009107T2 (de) 2008-06-19
UA84037C2 (ru) 2008-09-10
ZA200604976B (en) 2007-04-25
EP1720895A2 (en) 2006-11-15
WO2005061528A3 (en) 2005-09-09
AU2004303524A1 (en) 2005-07-07
DK1720895T3 (da) 2008-01-14
NZ547772A (en) 2009-01-31
JP2007515455A (ja) 2007-06-14
CA2549148A1 (en) 2005-07-07

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