AR034119A1 - Compuestos de 5-alquilpirido pirimidinas, composicion farmaceutica, uso para prepararla y metodo para inhibir cinasas con dichos compuestos - Google Patents

Compuestos de 5-alquilpirido pirimidinas, composicion farmaceutica, uso para prepararla y metodo para inhibir cinasas con dichos compuestos

Info

Publication number
AR034119A1
AR034119A1 ARP010101039A ARP010101039A AR034119A1 AR 034119 A1 AR034119 A1 AR 034119A1 AR P010101039 A ARP010101039 A AR P010101039A AR P010101039 A ARP010101039 A AR P010101039A AR 034119 A1 AR034119 A1 AR 034119A1
Authority
AR
Argentina
Prior art keywords
independently selected
lower alkyl
halogen
trifluoromethyl
carbocyclic group
Prior art date
Application number
ARP010101039A
Other languages
English (en)
Spanish (es)
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of AR034119A1 publication Critical patent/AR034119A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
ARP010101039A 2000-03-06 2001-03-05 Compuestos de 5-alquilpirido pirimidinas, composicion farmaceutica, uso para prepararla y metodo para inhibir cinasas con dichos compuestos AR034119A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US18712400P 2000-03-06 2000-03-06

Publications (1)

Publication Number Publication Date
AR034119A1 true AR034119A1 (es) 2004-02-04

Family

ID=22687699

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP010101039A AR034119A1 (es) 2000-03-06 2001-03-05 Compuestos de 5-alquilpirido pirimidinas, composicion farmaceutica, uso para prepararla y metodo para inhibir cinasas con dichos compuestos

Country Status (36)

Country Link
EP (1) EP1268476A1 (ja)
JP (1) JP2003528101A (ja)
KR (1) KR20020075805A (ja)
CN (1) CN1422268A (ja)
AP (1) AP2002002643A0 (ja)
AR (1) AR034119A1 (ja)
AU (1) AU2001233028A1 (ja)
BG (1) BG107161A (ja)
BR (1) BR0109056A (ja)
CA (1) CA2401368A1 (ja)
CO (1) CO5280200A1 (ja)
CR (1) CR6736A (ja)
CZ (1) CZ20022929A3 (ja)
DZ (1) DZ3308A1 (ja)
EA (1) EA200200802A1 (ja)
EE (1) EE200200506A (ja)
GT (1) GT200100037A (ja)
HN (1) HN2001000040A (ja)
HR (1) HRP20020798A2 (ja)
HU (1) HUP0300136A2 (ja)
IL (1) IL151480A0 (ja)
IS (1) IS6524A (ja)
MA (1) MA26881A1 (ja)
MX (1) MXPA02008535A (ja)
NO (1) NO20024235L (ja)
NZ (1) NZ520962A (ja)
OA (1) OA12227A (ja)
PA (1) PA8513201A1 (ja)
PE (1) PE20011177A1 (ja)
PL (1) PL358271A1 (ja)
SK (1) SK12472002A3 (ja)
SV (1) SV2001000338A (ja)
TN (1) TNSN01036A1 (ja)
WO (1) WO2001070741A1 (ja)
YU (1) YU66502A (ja)
ZA (1) ZA200207110B (ja)

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EP1333833B1 (en) 2000-10-23 2011-08-24 GlaxoSmithKline LLC Novel trisubstituted-8H-pyrido[2,3-d]pyrimidin-7-one compound for the treatment of CSBP/p38 kinase mediated diseases
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US20030105115A1 (en) * 2001-06-21 2003-06-05 Metcalf Chester A. Novel pyridopyrimidines and uses thereof
US20030100572A1 (en) * 2001-06-21 2003-05-29 Ariad Pharmaceuticals,Inc. Novel pyridopyrimidones and uses thereof
GEP20063909B (en) * 2002-01-22 2006-08-25 Warner Lambert Co 2-(PYRIDIN-2-YLAMINO)-PYRIDO[2,3d] PYRIMIDIN-7-ONES
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Also Published As

Publication number Publication date
EA200200802A1 (ru) 2003-02-27
AU2001233028A1 (en) 2001-10-03
KR20020075805A (ko) 2002-10-05
BG107161A (en) 2003-06-30
IS6524A (is) 2002-08-23
HN2001000040A (es) 2001-09-06
HUP0300136A2 (en) 2003-05-28
CR6736A (es) 2004-03-10
IL151480A0 (en) 2003-04-10
GT200100037A (es) 2002-03-04
MXPA02008535A (es) 2002-12-13
TNSN01036A1 (en) 2005-11-10
MA26881A1 (fr) 2004-12-20
CN1422268A (zh) 2003-06-04
NO20024235D0 (no) 2002-09-05
PA8513201A1 (es) 2003-06-30
YU66502A (sh) 2005-09-19
SV2001000338A (es) 2001-11-30
EP1268476A1 (en) 2003-01-02
JP2003528101A (ja) 2003-09-24
AP2002002643A0 (en) 2002-12-31
NO20024235L (no) 2002-11-05
EE200200506A (et) 2004-02-16
CA2401368A1 (en) 2001-09-27
BR0109056A (pt) 2003-06-03
CZ20022929A3 (cs) 2003-02-12
HRP20020798A2 (en) 2004-02-29
DZ3308A1 (fr) 2001-09-27
NZ520962A (en) 2003-09-26
WO2001070741A1 (en) 2001-09-27
OA12227A (en) 2004-03-18
CO5280200A1 (es) 2003-05-30
PE20011177A1 (es) 2001-11-23
SK12472002A3 (sk) 2003-04-01
ZA200207110B (en) 2003-12-04
PL358271A1 (en) 2004-08-09

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