AR026209A1 - Compuestos monociclicos basicos con accion nk-2 antagonista, procesos de fabricacion y formulas que los contienen - Google Patents

Compuestos monociclicos basicos con accion nk-2 antagonista, procesos de fabricacion y formulas que los contienen

Info

Publication number
AR026209A1
AR026209A1 ARP000105566A ARP000105566A AR026209A1 AR 026209 A1 AR026209 A1 AR 026209A1 AR P000105566 A ARP000105566 A AR P000105566A AR P000105566 A ARP000105566 A AR P000105566A AR 026209 A1 AR026209 A1 AR 026209A1
Authority
AR
Argentina
Prior art keywords
compounds
basic
manufacturing processes
monociclic
formulas containing
Prior art date
Application number
ARP000105566A
Other languages
English (en)
Original Assignee
Menarini Ricerche Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Menarini Ricerche Spa filed Critical Menarini Ricerche Spa
Publication of AR026209A1 publication Critical patent/AR026209A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/10—Drugs for disorders of the urinary system of the bladder
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)

Abstract

Se describen compuestos monocíclicos básicos de formula (1) utiles como antagonistas del receptor NK-2, se describen además métodos para la produccion dedichos compuestos y formulaciones que los contienen. Compuestos monocícliclos básicos con accion NK-2, antagonista, procesos de fabricacion y formulas que loscontienen.
ARP000105566A 1999-10-21 2000-10-23 Compuestos monociclicos basicos con accion nk-2 antagonista, procesos de fabricacion y formulas que los contienen AR026209A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT1999FI000217A IT1307809B1 (it) 1999-10-21 1999-10-21 Composti monociclici basici ad azione nk-2 antagonista, processi difabbricazione e formulazioni che li contengono.

Publications (1)

Publication Number Publication Date
AR026209A1 true AR026209A1 (es) 2003-01-29

Family

ID=11353095

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP000105566A AR026209A1 (es) 1999-10-21 2000-10-23 Compuestos monociclicos basicos con accion nk-2 antagonista, procesos de fabricacion y formulas que los contienen

Country Status (13)

Country Link
US (1) US7015196B1 (es)
EP (1) EP1224210B1 (es)
JP (1) JP2003512387A (es)
CN (1) CN1199987C (es)
AR (1) AR026209A1 (es)
AT (1) ATE256697T1 (es)
AU (1) AU7919900A (es)
CA (1) CA2388315A1 (es)
DE (1) DE60007345T2 (es)
ES (1) ES2211628T3 (es)
IT (1) IT1307809B1 (es)
PT (1) PT1224210E (es)
WO (1) WO2001029066A2 (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2258642T3 (es) 2001-07-02 2006-09-01 Astrazeneca Ab Derivados de piperidina utiles como moduladores de la actividad del receptor de quimiocina.
GB0120461D0 (en) 2001-08-22 2001-10-17 Astrazeneca Ab Novel compounds
GB0122503D0 (en) 2001-09-18 2001-11-07 Astrazeneca Ab Chemical compounds
MY130373A (en) 2001-10-29 2007-06-29 Malesci Sas Linear basic compounds having nk-2 antagonist activity and formulations thereof
SE0200843D0 (sv) 2002-03-19 2002-03-19 Astrazeneca Ab Chemical compounds
SE0200844D0 (sv) 2002-03-19 2002-03-19 Astrazeneca Ab Chemical compounds
SE0300957D0 (sv) 2003-04-01 2003-04-01 Astrazeneca Ab Chemical compounds
ITFI20040221A1 (it) * 2004-10-27 2005-01-27 Guidotti & C Spa Composizioni farmaceutiche a base di nk2 antagonisti per uso pediatrico
EP2402316A1 (en) 2005-07-21 2012-01-04 AstraZeneca AB (Publ) Piperidine derivatives
WO2007076875A2 (en) * 2006-01-06 2007-07-12 Aarhus Universitet Compounds acting on the serotonin transporter
UY38485A (es) 2018-11-27 2020-06-30 Novartis Ag Compuestos tetrámeros cíclicos como inhibidores de proproteína convertasa subtilisina/kexina tipo 9 (pcsk9), método de tratamiento, uso y su preparación

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8000470A (nl) 1980-01-25 1981-01-30 Akzo Nv Zonnecollector met een vloeistof opnemende laag.
US5187156A (en) * 1988-03-16 1993-02-16 Fujisawa Pharmaceutical Co., Ltd. Peptide compounds, processes for preparation thereof and pharmaceutical composition comprising the same
EP0606222A1 (en) 1991-08-08 1994-07-20 A. Menarini Industrie Farmaceutiche Riunite S.R.L. Cyclic hexapeptides as tachyquinin antagonists, their preparation and pharmaceutical compositions thereof
IT1262902B (it) 1992-04-15 1996-07-22 Menarini Farma Ind Composti triciclici antagonisti delle tachichinine, loro preparazione e loro uso in composizioni farmaceutiche.
DE19541283A1 (de) * 1995-11-06 1997-05-07 Boehringer Ingelheim Kg Neue Aminosäurederivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen
IT1291776B1 (it) 1997-02-07 1999-01-21 Menarini Ricerche Spa Composti monociclici a quattro residui bifunzionali, aventi azione nk-2 antagonista
IT1304888B1 (it) 1998-08-05 2001-04-05 Menarini Ricerche Spa Composti monociclici ad azione nk-2 antagonista e formulazioni che licontengono

Also Published As

Publication number Publication date
ES2211628T3 (es) 2004-07-16
EP1224210A2 (en) 2002-07-24
IT1307809B1 (it) 2001-11-19
ITFI990217A0 (it) 1999-10-21
US7015196B1 (en) 2006-03-21
WO2001029066A2 (en) 2001-04-26
CA2388315A1 (en) 2001-04-26
ATE256697T1 (de) 2004-01-15
CN1382154A (zh) 2002-11-27
AU7919900A (en) 2001-04-30
DE60007345D1 (de) 2004-01-29
CN1199987C (zh) 2005-05-04
EP1224210B1 (en) 2003-12-17
PT1224210E (pt) 2004-04-30
WO2001029066A3 (en) 2001-11-01
ITFI990217A1 (it) 2001-04-21
DE60007345T2 (de) 2004-11-11
JP2003512387A (ja) 2003-04-02

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