ATE256697T1 - Basische monocyclische verbindungen mit nk-2 antagonistischer wirkung, verfahren zu ihrer herstellung, und sie enthaltende mittel - Google Patents
Basische monocyclische verbindungen mit nk-2 antagonistischer wirkung, verfahren zu ihrer herstellung, und sie enthaltende mittelInfo
- Publication number
- ATE256697T1 ATE256697T1 AT00969509T AT00969509T ATE256697T1 AT E256697 T1 ATE256697 T1 AT E256697T1 AT 00969509 T AT00969509 T AT 00969509T AT 00969509 T AT00969509 T AT 00969509T AT E256697 T1 ATE256697 T1 AT E256697T1
- Authority
- AT
- Austria
- Prior art keywords
- production
- agents containing
- antagonistic action
- monocyclic compounds
- basic
- Prior art date
Links
- 230000003042 antagnostic effect Effects 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- Urology & Nephrology (AREA)
- Pulmonology (AREA)
- Biochemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT1999FI000217A IT1307809B1 (it) | 1999-10-21 | 1999-10-21 | Composti monociclici basici ad azione nk-2 antagonista, processi difabbricazione e formulazioni che li contengono. |
| PCT/EP2000/010181 WO2001029066A2 (en) | 1999-10-21 | 2000-10-17 | Basic monocyclic compounds having nk2 antagonist action, processes for their preparation, and formulations containing them |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE256697T1 true ATE256697T1 (de) | 2004-01-15 |
Family
ID=11353095
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT00969509T ATE256697T1 (de) | 1999-10-21 | 2000-10-17 | Basische monocyclische verbindungen mit nk-2 antagonistischer wirkung, verfahren zu ihrer herstellung, und sie enthaltende mittel |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US7015196B1 (de) |
| EP (1) | EP1224210B1 (de) |
| JP (1) | JP2003512387A (de) |
| CN (1) | CN1199987C (de) |
| AR (1) | AR026209A1 (de) |
| AT (1) | ATE256697T1 (de) |
| AU (1) | AU7919900A (de) |
| CA (1) | CA2388315A1 (de) |
| DE (1) | DE60007345T2 (de) |
| ES (1) | ES2211628T3 (de) |
| IT (1) | IT1307809B1 (de) |
| PT (1) | PT1224210E (de) |
| WO (1) | WO2001029066A2 (de) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL159256A0 (en) | 2001-07-02 | 2004-06-01 | Astrazeneca Ab | Piperidine derivatives useful as modulators of chemokine receptor activity |
| GB0120461D0 (en) | 2001-08-22 | 2001-10-17 | Astrazeneca Ab | Novel compounds |
| GB0122503D0 (en) | 2001-09-18 | 2001-11-07 | Astrazeneca Ab | Chemical compounds |
| MY130373A (en) | 2001-10-29 | 2007-06-29 | Malesci Sas | Linear basic compounds having nk-2 antagonist activity and formulations thereof |
| SE0200844D0 (sv) | 2002-03-19 | 2002-03-19 | Astrazeneca Ab | Chemical compounds |
| SE0200843D0 (sv) * | 2002-03-19 | 2002-03-19 | Astrazeneca Ab | Chemical compounds |
| SE0300957D0 (sv) | 2003-04-01 | 2003-04-01 | Astrazeneca Ab | Chemical compounds |
| ITFI20040221A1 (it) * | 2004-10-27 | 2005-01-27 | Guidotti & C Spa | Composizioni farmaceutiche a base di nk2 antagonisti per uso pediatrico |
| CA2615650A1 (en) | 2005-07-21 | 2007-01-25 | Astrazeneca Ab | Novel piperidine derivatives |
| US20100048713A1 (en) * | 2006-01-06 | 2010-02-25 | Aarhus Universitet | Compounds acting on the serotonin transporter |
| UY38485A (es) | 2018-11-27 | 2020-06-30 | Novartis Ag | Compuestos tetrámeros cíclicos como inhibidores de proproteína convertasa subtilisina/kexina tipo 9 (pcsk9), método de tratamiento, uso y su preparación |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL8000470A (nl) | 1980-01-25 | 1981-01-30 | Akzo Nv | Zonnecollector met een vloeistof opnemende laag. |
| US5187156A (en) * | 1988-03-16 | 1993-02-16 | Fujisawa Pharmaceutical Co., Ltd. | Peptide compounds, processes for preparation thereof and pharmaceutical composition comprising the same |
| JPH06509571A (ja) | 1991-08-08 | 1994-10-27 | エイ・メナリニ・インダストリー・ファーマシューティケ・リウニテ・エスアールエル | タキキニン拮抗薬としての環状ヘキサペプチドの製法およびその薬学的化合物 |
| IT1262902B (it) | 1992-04-15 | 1996-07-22 | Menarini Farma Ind | Composti triciclici antagonisti delle tachichinine, loro preparazione e loro uso in composizioni farmaceutiche. |
| DE19541283A1 (de) * | 1995-11-06 | 1997-05-07 | Boehringer Ingelheim Kg | Neue Aminosäurederivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen |
| IT1291776B1 (it) | 1997-02-07 | 1999-01-21 | Menarini Ricerche Spa | Composti monociclici a quattro residui bifunzionali, aventi azione nk-2 antagonista |
| IT1304888B1 (it) | 1998-08-05 | 2001-04-05 | Menarini Ricerche Spa | Composti monociclici ad azione nk-2 antagonista e formulazioni che licontengono |
-
1999
- 1999-10-21 IT IT1999FI000217A patent/IT1307809B1/it active
-
2000
- 2000-10-17 DE DE60007345T patent/DE60007345T2/de not_active Expired - Fee Related
- 2000-10-17 AU AU79199/00A patent/AU7919900A/en not_active Abandoned
- 2000-10-17 JP JP2001531864A patent/JP2003512387A/ja active Pending
- 2000-10-17 CA CA002388315A patent/CA2388315A1/en not_active Abandoned
- 2000-10-17 EP EP00969509A patent/EP1224210B1/de not_active Expired - Lifetime
- 2000-10-17 PT PT00969509T patent/PT1224210E/pt unknown
- 2000-10-17 US US10/111,430 patent/US7015196B1/en not_active Expired - Fee Related
- 2000-10-17 AT AT00969509T patent/ATE256697T1/de not_active IP Right Cessation
- 2000-10-17 WO PCT/EP2000/010181 patent/WO2001029066A2/en active IP Right Grant
- 2000-10-17 ES ES00969509T patent/ES2211628T3/es not_active Expired - Lifetime
- 2000-10-17 CN CNB008145679A patent/CN1199987C/zh not_active Expired - Fee Related
- 2000-10-23 AR ARP000105566A patent/AR026209A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2001029066A3 (en) | 2001-11-01 |
| ES2211628T3 (es) | 2004-07-16 |
| ITFI990217A1 (it) | 2001-04-21 |
| AU7919900A (en) | 2001-04-30 |
| IT1307809B1 (it) | 2001-11-19 |
| JP2003512387A (ja) | 2003-04-02 |
| CN1382154A (zh) | 2002-11-27 |
| ITFI990217A0 (it) | 1999-10-21 |
| EP1224210B1 (de) | 2003-12-17 |
| CN1199987C (zh) | 2005-05-04 |
| PT1224210E (pt) | 2004-04-30 |
| US7015196B1 (en) | 2006-03-21 |
| WO2001029066A2 (en) | 2001-04-26 |
| CA2388315A1 (en) | 2001-04-26 |
| AR026209A1 (es) | 2003-01-29 |
| DE60007345D1 (de) | 2004-01-29 |
| EP1224210A2 (de) | 2002-07-24 |
| DE60007345T2 (de) | 2004-11-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |