AR018868A1 - Composiciones farmaceuticas para la fragilidad musculoesqueletica, uso para la preparacion de medicamentos, estuche - Google Patents

Composiciones farmaceuticas para la fragilidad musculoesqueletica, uso para la preparacion de medicamentos, estuche

Info

Publication number
AR018868A1
AR018868A1 ARP990102847A ARP990102847A AR018868A1 AR 018868 A1 AR018868 A1 AR 018868A1 AR P990102847 A ARP990102847 A AR P990102847A AR P990102847 A ARP990102847 A AR P990102847A AR 018868 A1 AR018868 A1 AR 018868A1
Authority
AR
Argentina
Prior art keywords
fragility
compositions
medicines
preparation
case
Prior art date
Application number
ARP990102847A
Other languages
English (en)
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of AR018868A1 publication Critical patent/AR018868A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/02Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Se describen composiciones de combinacion farmacéutica y procedimientos, que comprenden (-)-cis-6-fenil-5-(4-(2-pirrolidin-1-il-etoxi)-fenil)-5,6,7,8-tetrahhidronaftaleno-2-ol o una sal farmacéuticamente aceptable del mismo y 2-amino-N-(1(R)-(2,4-difluoro-benciloximetil)-2-oxo-2-(3-oxo-3a(R)-piridin-2-ilmetil)-2-(2,2,2-trifluoro-etil)-2,3,3a,4,6,7-hexahidro-pirazolo[4,3-c]piridin-5-il)-2-metil-propionamida o una sal farmacéuticamente aceptable de lamisma, a procedimientos de uso de tales composiciones y a estuches que contienen tales composiciones. Las composiciones son utiles para el tratamientode la fragilidad musculoesquelética, incluyendo la osteoporosis, fracturas osteoporoticas, reduccion de masa osea, fragilidad y reduccion de masamuscular.
ARP990102847A 1998-06-16 1999-06-15 Composiciones farmaceuticas para la fragilidad musculoesqueletica, uso para la preparacion de medicamentos, estuche AR018868A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8942498P 1998-06-16 1998-06-16

Publications (1)

Publication Number Publication Date
AR018868A1 true AR018868A1 (es) 2001-12-12

Family

ID=22217565

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP990102847A AR018868A1 (es) 1998-06-16 1999-06-15 Composiciones farmaceuticas para la fragilidad musculoesqueletica, uso para la preparacion de medicamentos, estuche

Country Status (29)

Country Link
EP (1) EP1085867A1 (es)
JP (1) JP2002518328A (es)
KR (1) KR20010052817A (es)
CN (1) CN1305378A (es)
AP (1) AP9901581A0 (es)
AR (1) AR018868A1 (es)
AU (1) AU3342099A (es)
BG (1) BG105128A (es)
BR (1) BR9911357A (es)
CA (1) CA2335112A1 (es)
CO (1) CO5070586A1 (es)
EA (1) EA200001189A1 (es)
GT (1) GT199900083A (es)
HR (1) HRP20000857A2 (es)
HU (1) HUP0102395A2 (es)
ID (1) ID26726A (es)
IL (1) IL139587A0 (es)
IS (1) IS5727A (es)
MA (1) MA26648A1 (es)
NO (1) NO20006381D0 (es)
OA (1) OA11569A (es)
PA (1) PA8472101A1 (es)
PE (1) PE20000633A1 (es)
PL (1) PL345064A1 (es)
SK (1) SK18902000A3 (es)
TN (1) TNSN99118A1 (es)
UY (1) UY25557A1 (es)
WO (1) WO1999065488A1 (es)
ZA (1) ZA993973B (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1004306A3 (en) * 1998-08-06 2000-06-07 Pfizer Products Inc. Estrogen agonists/antagonists
AU2001276608A1 (en) * 2000-08-30 2002-03-13 Pfizer Products Inc. Sustained release formulations for growth hormone secretagogues
IL145106A0 (en) * 2000-08-30 2002-06-30 Pfizer Prod Inc Intermittent administration of a geowth hormone secretagogue
US7524866B2 (en) 2001-11-29 2009-04-28 Gtx, Inc. Prevention and treatment of androgen—deprivation induced osteoporosis
JP2005515988A (ja) * 2001-11-29 2005-06-02 ジーティーエックス・インコーポレイテッド 骨粗鬆症を引き起こすアンドロゲン欠乏の予防及び治療
US7476653B2 (en) 2003-06-18 2009-01-13 Tranzyme Pharma, Inc. Macrocyclic modulators of the ghrelin receptor
CU23558A1 (es) 2006-02-28 2010-07-20 Ct Ingenieria Genetica Biotech Compuestos análogos a los secretagogos peptidicos de la hormona de crecimiento
EP2644618B1 (en) 2007-02-09 2016-08-17 Ocera Therapeutics, Inc. tether intermediates for the synthesis of macrocyclic ghrelin receptor modulators

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA51676C2 (uk) * 1995-11-02 2002-12-16 Пфайзер Інк. (-)цис-6(s)-феніл-5(r)[4-(2-піролідин-1-ілетокси)феніл]-5,6,7,8-тетрагідронафталін-2-ол d-тартрат, спосіб його одержання, спосіб лікування захворювань, що піддаються лікуванню агоністами естрогену, та фармацевтична композиція
TW432073B (en) * 1995-12-28 2001-05-01 Pfizer Pyrazolopyridine compounds
HN1996000101A (es) * 1996-02-28 1997-06-26 Inc Pfizer Terapia combinada para la osteoporosis

Also Published As

Publication number Publication date
IL139587A0 (en) 2002-02-10
CA2335112A1 (en) 1999-12-23
PA8472101A1 (es) 2000-09-29
NO20006381L (no) 2000-12-14
JP2002518328A (ja) 2002-06-25
CN1305378A (zh) 2001-07-25
NO20006381D0 (no) 2000-12-14
HRP20000857A2 (en) 2001-10-31
GT199900083A (es) 2000-12-05
MA26648A1 (fr) 2004-12-20
HUP0102395A2 (hu) 2001-11-28
AP9901581A0 (en) 1999-06-30
EA200001189A1 (ru) 2001-06-25
KR20010052817A (ko) 2001-06-25
SK18902000A3 (sk) 2001-12-03
WO1999065488A1 (en) 1999-12-23
TNSN99118A1 (fr) 2005-11-10
ZA993973B (en) 2000-12-15
ID26726A (id) 2001-02-01
UY25557A1 (es) 2001-01-31
PE20000633A1 (es) 2000-07-26
CO5070586A1 (es) 2001-08-28
EP1085867A1 (en) 2001-03-28
IS5727A (is) 2000-11-24
PL345064A1 (en) 2001-11-19
BG105128A (en) 2001-11-30
BR9911357A (pt) 2001-03-13
AU3342099A (en) 2000-01-05
OA11569A (en) 2004-07-01

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Legal Events

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