AR012872A1 - Uso del mometanosulfonato del acido (e)-alfa-[2-n-butil-1-[(carboxifenil)metil]-1-h-imidazol-5- il]metilen-2-tiofenpropionico para la fabricacion de un medicamento ycomposicion farmaceutica que lo comprende para tratar hipertension sistolica aislada. - Google Patents
Uso del mometanosulfonato del acido (e)-alfa-[2-n-butil-1-[(carboxifenil)metil]-1-h-imidazol-5- il]metilen-2-tiofenpropionico para la fabricacion de un medicamento ycomposicion farmaceutica que lo comprende para tratar hipertension sistolica aislada.Info
- Publication number
- AR012872A1 AR012872A1 ARP980102464A ARP980102464A AR012872A1 AR 012872 A1 AR012872 A1 AR 012872A1 AR P980102464 A ARP980102464 A AR P980102464A AR P980102464 A ARP980102464 A AR P980102464A AR 012872 A1 AR012872 A1 AR 012872A1
- Authority
- AR
- Argentina
- Prior art keywords
- methylene
- alpha
- butyl
- methyl
- acid
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Fixed Capacitors And Capacitor Manufacturing Machines (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Abstract
La utilizacion de ácido (E)-alfa-[2-n-butil-1-[(4-carboxifenil)metil]-1-H- imidazol-5-il]metilen-2-tiofenpropionico (eprosartán) en la fabricacion de unmedicamento que se destina para el tratamiento de hipertension sistolica aislada.Una composicion farmacéutica para utilizacion en el tratamiento dehipertension sistolica aislada que comprende ácido (E)-alfa-[2-n-butil-1-[(4- carboxifenil)metil]-1-H-imidazol-5-il]metilen-2-tiofdenpropionico (eprosartán yun vehículo farmacéuticamente aceptable.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US4780097P | 1997-05-27 | 1997-05-27 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR012872A1 true AR012872A1 (es) | 2000-11-22 |
Family
ID=21951046
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP980102464A AR012872A1 (es) | 1997-05-27 | 1998-05-27 | Uso del mometanosulfonato del acido (e)-alfa-[2-n-butil-1-[(carboxifenil)metil]-1-h-imidazol-5- il]metilen-2-tiofenpropionico para la fabricacion de un medicamento ycomposicion farmaceutica que lo comprende para tratar hipertension sistolica aislada. |
Country Status (24)
Country | Link |
---|---|
US (1) | US20020040045A1 (es) |
EP (1) | EP1003506B1 (es) |
JP (1) | JP2002500673A (es) |
KR (1) | KR20010013014A (es) |
CN (1) | CN1257427A (es) |
AR (1) | AR012872A1 (es) |
AT (1) | ATE307580T1 (es) |
AU (1) | AU740646B2 (es) |
BR (1) | BR9809611A (es) |
CA (1) | CA2288722C (es) |
CZ (1) | CZ298390B6 (es) |
DE (1) | DE69832075T2 (es) |
ES (1) | ES2251083T3 (es) |
HU (1) | HUP0003249A3 (es) |
IL (1) | IL132154A (es) |
MX (1) | MXPA99010970A (es) |
NO (1) | NO326141B1 (es) |
NZ (1) | NZ337888A (es) |
PL (1) | PL191971B1 (es) |
SA (1) | SA98190174B1 (es) |
TR (1) | TR199902914T2 (es) |
TW (1) | TW579296B (es) |
WO (1) | WO1998053816A1 (es) |
ZA (1) | ZA984421B (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2006076097A2 (en) * | 2004-12-07 | 2006-07-20 | Nektar Therapeutics | Stable non-crystalline formulation comprising losartan |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US544080A (en) * | 1895-08-06 | Centrifugal filtering-machine | ||
US5185351A (en) * | 1989-06-14 | 1993-02-09 | Smithkline Beecham Corporation | Imidazolyl-alkenoic acids useful as angiotensin II receptor antagonists |
US5418250A (en) * | 1989-06-14 | 1995-05-23 | Smithkline Beecham Corporation | Imidazolyl-alkenoic acids useful as angiotensin II receptor antagonists |
JPH05199342A (ja) * | 1991-05-20 | 1993-08-06 | Xerox Corp | 無声の手書きによる携帯式通信装置および方法 |
-
1998
- 1998-05-25 ZA ZA984421A patent/ZA984421B/xx unknown
- 1998-05-27 NZ NZ337888A patent/NZ337888A/en unknown
- 1998-05-27 PL PL336886A patent/PL191971B1/pl not_active IP Right Cessation
- 1998-05-27 DE DE69832075T patent/DE69832075T2/de not_active Expired - Lifetime
- 1998-05-27 AT AT98923815T patent/ATE307580T1/de not_active IP Right Cessation
- 1998-05-27 CA CA002288722A patent/CA2288722C/en not_active Expired - Fee Related
- 1998-05-27 HU HU0003249A patent/HUP0003249A3/hu unknown
- 1998-05-27 IL IL13215498A patent/IL132154A/en not_active IP Right Cessation
- 1998-05-27 KR KR1019997010988A patent/KR20010013014A/ko not_active Application Discontinuation
- 1998-05-27 CN CN98805305A patent/CN1257427A/zh active Pending
- 1998-05-27 BR BR9809611-7A patent/BR9809611A/pt not_active Application Discontinuation
- 1998-05-27 AU AU76017/98A patent/AU740646B2/en not_active Ceased
- 1998-05-27 AR ARP980102464A patent/AR012872A1/es not_active Application Discontinuation
- 1998-05-27 TR TR1999/02914T patent/TR199902914T2/xx unknown
- 1998-05-27 ES ES98923815T patent/ES2251083T3/es not_active Expired - Lifetime
- 1998-05-27 TW TW087108204A patent/TW579296B/zh not_active IP Right Cessation
- 1998-05-27 MX MXPA99010970A patent/MXPA99010970A/es not_active IP Right Cessation
- 1998-05-27 EP EP98923815A patent/EP1003506B1/en not_active Expired - Lifetime
- 1998-05-27 CZ CZ0420099A patent/CZ298390B6/cs not_active IP Right Cessation
- 1998-05-27 WO PCT/US1998/010794 patent/WO1998053816A1/en active IP Right Grant
- 1998-05-27 JP JP50086599A patent/JP2002500673A/ja active Pending
- 1998-06-17 SA SA98190174A patent/SA98190174B1/ar unknown
-
1999
- 1999-11-26 NO NO19995797A patent/NO326141B1/no not_active IP Right Cessation
-
2001
- 2001-10-24 US US09/999,808 patent/US20020040045A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
ZA984421B (en) | 1998-11-27 |
EP1003506B1 (en) | 2005-10-26 |
AU740646B2 (en) | 2001-11-08 |
NO326141B1 (no) | 2008-10-06 |
SA98190174B1 (ar) | 2006-05-13 |
PL191971B1 (pl) | 2006-07-31 |
HUP0003249A3 (en) | 2002-02-28 |
NO995797D0 (no) | 1999-11-26 |
DE69832075D1 (de) | 2005-12-01 |
NZ337888A (en) | 2001-04-27 |
MXPA99010970A (es) | 2005-07-25 |
NO995797L (no) | 1999-11-26 |
CZ298390B6 (cs) | 2007-09-19 |
IL132154A (en) | 2002-12-01 |
CA2288722A1 (en) | 1998-12-03 |
CN1257427A (zh) | 2000-06-21 |
JP2002500673A (ja) | 2002-01-08 |
US20020040045A1 (en) | 2002-04-04 |
IL132154A0 (en) | 2001-03-19 |
BR9809611A (pt) | 2000-07-04 |
PL336886A1 (en) | 2000-07-17 |
CA2288722C (en) | 2007-04-24 |
CZ420099A3 (cs) | 2000-09-13 |
AU7601798A (en) | 1998-12-30 |
TR199902914T2 (xx) | 2000-06-21 |
ATE307580T1 (de) | 2005-11-15 |
EP1003506A1 (en) | 2000-05-31 |
EP1003506A4 (en) | 2000-11-29 |
ES2251083T3 (es) | 2006-04-16 |
WO1998053816A1 (en) | 1998-12-03 |
KR20010013014A (ko) | 2001-02-26 |
DE69832075T2 (de) | 2006-07-13 |
TW579296B (en) | 2004-03-11 |
HUP0003249A2 (hu) | 2002-01-28 |
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Legal Events
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FC | Refusal |