AP2011005774A0 - Glucagon analogues. - Google Patents
Glucagon analogues.Info
- Publication number
- AP2011005774A0 AP2011005774A0 AP2011005774A AP2011005774A AP2011005774A0 AP 2011005774 A0 AP2011005774 A0 AP 2011005774A0 AP 2011005774 A AP2011005774 A AP 2011005774A AP 2011005774 A AP2011005774 A AP 2011005774A AP 2011005774 A0 AP2011005774 A0 AP 2011005774A0
- Authority
- AP
- ARIPO
- Prior art keywords
- glucagon analogues
- glucagon
- analogues
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/605—Glucagons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/26—Glucagons
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12N—MICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
- C12N15/00—Mutation or genetic engineering; DNA or RNA concerning genetic engineering, vectors, e.g. plasmids, or their isolation, preparation or purification; Use of hosts therefor
- C12N15/09—Recombinant DNA-technology
- C12N15/11—DNA or RNA fragments; Modified forms thereof; Non-coding nucleic acids having a biological activity
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
AP2011005774A AP2011005774A0 (en) | 2008-12-15 | 2008-12-15 | Glucagon analogues. |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/GB2008/004121 WO2010070251A1 (en) | 2008-12-15 | 2008-12-15 | Glucagon analogues |
AP2011005774A AP2011005774A0 (en) | 2008-12-15 | 2008-12-15 | Glucagon analogues. |
Publications (1)
Publication Number | Publication Date |
---|---|
AP2011005774A0 true AP2011005774A0 (en) | 2011-06-30 |
Family
ID=40428061
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AP2011005774A AP2011005774A0 (en) | 2008-12-15 | 2008-12-15 | Glucagon analogues. |
Country Status (19)
Country | Link |
---|---|
US (2) | US8685919B2 (ja) |
EP (2) | EP2370459A1 (ja) |
JP (1) | JP5635529B2 (ja) |
KR (2) | KR20150116912A (ja) |
CN (1) | CN102282167B (ja) |
AP (1) | AP2011005774A0 (ja) |
AU (1) | AU2008365555B2 (ja) |
BR (1) | BRPI0823378A2 (ja) |
CA (1) | CA2747109A1 (ja) |
EA (1) | EA020537B1 (ja) |
HK (1) | HK1203531A1 (ja) |
IL (1) | IL213477A0 (ja) |
MA (1) | MA32970B1 (ja) |
MX (1) | MX2011006313A (ja) |
MY (1) | MY160219A (ja) |
SG (1) | SG172170A1 (ja) |
TN (1) | TN2011000295A1 (ja) |
UA (1) | UA104605C2 (ja) |
WO (1) | WO2010070251A1 (ja) |
Families Citing this family (64)
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US7563770B2 (en) | 2005-05-04 | 2009-07-21 | Zealand Pharma A/S | Glucagon-like-peptide-2 (GLP-2) analogues |
BRPI0718566A2 (pt) | 2006-11-08 | 2014-03-11 | Zealand Pharma As | Peptídeo, análogo do mesmo, composição farmacêutica, usos de um análogo de peptídeo, e de uma molécula de ácido nucléico, de um vetor de expressão, ou de uma célula hospedeira, molécula de ácido nucléico, vetor de expressão, célula hospedeira, métodos para produzir o análogo de peptídeo-2 tipo-glucagon (glp-2), e, kit terapêutico. |
KR20110126591A (ko) | 2008-12-15 | 2011-11-23 | 질랜드 파마 에이/에스 | 글루카곤 유사체 |
BRPI0823377A2 (pt) | 2008-12-15 | 2016-09-27 | Zealand Pharma As | análogos de glucagon |
JP5635530B2 (ja) | 2008-12-15 | 2014-12-03 | ジーランド ファーマ アクティーゼルスカブ | グルカゴン類似体 |
PE20121130A1 (es) * | 2009-07-13 | 2012-08-30 | Zealand Pharma As | Analogos de glucagon acilados |
AU2011247452B2 (en) | 2010-04-27 | 2016-03-17 | Zealand Pharma A/S | Peptide conjugates of GLP-1 receptor agonists and gastrin and their use |
AR081975A1 (es) | 2010-06-23 | 2012-10-31 | Zealand Pharma As | Analogos de glucagon |
AP2013006671A0 (en) * | 2010-06-24 | 2013-01-31 | Zealand Pharma As | Glucagon analogues |
KR20140043709A (ko) * | 2011-01-20 | 2014-04-10 | 질랜드 파마 에이/에스 | 아실화 글루카곤 유사체와 인슐린 유사체의 조합 |
TWI596110B (zh) | 2011-09-23 | 2017-08-21 | 諾佛 儂迪克股份有限公司 | 新穎升糖素類似物 |
AU2012331053A1 (en) | 2011-11-03 | 2014-05-29 | Zealand Pharma A/S | GLP-1 receptor agonist peptide gastrin conjugates |
AU2013255752B2 (en) * | 2012-05-03 | 2017-11-09 | Zealand Pharma A/S | Glucagon-like-peptide-2 (GLP-2) analogues |
US10100097B2 (en) | 2012-05-03 | 2018-10-16 | Zealand Pharma A/S | GIP-GLP-1 dual agonist compounds and methods |
EP2664374A1 (en) * | 2012-05-15 | 2013-11-20 | F. Hoffmann-La Roche AG | Lysin-glutamic acid dipeptide derivatives |
SG11201407860PA (en) | 2012-06-14 | 2014-12-30 | Sanofi Sa | Exendin-4 peptide analogues |
DK2875043T3 (en) | 2012-07-23 | 2017-03-27 | Zealand Pharma As | glucagon |
TWI608013B (zh) * | 2012-09-17 | 2017-12-11 | 西蘭製藥公司 | 升糖素類似物 |
AR092873A1 (es) | 2012-09-26 | 2015-05-06 | Cadila Healthcare Ltd | Peptidos como agonistas triples de los receptores de gip, glp-1 y glugagon |
UA116217C2 (uk) | 2012-10-09 | 2018-02-26 | Санофі | Пептидна сполука як подвійний агоніст рецепторів glp1-1 та глюкагону |
UA116553C2 (uk) | 2012-12-21 | 2018-04-10 | Санофі | Пептидна сполука - агоніст рецептора glp-1 i glp |
CA2907454C (en) | 2013-03-21 | 2021-05-04 | Sanofi-Aventis Deutschland Gmbh | Synthesis of hydantoin containing peptide products |
CN105102427B (zh) | 2013-03-21 | 2018-09-07 | 赛诺菲-安万特德国有限公司 | 含有环状酰亚胺的肽产物的合成 |
AR095986A1 (es) | 2013-04-03 | 2015-11-25 | Sanofi Sa | Proteínas modificadas que regulan glucosa en sangre con perfil alterado de actividad farmacológica y preparación de las mismas |
CN105307672B (zh) | 2013-04-18 | 2021-01-05 | 诺和诺德股份有限公司 | 用于医学用途的稳定、延长的glp-1/胰高血糖素受体共激动剂 |
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WO2016198624A1 (en) | 2015-06-12 | 2016-12-15 | Sanofi | Exendin-4 derivatives as trigonal glp-1/glucagon/gip receptor agonists |
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US8993516B2 (en) | 2008-04-14 | 2015-03-31 | Case Western Reserve University | Meal-time insulin analogues of enhanced stability |
MX2010011329A (es) | 2008-04-22 | 2011-03-15 | Univ Case Western Reserve | Analogos de insulina especificos de isoforma. |
TWI451876B (zh) | 2008-06-13 | 2014-09-11 | Lilly Co Eli | 聚乙二醇化之離脯胰島素化合物 |
EP2300037B1 (en) | 2008-06-17 | 2016-03-30 | Indiana University Research and Technology Corporation | Glucagon/glp-1 receptor co-agonists |
CN104447980A (zh) | 2008-06-17 | 2015-03-25 | 印第安纳大学研究及科技有限公司 | 在生理pH缓冲液中具有增强的溶解性和稳定性的胰高血糖素类似物 |
PL219335B1 (pl) | 2008-07-04 | 2015-04-30 | Inst Biotechnologii I Antybiotyków | Pochodna insuliny lub jej farmaceutycznie dopuszczalna sól, jej zastosowanie oraz zawierająca ją kompozycja farmaceutyczna |
MY158627A (en) | 2008-07-31 | 2016-10-31 | Univ Case Western Reserve | Halogen-stabilized insulin |
BRPI0823377A2 (pt) | 2008-12-15 | 2016-09-27 | Zealand Pharma As | análogos de glucagon |
JP5635530B2 (ja) | 2008-12-15 | 2014-12-03 | ジーランド ファーマ アクティーゼルスカブ | グルカゴン類似体 |
KR20110126591A (ko) | 2008-12-15 | 2011-11-23 | 질랜드 파마 에이/에스 | 글루카곤 유사체 |
US8697632B2 (en) | 2008-12-19 | 2014-04-15 | Indiana University Research And Technology Corporation | Amide based insulin prodrugs |
AU2009335712B2 (en) | 2008-12-19 | 2015-09-17 | Indiana University Research And Technology Corporation | Insulin analogs |
CN101519446A (zh) | 2009-03-31 | 2009-09-02 | 上海一就生物医药有限公司 | 一种重组人胰岛素及其类似物的制备方法 |
PE20121130A1 (es) | 2009-07-13 | 2012-08-30 | Zealand Pharma As | Analogos de glucagon acilados |
CN102892425A (zh) | 2010-01-20 | 2013-01-23 | 西兰制药公司 | 心脏病症的治疗 |
AR081975A1 (es) | 2010-06-23 | 2012-10-31 | Zealand Pharma As | Analogos de glucagon |
AP2013006671A0 (en) | 2010-06-24 | 2013-01-31 | Zealand Pharma As | Glucagon analogues |
KR20140043709A (ko) | 2011-01-20 | 2014-04-10 | 질랜드 파마 에이/에스 | 아실화 글루카곤 유사체와 인슐린 유사체의 조합 |
-
2008
- 2008-12-15 CA CA2747109A patent/CA2747109A1/en not_active Abandoned
- 2008-12-15 UA UAA201108817A patent/UA104605C2/uk unknown
- 2008-12-15 JP JP2011540187A patent/JP5635529B2/ja not_active Expired - Fee Related
- 2008-12-15 EP EP08875670A patent/EP2370459A1/en not_active Withdrawn
- 2008-12-15 US US13/139,493 patent/US8685919B2/en not_active Expired - Fee Related
- 2008-12-15 KR KR1020157027018A patent/KR20150116912A/ko not_active Application Discontinuation
- 2008-12-15 CN CN200880132682.4A patent/CN102282167B/zh not_active Expired - Fee Related
- 2008-12-15 BR BRPI0823378A patent/BRPI0823378A2/pt not_active IP Right Cessation
- 2008-12-15 MY MYPI2011002751A patent/MY160219A/en unknown
- 2008-12-15 MX MX2011006313A patent/MX2011006313A/es active IP Right Grant
- 2008-12-15 AP AP2011005774A patent/AP2011005774A0/xx unknown
- 2008-12-15 EP EP14175826.8A patent/EP2799447B1/en active Active
- 2008-12-15 EA EA201190047A patent/EA020537B1/ru not_active IP Right Cessation
- 2008-12-15 AU AU2008365555A patent/AU2008365555B2/en not_active Ceased
- 2008-12-15 KR KR1020117016184A patent/KR20110126589A/ko not_active Application Discontinuation
- 2008-12-15 WO PCT/GB2008/004121 patent/WO2010070251A1/en active Application Filing
- 2008-12-15 SG SG2011043700A patent/SG172170A1/en unknown
- 2008-12-15 MA MA34020A patent/MA32970B1/fr unknown
-
2011
- 2011-06-10 TN TN2011000295A patent/TN2011000295A1/fr unknown
- 2011-06-12 IL IL213477A patent/IL213477A0/en unknown
-
2014
- 2014-03-03 US US14/195,533 patent/US20150080295A1/en not_active Abandoned
-
2015
- 2015-05-05 HK HK15104289.5A patent/HK1203531A1/xx unknown
Also Published As
Publication number | Publication date |
---|---|
EP2799447A2 (en) | 2014-11-05 |
MX2011006313A (es) | 2011-09-27 |
JP5635529B2 (ja) | 2014-12-03 |
HK1203531A1 (en) | 2015-10-30 |
KR20110126589A (ko) | 2011-11-23 |
US8685919B2 (en) | 2014-04-01 |
WO2010070251A1 (en) | 2010-06-24 |
UA104605C2 (uk) | 2014-02-25 |
CN102282167B (zh) | 2014-08-13 |
IL213477A0 (en) | 2011-07-31 |
US20150080295A1 (en) | 2015-03-19 |
MA32970B1 (fr) | 2012-01-02 |
KR20150116912A (ko) | 2015-10-16 |
JP2012511899A (ja) | 2012-05-31 |
CA2747109A1 (en) | 2010-06-24 |
BRPI0823378A2 (pt) | 2019-09-24 |
SG172170A1 (en) | 2011-07-28 |
US20110286982A1 (en) | 2011-11-24 |
AU2008365555B2 (en) | 2016-01-14 |
EA201190047A1 (ru) | 2012-02-28 |
EP2799447B1 (en) | 2016-11-23 |
EP2370459A1 (en) | 2011-10-05 |
EP2799447A3 (en) | 2014-12-31 |
EA020537B1 (ru) | 2014-11-28 |
CN102282167A (zh) | 2011-12-14 |
TN2011000295A1 (en) | 2012-12-17 |
AU2008365555A1 (en) | 2011-07-21 |
MY160219A (en) | 2017-02-28 |
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