ZA9811124B - Novel salts of metformin and method. - Google Patents

Novel salts of metformin and method.

Info

Publication number
ZA9811124B
ZA9811124B ZA9811124A ZA9811124A ZA9811124B ZA 9811124 B ZA9811124 B ZA 9811124B ZA 9811124 A ZA9811124 A ZA 9811124A ZA 9811124 A ZA9811124 A ZA 9811124A ZA 9811124 B ZA9811124 B ZA 9811124B
Authority
ZA
South Africa
Prior art keywords
metformin
novel salts
salts
novel
Prior art date
Application number
ZA9811124A
Other languages
English (en)
Inventor
Peter Timmins
William J Winter
Sushil K Srivastava
Alison E Bretnall
Chenkou Wei
Gerald L Powers
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of ZA9811124B publication Critical patent/ZA9811124B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/20—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylguanidines
    • C07C279/24—Y being a hetero atom
    • C07C279/26—X and Y being nitrogen atoms, i.e. biguanides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ZA9811124A 1997-12-08 1998-12-04 Novel salts of metformin and method. ZA9811124B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US98658697A 1997-12-08 1997-12-08

Publications (1)

Publication Number Publication Date
ZA9811124B true ZA9811124B (en) 2000-06-05

Family

ID=25532567

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA9811124A ZA9811124B (en) 1997-12-08 1998-12-04 Novel salts of metformin and method.

Country Status (11)

Country Link
US (1) US6031004A (ja)
EP (1) EP1039890B1 (ja)
JP (1) JP4278863B2 (ja)
AR (1) AR017819A1 (ja)
AT (1) ATE261935T1 (ja)
AU (1) AU738804B2 (ja)
CA (1) CA2312990C (ja)
DE (1) DE69822505T2 (ja)
ES (1) ES2216335T3 (ja)
WO (1) WO1999029314A1 (ja)
ZA (1) ZA9811124B (ja)

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CN101855204B (zh) * 2007-09-21 2013-09-11 韩兀生物制药株式会社 N,n-二甲基亚氨二羰酸二酰胺二羧酸盐、其制备方法及其药物组合物
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WO2011008053A2 (ko) * 2009-07-17 2011-01-20 한올바이오파마주식회사 Ｎ,ｎ-디메틸 이미도디카르본이미딕 디아미드의 프로피온산염, 이의 제조방법, 이를 포함하는 약제학적 조성물 및 이를 포함하는 복합제제
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CN102391160A (zh) * 2011-11-23 2012-03-28 黎波 二甲双胍与2，5-二羟基苯磺酸盐以及二甲双胍与2，5-二羟基苯磺酸盐的复方组合物
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WO2017195086A1 (en) * 2016-05-10 2017-11-16 Sarath Kumar Kamavarapu Salts of n,n-dimethylbiguanide and preparation methods thereof
WO2018034627A1 (en) 2016-08-18 2018-02-22 İlko Ilaç Sanayi Ve Ticaret Anonim Şirketi Pharmaceutical composition of antidiabetic tablet
JP2021528738A (ja) 2018-06-14 2021-10-21 アストラゼネカ・ユーケイ・リミテッドＡｓｔｒａＺｅｎｅｃａ ＵＫ Ｌｉｍｉｔｅｄ メトホルミン医薬組成物を用いて血糖を低下させるための方法
CN113105367B (zh) * 2021-03-30 2022-08-02 广州大学 一类二甲双胍盐及其制备方法和应用

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Also Published As

Publication number Publication date
CA2312990A1 (en) 1999-06-17
AU738804B2 (en) 2001-09-27
AR017819A1 (es) 2001-10-24
DE69822505T2 (de) 2005-01-20
EP1039890B1 (en) 2004-03-17
WO1999029314A1 (en) 1999-06-17
JP4278863B2 (ja) 2009-06-17
ATE261935T1 (de) 2004-04-15
US6031004A (en) 2000-02-29
DE69822505D1 (de) 2004-04-22
ES2216335T3 (es) 2004-10-16
EP1039890A4 (en) 2001-04-04
EP1039890A1 (en) 2000-10-04
JP2001525361A (ja) 2001-12-11
CA2312990C (en) 2008-04-29
AU1602699A (en) 1999-06-28

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