ZA771944B - Process for the preparation of aminoglycoside antibiotics and novel intermediates therefor - Google Patents

Process for the preparation of aminoglycoside antibiotics and novel intermediates therefor

Info

Publication number
ZA771944B
ZA771944B ZA00771944A ZA771944A ZA771944B ZA 771944 B ZA771944 B ZA 771944B ZA 00771944 A ZA00771944 A ZA 00771944A ZA 771944 A ZA771944 A ZA 771944A ZA 771944 B ZA771944 B ZA 771944B
Authority
ZA
South Africa
Prior art keywords
preparation
novel intermediates
aminoglycoside antibiotics
intermediates therefor
therefor
Prior art date
Application number
ZA00771944A
Other languages
English (en)
Inventor
R Plews
W Million
K Richardson
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of ZA771944B publication Critical patent/ZA771944B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ZA00771944A 1976-04-14 1977-03-30 Process for the preparation of aminoglycoside antibiotics and novel intermediates therefor ZA771944B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB15421/76A GB1530201A (en) 1976-04-14 1976-04-14 Process for the preparation of aminoglycoside antibiotics and intermediates therefor

Publications (1)

Publication Number Publication Date
ZA771944B true ZA771944B (en) 1978-03-29

Family

ID=10058845

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA00771944A ZA771944B (en) 1976-04-14 1977-03-30 Process for the preparation of aminoglycoside antibiotics and novel intermediates therefor

Country Status (28)

Country Link
JP (2) JPS52139044A (fr)
AR (1) AR219074A1 (fr)
AT (1) AT356267B (fr)
AU (1) AU497416B2 (fr)
BE (1) BE853564A (fr)
BG (2) BG28072A4 (fr)
CA (1) CA1083568A (fr)
CH (1) CH622528A5 (fr)
CS (1) CS202570B2 (fr)
DD (2) DD135496A5 (fr)
DE (1) DE2716533C3 (fr)
DK (1) DK164277A (fr)
EG (1) EG12909A (fr)
ES (1) ES457793A1 (fr)
FI (1) FI771144A (fr)
FR (1) FR2348223A1 (fr)
GB (1) GB1530201A (fr)
GR (1) GR68936B (fr)
IE (1) IE45030B1 (fr)
IL (1) IL51775A (fr)
LU (1) LU77108A1 (fr)
NL (1) NL7703567A (fr)
NZ (1) NZ183733A (fr)
PH (1) PH14029A (fr)
PL (2) PL197372A1 (fr)
PT (1) PT66422B (fr)
RO (2) RO79969A (fr)
ZA (1) ZA771944B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2924659A1 (de) * 1979-06-19 1981-01-22 Bayer Ag Pseudotrisaccharide, ihre herstellung und verwendung als arzneimittel
JPH0414628Y2 (fr) * 1984-12-13 1992-04-02
JPS61191642U (fr) * 1985-05-20 1986-11-28
IT1225484B (it) * 1987-11-27 1990-11-14 Pierrel Spa Procedimento di sintesi dell'amikacina
CN101481397B (zh) * 2009-01-23 2012-10-31 北京大学 一种新的卡那霉素a衍生物及其制备方法和用途
DK3400944T3 (da) 2010-11-08 2020-10-12 Albireo Ab Ibat-inhibitorer til behandling af leversygdomme
WO2015199147A1 (fr) 2014-06-25 2015-12-30 味の素株式会社 Préparation pharmaceutique solide, et procédé d'inhibition ou d'atténuation de coloration de celle-ci
JP6581082B2 (ja) 2014-06-25 2019-09-25 Ｅａファーマ株式会社 固形製剤及びその安定化方法
EP3012252A1 (fr) 2014-10-24 2016-04-27 Ferring BV Formes crystallines d'Elobixibat
US10441605B2 (en) 2016-02-09 2019-10-15 Albireo Ab Oral cholestyramine formulation and use thereof
US10441604B2 (en) 2016-02-09 2019-10-15 Albireo Ab Cholestyramine pellets and methods for preparation thereof
US10786529B2 (en) 2016-02-09 2020-09-29 Albireo Ab Oral cholestyramine formulation and use thereof
US11007142B2 (en) 2018-08-09 2021-05-18 Albireo Ab Oral cholestyramine formulation and use thereof
US10722457B2 (en) 2018-08-09 2020-07-28 Albireo Ab Oral cholestyramine formulation and use thereof

Also Published As

Publication number Publication date
EG12909A (en) 1979-12-31
DD130661A5 (de) 1978-04-19
BG27759A3 (en) 1979-12-12
BE853564A (fr) 1977-10-13
IE45030L (en) 1977-10-14
ATA261477A (de) 1979-09-15
DE2716533A1 (de) 1977-11-03
CS202570B2 (en) 1981-01-30
JPS5549587B2 (fr) 1980-12-12
PT66422A (en) 1977-05-01
JPS535141A (en) 1978-01-18
AT356267B (de) 1980-04-25
NL7703567A (nl) 1977-10-18
GB1530201A (en) 1978-10-25
RO79969B (ro) 1983-01-30
IL51775A0 (en) 1977-05-31
FR2348223A1 (fr) 1977-11-10
JPS5421326B2 (fr) 1979-07-30
GR68936B (fr) 1982-03-29
CA1083568A (fr) 1980-08-12
IL51775A (en) 1980-07-31
DE2716533B2 (de) 1981-04-30
AU2372177A (en) 1978-10-05
PT66422B (en) 1978-09-18
DD135496A5 (de) 1979-05-09
IE45030B1 (en) 1982-06-02
JPS52139044A (en) 1977-11-19
BG28072A4 (en) 1980-02-25
PH14029A (en) 1980-12-12
LU77108A1 (fr) 1979-01-18
AU497416B2 (en) 1978-12-14
PL197372A1 (pl) 1979-06-18
RO74431A (fr) 1981-08-30
CH622528A5 (en) 1981-04-15
PL112867B1 (en) 1980-11-29
ES457793A1 (es) 1978-08-01
DK164277A (da) 1977-10-15
FI771144A (fr) 1977-10-15
NZ183733A (en) 1979-12-11
DE2716533C3 (de) 1982-05-13
AR219074A1 (es) 1980-07-31
RO79969A (fr) 1983-02-01

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