ZA761043B - New piperazinylimino rifamycins - Google Patents
New piperazinylimino rifamycinsInfo
- Publication number
- ZA761043B ZA761043B ZA1043A ZA761043A ZA761043B ZA 761043 B ZA761043 B ZA 761043B ZA 1043 A ZA1043 A ZA 1043A ZA 761043 A ZA761043 A ZA 761043A ZA 761043 B ZA761043 B ZA 761043B
- Authority
- ZA
- South Africa
- Prior art keywords
- piperazinylimino
- rifamycins
- new
- piperazinylimino rifamycins
- new piperazinylimino
- Prior art date
Links
- 229930189077 Rifamycin Natural products 0.000 title 1
- -1 piperazinylimino rifamycins Chemical class 0.000 title 1
- 229940081192 rifamycins Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB10020/75A GB1478563A (en) | 1975-03-05 | 1975-03-05 | Rifamycin derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA761043B true ZA761043B (en) | 1977-01-26 |
Family
ID=9959968
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA1043A ZA761043B (en) | 1975-03-05 | 1976-02-23 | New piperazinylimino rifamycins |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US4002752A (enExample) |
| JP (1) | JPS51113900A (enExample) |
| AR (1) | AR210113A1 (enExample) |
| AT (1) | AT344896B (enExample) |
| BE (1) | BE839255A (enExample) |
| CA (1) | CA1057748A (enExample) |
| CH (1) | CH610325A5 (enExample) |
| DD (1) | DD123888A5 (enExample) |
| DE (1) | DE2608218C3 (enExample) |
| DK (1) | DK136655B (enExample) |
| ES (1) | ES445790A1 (enExample) |
| FI (1) | FI59102C (enExample) |
| FR (1) | FR2302742A1 (enExample) |
| GB (1) | GB1478563A (enExample) |
| HK (1) | HK35282A (enExample) |
| HU (1) | HU170451B (enExample) |
| IE (1) | IE42881B1 (enExample) |
| KE (1) | KE3099A (enExample) |
| LU (1) | LU74478A1 (enExample) |
| MX (1) | MX3737E (enExample) |
| NL (1) | NL165745C (enExample) |
| NO (1) | NO143796C (enExample) |
| PT (1) | PT64866B (enExample) |
| SE (1) | SE420728B (enExample) |
| SU (1) | SU575030A3 (enExample) |
| YU (1) | YU39477B (enExample) |
| ZA (1) | ZA761043B (enExample) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2728869A1 (de) * | 1976-06-25 | 1977-12-29 | Antibiotice Iasi Intreprindere | Rifamycinen und verfahren zu deren herstellung |
| GR64108B (en) * | 1977-04-15 | 1980-01-24 | Dso Pharmachim | Method for the preparation of azomethine-derivatives of rifamycin s.v |
| GB1576886A (en) * | 1977-04-20 | 1980-10-15 | Lepetit Spa | Rifamycin derivatives |
| GB1594134A (en) * | 1977-11-25 | 1981-07-30 | Holco Investment Inc | Rifamycins |
| AU536524B2 (en) * | 1979-06-28 | 1984-05-10 | Gruppo Lepetit S.P.A. | Water soluble hydrozones of 3-formylifamyan |
| US4447432A (en) * | 1981-11-17 | 1984-05-08 | Farmitalia Carlo Erba S.P.A. | Azino rifamycins |
| US4681938A (en) * | 1984-08-27 | 1987-07-21 | Ciba-Geigy Corporation | Novel polycyclic hydrazones of rifamycins, their manufacture, and their pharmaceutical compositions for treating tuberculosis |
| HUT47586A (en) * | 1985-10-18 | 1989-03-28 | Ciba Geigy Ag | Process for production of substituated 3-/4-benzil-piperazinil/-piphamicins |
| AU621811B2 (en) * | 1987-09-25 | 1992-03-26 | Ciba-Geigy Ag | Diacyl derivatives of 4-(trialkylbenzyl)-piperazinyl compounds |
| GB8816620D0 (en) * | 1988-07-13 | 1988-08-17 | Lepetit Spa | Rifapentine hydrohalides |
| CA2082809C (en) * | 1990-06-29 | 1995-10-17 | Marino Nebuloni | Pure crystalline form of rifapentine |
| US8404664B2 (en) | 2005-08-11 | 2013-03-26 | Targanta Therapeutics, Inc. | Phosphonated Rifamycins and uses thereof for the prevention and treatment of bone and joint infections |
| US8524691B2 (en) | 2008-08-13 | 2013-09-03 | The Medicines Company | Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections |
| RU2496475C2 (ru) | 2011-10-26 | 2013-10-27 | Александр Васильевич Иващенко | Фармацевтическая композиция и набор для лечения бактериальных инфекций |
| CN104736152B (zh) | 2012-08-13 | 2018-01-23 | 阿迪帕姆单人股份公司 | 包含3‑甲酰基利福霉素sv和3‑甲酰基利福霉素s的3‑(4‑肉桂基‑1‑哌嗪基)氨基衍生物的药物制剂以及它们的制备方法 |
| CN103951677B (zh) * | 2014-03-17 | 2016-04-06 | 四川省长征药业股份有限公司 | 利福喷丁的制备方法 |
| WO2022225384A1 (es) * | 2021-04-21 | 2022-10-27 | Interquim, S.A. De C.V. | Proceso de obtención de rifapentina. con una nueva forma cristalina |
| CN115047122B (zh) * | 2022-06-29 | 2023-05-02 | 重庆华邦胜凯制药有限公司 | 利福喷丁及其合成过程中所产生的杂质的分析方法 |
| CN117186032A (zh) * | 2023-09-08 | 2023-12-08 | 徐州博康信息化学品有限公司 | 1-氨基-4-环戊基哌嗪及其中间体的制备方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR208F (enExample) * | 1964-07-31 | |||
| AR205434A1 (es) * | 1972-03-27 | 1976-05-07 | Lepetit Spa | Proceso para la preparacion de 3-acilhidrazonometil rifamicinas sv |
| GB1392272A (en) * | 1972-05-31 | 1975-04-30 | Lepetit Spa | 3-formylrifamycin azines |
-
1975
- 1975-03-05 GB GB10020/75A patent/GB1478563A/en not_active Expired
-
1976
- 1976-02-19 NO NO760549A patent/NO143796C/no unknown
- 1976-02-23 ZA ZA1043A patent/ZA761043B/xx unknown
- 1976-02-23 SE SE7602122A patent/SE420728B/xx not_active IP Right Cessation
- 1976-02-25 DK DK78476AA patent/DK136655B/da not_active IP Right Cessation
- 1976-02-26 US US05/661,587 patent/US4002752A/en not_active Expired - Lifetime
- 1976-02-28 DE DE2608218A patent/DE2608218C3/de not_active Expired
- 1976-03-03 NL NL7602191.A patent/NL165745C/xx not_active IP Right Cessation
- 1976-03-03 SU SU7602329559A patent/SU575030A3/ru active
- 1976-03-03 AR AR262431A patent/AR210113A1/es active
- 1976-03-04 CA CA247,156A patent/CA1057748A/en not_active Expired
- 1976-03-04 PT PT64866A patent/PT64866B/pt unknown
- 1976-03-04 CH CH271376A patent/CH610325A5/xx not_active IP Right Cessation
- 1976-03-04 HU HULE790A patent/HU170451B/hu unknown
- 1976-03-04 MX MX7636U patent/MX3737E/es unknown
- 1976-03-04 LU LU74478A patent/LU74478A1/xx unknown
- 1976-03-04 IE IE448/76A patent/IE42881B1/en not_active IP Right Cessation
- 1976-03-04 JP JP51023701A patent/JPS51113900A/ja active Granted
- 1976-03-05 ES ES445790A patent/ES445790A1/es not_active Expired
- 1976-03-05 AT AT162876A patent/AT344896B/de not_active IP Right Cessation
- 1976-03-05 FR FR7606379A patent/FR2302742A1/fr active Granted
- 1976-03-05 BE BE164907A patent/BE839255A/xx not_active IP Right Cessation
- 1976-03-05 DD DD191727A patent/DD123888A5/xx unknown
- 1976-03-05 FI FI760561A patent/FI59102C/fi not_active IP Right Cessation
- 1976-03-05 YU YU572/76A patent/YU39477B/xx unknown
-
1980
- 1980-11-01 KE KE3099A patent/KE3099A/xx unknown
-
1982
- 1982-08-03 HK HK352/82A patent/HK35282A/xx unknown
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