ZA200802163B - 5-(phenylisoxazolylethoxy)-triazol-3-YL substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders - Google Patents

5-(phenylisoxazolylethoxy)-triazol-3-YL substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders

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Publication number
ZA200802163B
ZA200802163B ZA200802163A ZA200802163A ZA200802163B ZA 200802163 B ZA200802163 B ZA 200802163B ZA 200802163 A ZA200802163 A ZA 200802163A ZA 200802163 A ZA200802163 A ZA 200802163A ZA 200802163 B ZA200802163 B ZA 200802163B
Authority
ZA
South Africa
Prior art keywords
phenylisoxazolylethoxy
psychiatric
triazol
neurological
treatment
Prior art date
Application number
ZA200802163A
Other languages
English (en)
Inventor
Minidis Alexander
Wensbo David
Slassi Abdelmalik
Isaac Methvin
Ericsson Caroline
Profir Veronica
Bergstrom Per-Olov
Edwards Louise
Arora Jalaj
Xin Tao
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of ZA200802163B publication Critical patent/ZA200802163B/xx

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P27/00—Drugs for disorders of the senses
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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  • Engineering & Computer Science (AREA)
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  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Psychiatry (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Emergency Medicine (AREA)
  • Psychology (AREA)
  • Rheumatology (AREA)
  • Virology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Immunology (AREA)
  • AIDS & HIV (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
ZA200802163A 2005-09-29 2008-03-07 5-(phenylisoxazolylethoxy)-triazol-3-YL substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders ZA200802163B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US72152705P 2005-09-29 2005-09-29

Publications (1)

Publication Number Publication Date
ZA200802163B true ZA200802163B (en) 2009-09-30

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ZA200802163A ZA200802163B (en) 2005-09-29 2008-03-07 5-(phenylisoxazolylethoxy)-triazol-3-YL substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders

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Country Link
US (4) US7476684B2 (OSRAM)
EP (1) EP1934209A1 (OSRAM)
JP (2) JP2009510064A (OSRAM)
KR (1) KR20080050421A (OSRAM)
CN (1) CN101273037A (OSRAM)
AR (1) AR058807A1 (OSRAM)
AU (1) AU2006297462A1 (OSRAM)
BR (1) BRPI0616228A2 (OSRAM)
CA (1) CA2623009A1 (OSRAM)
EC (1) ECSP088283A (OSRAM)
IL (1) IL189990A0 (OSRAM)
NO (1) NO20081434L (OSRAM)
RU (1) RU2008108219A (OSRAM)
TW (1) TW200800976A (OSRAM)
UA (1) UA92503C2 (OSRAM)
UY (1) UY29796A1 (OSRAM)
WO (1) WO2007040982A1 (OSRAM)
ZA (1) ZA200802163B (OSRAM)

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US8080568B1 (en) * 2010-06-29 2011-12-20 Ewha University - Industry Collaboration Foundation 2-pyridyl substituted imidazoles as therapeutic ALK5 and/or ALK4 inhibitors
UA112418C2 (uk) * 2010-09-07 2016-09-12 Астеллас Фарма Інк. Терапевтичний болезаспокійливий засіб
JP2013544874A (ja) 2010-12-08 2013-12-19 オスロ ユニヴァーシティー ホスピタル エイチエフ Ｗｎｔシグナル伝達経路阻害薬としてのトリアゾール誘導体
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WO2005077345A1 (en) 2004-02-03 2005-08-25 Astrazeneca Ab Compounds for the treatment of gastro-esophageal reflux disease
CA2556268A1 (en) 2004-02-18 2005-09-01 Astrazeneca Ab Acetylinic piperazine compounds and their use as metabotropic glutamate receptor antagonists
UA85576C2 (ru) 2004-02-18 2009-02-10 Астразенека Аб Тетразольные соединения и их применение в качестве метаботропических антагонистов рецепторов глутамата
SI1716152T1 (sl) 2004-02-18 2008-12-31 Astrazeneca Ab Kondenzirane heterociklične spojine in njihova uporaba kot antagonisti metabotropnega receptorja za zdravljenje gastrointestinalnih motenj
RU2006127575A (ru) 2004-02-18 2008-03-27 Астразенека Аб (Se) Соединение триазола и их применение в качестве антагонистов метаботропного рецептора глутамата
NZ548693A (en) 2004-02-18 2010-05-28 Astrazeneca Ab Polyheterocyclic compounds and their use as metabotropic glutamate receptor antagonists
US7585881B2 (en) 2004-02-18 2009-09-08 Astrazeneca Ab Additional heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
UY29796A1 (es) * 2005-09-29 2007-04-30 Astrazeneca Ab Nuevos compuestos para el tratamiento de trastornos neurológicos, psiquiátricos o del dolor

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IL189990A0 (en) 2008-08-07
US20070270469A1 (en) 2007-11-22
US7476684B2 (en) 2009-01-13
US20070129408A1 (en) 2007-06-07
UY29796A1 (es) 2007-04-30
US20070270468A1 (en) 2007-11-22
UA92503C2 (ru) 2010-11-10
TW200800976A (en) 2008-01-01
JP2010013476A (ja) 2010-01-21
CA2623009A1 (en) 2007-04-12
RU2008108219A (ru) 2009-11-10
KR20080050421A (ko) 2008-06-05
CN101273037A (zh) 2008-09-24
JP2009510064A (ja) 2009-03-12
BRPI0616228A2 (pt) 2011-06-14
US20080227824A1 (en) 2008-09-18
AR058807A1 (es) 2008-02-27
NO20081434L (no) 2008-05-19
WO2007040982A1 (en) 2007-04-12
AU2006297462A1 (en) 2007-04-12
EP1934209A1 (en) 2008-06-25

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