IL189990A0 - 5-(phenylisoxazolylethoxy) -triazol-3-yl substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders - Google Patents

5-(phenylisoxazolylethoxy) -triazol-3-yl substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders

Info

Publication number
IL189990A0
IL189990A0 IL189990A IL18999008A IL189990A0 IL 189990 A0 IL189990 A0 IL 189990A0 IL 189990 A IL189990 A IL 189990A IL 18999008 A IL18999008 A IL 18999008A IL 189990 A0 IL189990 A0 IL 189990A0
Authority
IL
Israel
Prior art keywords
phenylisoxazolylethoxy
psychiatric
triazol
neurological
treatment
Prior art date
Application number
IL189990A
Other languages
English (en)
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of IL189990A0 publication Critical patent/IL189990A0/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A—HUMAN NECESSITIES
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    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
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    • A61P27/00—Drugs for disorders of the senses
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
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    • A—HUMAN NECESSITIES
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    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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    • A61P31/18—Antivirals for RNA viruses for HIV
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Emergency Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Virology (AREA)
  • Hospice & Palliative Care (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Anesthesiology (AREA)
IL189990A 2005-09-29 2008-03-06 5-(phenylisoxazolylethoxy) -triazol-3-yl substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders IL189990A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US72152705P 2005-09-29 2005-09-29
PCT/US2006/036423 WO2007040982A1 (en) 2005-09-29 2006-09-20 5- (phenylisoxazolylethoxy) -triazol- 3 -yl substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders

Publications (1)

Publication Number Publication Date
IL189990A0 true IL189990A0 (en) 2008-08-07

Family

ID=37745801

Family Applications (1)

Application Number Title Priority Date Filing Date
IL189990A IL189990A0 (en) 2005-09-29 2008-03-06 5-(phenylisoxazolylethoxy) -triazol-3-yl substituted pyridine compounds for the treatment of neurological, psychiatric or pain disorders

Country Status (18)

Country Link
US (4) US20080227824A1 (OSRAM)
EP (1) EP1934209A1 (OSRAM)
JP (2) JP2009510064A (OSRAM)
KR (1) KR20080050421A (OSRAM)
CN (1) CN101273037A (OSRAM)
AR (1) AR058807A1 (OSRAM)
AU (1) AU2006297462A1 (OSRAM)
BR (1) BRPI0616228A2 (OSRAM)
CA (1) CA2623009A1 (OSRAM)
EC (1) ECSP088283A (OSRAM)
IL (1) IL189990A0 (OSRAM)
NO (1) NO20081434L (OSRAM)
RU (1) RU2008108219A (OSRAM)
TW (1) TW200800976A (OSRAM)
UA (1) UA92503C2 (OSRAM)
UY (1) UY29796A1 (OSRAM)
WO (1) WO2007040982A1 (OSRAM)
ZA (1) ZA200802163B (OSRAM)

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EA201000656A1 (ru) * 2007-10-26 2010-12-30 Астразенека Аб Аминопроизводные 1,2,4-триазола в качестве модуляторов mglur5
TW201011016A (en) * 2008-08-12 2010-03-16 Astrazeneca Ab New compounds 501
EP2323658A4 (en) * 2008-08-12 2011-10-05 Astrazeneca Ab NEW CRYSTALLINE FORM OF (5- {(IR) -1- [5- (3-CHLOROPHENYL) ISOXAZOL-3-YL] ETHOXY} -4-METHYL-4H-L, 2, 4-TRIAZOL-3-YL) - PYRIDINE
AU2009307825A1 (en) * 2008-10-22 2010-04-29 Rick FRIEDMAN Treatment and/or prevention of inner ear conditions by modulation of a metabotropic glutamate receptor
EP2376474A4 (en) * 2008-12-12 2012-07-04 Astrazeneca Ab A NEW METHOD FOR THE PRODUCTION OF 4- [4-METHYL-5- (C1-10-ALKYLTHIO / C5-10-ARYL-C1-6-ALKYLTHIO) -4H-1,2,4-TRIAZOL-2-YL] PYRIDINES
SG171755A1 (en) * 2008-12-18 2011-07-28 Astrazeneca Ab New process for the preparation of 1- [5- (3-chloro-phenyl) - isooxazol-3-yl] -ethanone and (r) -1- [5- (3-chloro-phenyl) - isooxazol-3-yl] -ethanol
WO2010071559A1 (en) * 2008-12-18 2010-06-24 Astrazeneca Ab Processes for the manufacture of 3-{4-methyl-5- [ (ir) -1- (2- (3-methylphenyl) -2h-tetrazol-5-yl) -ethoxy] -4h- [1,2, 4] triazol-3-yl} -pyridine, 4-methyl-3-methylthio-5- (3- pyridyl)-l,2,4-triazole, and (ir) -1- [2- (3-methylphenyl) -2h- tetrazol-5-yl] ethanol
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US8835444B2 (en) 2010-02-02 2014-09-16 Novartis Ag Cyclohexyl amide derivatives as CRF receptor antagonists
US8080568B1 (en) * 2010-06-29 2011-12-20 Ewha University - Industry Collaboration Foundation 2-pyridyl substituted imidazoles as therapeutic ALK5 and/or ALK4 inhibitors
UA112418C2 (uk) 2010-09-07 2016-09-12 Астеллас Фарма Інк. Терапевтичний болезаспокійливий засіб
WO2012076898A1 (en) 2010-12-08 2012-06-14 Oslo University Hospital Hf Triazole derivatives as wnt signaling pathway inhibitors
CA2830458A1 (en) 2011-03-18 2012-09-27 Novartis Ag Combinations of alpha 7 nicotinic acetylcholine receptor activators and mglur5 antagonists for use in dopamine induced dyskinesia in parkinson's disease
WO2016163754A1 (en) * 2015-04-07 2016-10-13 Medpacto Inc. Pharmaceutical composition for preventing or treating cancer and method using thereof
KR20160120157A (ko) 2015-04-07 2016-10-17 주식회사 메드팩토 암 예방 또는 치료용 약학적 조성물 및 이를 이용한 방법
KR102027368B1 (ko) * 2018-05-29 2019-10-01 서울대학교산학협력단 통증의 강도를 측정하는 방법
CN113329754A (zh) 2018-11-20 2021-08-31 麻雀制药股份有限公司 用于施用皮质类固醇的方法
MX2021013849A (es) 2019-05-15 2022-01-07 Claes Thulin 4-[5-[(rac)-1-[5-(3-clorofenil)-3-isoxazolil]etoxi]-4-metil-4h-1, 2,4-triazol-3-il]piridina para usar en la prevencion y/o el tratamiento del dolor en un animal.
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BRPI0507501A (pt) 2004-02-18 2007-06-26 Astrazeneca Ab composto, composição farmacêutica, uso do composto, método para o tratamento de distúrbios mediados por mglur5, e, método para inibir a ativação de receptores de mglur5
EP1716125B1 (en) 2004-02-18 2013-06-19 AstraZeneca AB Tetrazole compounds and their use as metabotropic glutamate receptor antagonits
BRPI0507495A (pt) 2004-02-18 2007-07-10 Astrazeneca Ab composto, composição farmacêutica, uso do composto método para o tratamento de distúrbios mediados por mglur5, e, método para inibir a ativação de receptores de mglur5
UY29796A1 (es) * 2005-09-29 2007-04-30 Astrazeneca Ab Nuevos compuestos para el tratamiento de trastornos neurológicos, psiquiátricos o del dolor

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ZA200802163B (en) 2009-09-30
US20070129408A1 (en) 2007-06-07
NO20081434L (no) 2008-05-19
ECSP088283A (es) 2008-04-28
EP1934209A1 (en) 2008-06-25
US20070270469A1 (en) 2007-11-22
AR058807A1 (es) 2008-02-27
TW200800976A (en) 2008-01-01
JP2009510064A (ja) 2009-03-12
UY29796A1 (es) 2007-04-30
KR20080050421A (ko) 2008-06-05
US20080227824A1 (en) 2008-09-18
CA2623009A1 (en) 2007-04-12
WO2007040982A1 (en) 2007-04-12
US20070270468A1 (en) 2007-11-22
BRPI0616228A2 (pt) 2011-06-14
AU2006297462A1 (en) 2007-04-12
RU2008108219A (ru) 2009-11-10
UA92503C2 (ru) 2010-11-10
US7476684B2 (en) 2009-01-13
CN101273037A (zh) 2008-09-24
JP2010013476A (ja) 2010-01-21

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