ZA200602442B - Pyridine derivatives and use thereof as urotensin II antagonists - Google Patents

Pyridine derivatives and use thereof as urotensin II antagonists Download PDF

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Publication number
ZA200602442B
ZA200602442B ZA200602442A ZA200602442A ZA200602442B ZA 200602442 B ZA200602442 B ZA 200602442B ZA 200602442 A ZA200602442 A ZA 200602442A ZA 200602442 A ZA200602442 A ZA 200602442A ZA 200602442 B ZA200602442 B ZA 200602442B
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ZA
South Africa
Prior art keywords
ethyl
pyridin
piperidin
ureido
benzenesulfonamide
Prior art date
Application number
ZA200602442A
Other languages
English (en)
Inventor
Mathys Boris
Scherz Michael
Clozel Martine
Bur Daniel
Mueller Claus
Weller Thomas
Joerg Velker
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of ZA200602442B publication Critical patent/ZA200602442B/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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ZA200602442A 2003-09-26 2006-03-24 Pyridine derivatives and use thereof as urotensin II antagonists ZA200602442B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP0310746 2003-09-26

Publications (1)

Publication Number Publication Date
ZA200602442B true ZA200602442B (en) 2007-09-26

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ID=34384524

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ZA200602442A ZA200602442B (en) 2003-09-26 2006-03-24 Pyridine derivatives and use thereof as urotensin II antagonists

Country Status (18)

Country Link
US (1) US7750161B2 (https=)
EP (1) EP1670470B1 (https=)
JP (1) JP4851328B2 (https=)
KR (1) KR20070014108A (https=)
CN (1) CN1856305B (https=)
AR (1) AR045949A1 (https=)
AT (1) ATE427748T1 (https=)
AU (1) AU2004275488A1 (https=)
BR (1) BRPI0414777A (https=)
CA (1) CA2540196C (https=)
DE (1) DE602004020486D1 (https=)
IL (1) IL174497A0 (https=)
MX (1) MXPA06003264A (https=)
NO (1) NO20061395L (https=)
RU (1) RU2006113948A (https=)
TW (1) TW200526630A (https=)
WO (1) WO2005030209A1 (https=)
ZA (1) ZA200602442B (https=)

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NO20061395L (no) 2006-06-22
JP4851328B2 (ja) 2012-01-11
RU2006113948A (ru) 2007-11-10
CN1856305B (zh) 2010-04-28
DE602004020486D1 (de) 2009-05-20
CA2540196C (en) 2012-03-20
ATE427748T1 (de) 2009-04-15
MXPA06003264A (es) 2006-06-08
AU2004275488A1 (en) 2005-04-07
WO2005030209A1 (en) 2005-04-07
CA2540196A1 (en) 2005-04-07
CN1856305A (zh) 2006-11-01
WO2005030209A8 (en) 2006-05-11
US20070043081A1 (en) 2007-02-22
AR045949A1 (es) 2005-11-16
US7750161B2 (en) 2010-07-06
BRPI0414777A (pt) 2006-11-21
EP1670470A1 (en) 2006-06-21
JP2007506692A (ja) 2007-03-22
TW200526630A (en) 2005-08-16
EP1670470B1 (en) 2009-04-08
IL174497A0 (en) 2006-08-01
KR20070014108A (ko) 2007-01-31

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