ZA200600291B - Anthranylamide pyridones that inhibit VEGFR-2 and VEGFR-3 - Google Patents
Anthranylamide pyridones that inhibit VEGFR-2 and VEGFR-3 Download PDFInfo
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- ZA200600291B ZA200600291B ZA200600291A ZA200600291A ZA200600291B ZA 200600291 B ZA200600291 B ZA 200600291B ZA 200600291 A ZA200600291 A ZA 200600291A ZA 200600291 A ZA200600291 A ZA 200600291A ZA 200600291 B ZA200600291 B ZA 200600291B
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Classifications
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- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D213/63—One oxygen atom
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Landscapes
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- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Dermatology (AREA)
- Ophthalmology & Optometry (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Diabetes (AREA)
- Surgery (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Vascular Medicine (AREA)
- Pain & Pain Management (AREA)
- Physical Education & Sports Medicine (AREA)
- Transplantation (AREA)
- Gastroenterology & Hepatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10327719A DE10327719A1 (de) | 2003-06-13 | 2003-06-13 | VEGFR-2 und VEGFR-3 Inhibitorische Anthranylamidpyridone |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200600291B true ZA200600291B (en) | 2007-03-28 |
Family
ID=33520741
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200600291A ZA200600291B (en) | 2003-06-13 | 2006-01-12 | Anthranylamide pyridones that inhibit VEGFR-2 and VEGFR-3 |
Country Status (18)
| Country | Link |
|---|---|
| EP (1) | EP1633713A1 (zh) |
| JP (1) | JP2006527228A (zh) |
| KR (1) | KR20060021887A (zh) |
| CN (1) | CN1805936A (zh) |
| AU (1) | AU2004247377A1 (zh) |
| BR (1) | BRPI0411360A (zh) |
| CA (1) | CA2526041A1 (zh) |
| CR (1) | CR8127A (zh) |
| DE (1) | DE10327719A1 (zh) |
| EA (1) | EA200501885A1 (zh) |
| EC (1) | ECSP066280A (zh) |
| IL (1) | IL171898A0 (zh) |
| MX (1) | MXPA05013586A (zh) |
| NO (1) | NO20060196L (zh) |
| RS (1) | RS20050831A (zh) |
| UA (1) | UA81323C2 (zh) |
| WO (1) | WO2004111005A1 (zh) |
| ZA (1) | ZA200600291B (zh) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR20060071812A (ko) * | 2004-12-22 | 2006-06-27 | 주식회사 엘지생명과학 | 신규한 3-(2-아미노-6-피리디닐)-4-히드록시페닐 아민유도체 |
| JP6069356B2 (ja) * | 2012-01-05 | 2017-02-01 | クラノテク・アクチボラグ | 線維症又は線維症関連疾患の治療に使用するための、抗血管新生性のインテグリンα５β１阻害剤であるキノリン化合物 |
| CN106496107A (zh) * | 2016-08-31 | 2017-03-15 | 浙江永宁药业股份有限公司 | Vegfr‑2抑制剂及其制备方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9824579D0 (en) * | 1998-11-10 | 1999-01-06 | Novartis Ag | Organic compounds |
| UA71587C2 (uk) * | 1998-11-10 | 2004-12-15 | Шерінг Акцієнгезелльшафт | Аміди антранілової кислоти та їхнє застосування як лікарських засобів |
| DE10023486C1 (de) * | 2000-05-09 | 2002-03-14 | Schering Ag | Ortho substituierte Anthranilsäureamide und deren Verwendung als Arzneimittel |
| US20040254185A1 (en) * | 2001-05-08 | 2004-12-16 | Alexander Ernst | Selective anthranilamide pyridine amides as inhibitors of vegfr-2 and vegfr-3 |
| GB0126902D0 (en) * | 2001-11-08 | 2002-01-02 | Novartis Ag | Organic compounds |
| DE10228090A1 (de) * | 2002-06-19 | 2004-01-15 | Schering Ag | Ausgewählte Anthranylamidpyridinamide und deren Verwendung als Arzneimittel |
-
2003
- 2003-06-13 DE DE10327719A patent/DE10327719A1/de not_active Ceased
-
2004
- 2004-06-09 RS YUP-2005/0831A patent/RS20050831A/sr unknown
- 2004-06-09 WO PCT/EP2004/006236 patent/WO2004111005A1/de active Application Filing
- 2004-06-09 JP JP2006515873A patent/JP2006527228A/ja active Pending
- 2004-06-09 EA EA200501885A patent/EA200501885A1/ru unknown
- 2004-06-09 MX MXPA05013586A patent/MXPA05013586A/es unknown
- 2004-06-09 CA CA002526041A patent/CA2526041A1/en not_active Abandoned
- 2004-06-09 BR BRPI0411360-8A patent/BRPI0411360A/pt not_active IP Right Cessation
- 2004-06-09 AU AU2004247377A patent/AU2004247377A1/en not_active Abandoned
- 2004-06-09 KR KR1020057023901A patent/KR20060021887A/ko not_active Application Discontinuation
- 2004-06-09 EP EP04739742A patent/EP1633713A1/de not_active Withdrawn
- 2004-06-09 CN CNA2004800163643A patent/CN1805936A/zh active Pending
- 2004-09-06 UA UAA200512752A patent/UA81323C2/uk unknown
-
2005
- 2005-11-10 IL IL171898A patent/IL171898A0/en unknown
- 2005-12-09 CR CR8127A patent/CR8127A/es not_active Application Discontinuation
-
2006
- 2006-01-12 ZA ZA200600291A patent/ZA200600291B/en unknown
- 2006-01-12 NO NO20060196A patent/NO20060196L/no not_active Application Discontinuation
- 2006-01-12 EC EC2006006280A patent/ECSP066280A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU2004247377A1 (en) | 2004-12-23 |
| RS20050831A (sr) | 2008-04-04 |
| WO2004111005A1 (de) | 2004-12-23 |
| MXPA05013586A (es) | 2006-03-09 |
| UA81323C2 (en) | 2007-12-25 |
| DE10327719A1 (de) | 2005-01-20 |
| KR20060021887A (ko) | 2006-03-08 |
| JP2006527228A (ja) | 2006-11-30 |
| CN1805936A (zh) | 2006-07-19 |
| BRPI0411360A (pt) | 2006-07-25 |
| ECSP066280A (es) | 2006-07-28 |
| CR8127A (es) | 2006-05-29 |
| CA2526041A1 (en) | 2004-12-23 |
| IL171898A0 (en) | 2006-04-10 |
| NO20060196L (no) | 2006-01-12 |
| EP1633713A1 (de) | 2006-03-15 |
| EA200501885A1 (ru) | 2006-06-30 |
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