ZA200503873B - Carbostyril derivatives and serotonin reuptake inhibitors for treatment of mood disorders - Google Patents
Carbostyril derivatives and serotonin reuptake inhibitors for treatment of mood disorders Download PDFInfo
- Publication number
- ZA200503873B ZA200503873B ZA200503873A ZA200503873A ZA200503873B ZA 200503873 B ZA200503873 B ZA 200503873B ZA 200503873 A ZA200503873 A ZA 200503873A ZA 200503873 A ZA200503873 A ZA 200503873A ZA 200503873 B ZA200503873 B ZA 200503873B
- Authority
- ZA
- South Africa
- Prior art keywords
- aripiprazole
- disorder
- serotonin reuptake
- composition
- depression
- Prior art date
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- 229960002675 xylitol Drugs 0.000 description 1
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Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/138—Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
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- A—HUMAN NECESSITIES
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
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- A—HUMAN NECESSITIES
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- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
- A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/4525—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with oxygen as a ring hetero atom
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- A—HUMAN NECESSITIES
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- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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| US47048103P | 2003-05-14 | 2003-05-14 |
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| ZA200503873B true ZA200503873B (en) | 2006-08-30 |
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| JP (1) | JP4284524B2 (ru) |
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| WO (1) | WO2004060374A1 (ru) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| LT1626721T (lt) * | 2003-05-23 | 2017-01-25 | Otsuka Pharmaceutical Co., Ltd. | Karbostirilo dariniai ir nuotaikos stabilizatoriai, skirti nuotaikos sutrikimų gydymui |
| EP1797039A1 (en) * | 2004-09-13 | 2007-06-20 | Matrix Laboratories Ltd | Process for the preparation of polymorphs, solvates of aripiprazole using aripiprazole acid salts |
| RU2007119648A (ru) * | 2004-10-28 | 2008-12-10 | СК Холдингз Ко. | Способ лечения депрессии |
| TWI320783B (en) | 2005-04-14 | 2010-02-21 | Otsuka Pharma Co Ltd | Heterocyclic compound |
| GB2456183A (en) | 2008-01-04 | 2009-07-08 | Gw Pharma Ltd | Anti-psychotic composition comprising cannabinoids and anti-psychotic medicament |
| AR085840A1 (es) | 2011-04-05 | 2013-10-30 | Otsuka Pharma Co Ltd | Medicamento que contiene un compuesto que es 7-[4-(4-benzo[b]tiofen-4-il-piperazin-1-il)butoxi]-1h-quinolin-2-ona |
| JO3227B1 (ar) | 2011-09-08 | 2018-03-08 | Otsuka Pharma Co Ltd | مشتقات بنزو ثيوفين بها استبدال ببرازين كعوامل مضادة للذهان |
| JOP20200109A1 (ar) | 2012-04-23 | 2017-06-16 | Otsuka Pharma Co Ltd | مستحضر قابل للحقن |
| US20150174247A1 (en) | 2012-06-29 | 2015-06-25 | Maruishi Pharmaceutical Co., Ltd. | Oral pharmaceutical preparation of aripiprazole |
| GB2542155B (en) | 2015-09-09 | 2018-08-01 | Gw Pharma Ltd | Use of cannabidiol in the treatment of mental disorders |
| CN111455019A (zh) * | 2018-05-03 | 2020-07-28 | 杭州端丽生物技术有限公司 | 化合物fty720在制备治疗行为和运动异常检测标记物中的应用 |
| JP7211136B2 (ja) * | 2019-02-14 | 2023-01-24 | ニプロ株式会社 | 錠剤、および、その製造方法 |
| EP3970710A4 (en) | 2019-05-13 | 2023-06-14 | VASTHERA Co. Ltd. | PHARMACEUTICAL COMPOSITION FOR THE PREVENTION OR TREATMENT OF DEGENERATIVE BRAIN DISEASES BY ACTIVATION OF AUTOPHAGY |
| KR20200132730A (ko) | 2019-05-15 | 2020-11-25 | 연세대학교 산학협력단 | 오토파지 활성화제를 유효성분으로 포함하는 심뇌혈관 질환의 예방 또는 치료용 조성물 |
| US11080484B1 (en) * | 2020-10-08 | 2021-08-03 | Omniscient Neurotechnology Pty Limited | Natural language processing of electronic records |
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2004
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2005
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2006
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2007
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2008
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-
2010
- 2010-12-16 HK HK10111807.8A patent/HK1145291A1/xx not_active IP Right Cessation
-
2014
- 2014-04-15 US US14/252,907 patent/US9387182B2/en not_active Expired - Lifetime
-
2016
- 2016-06-08 US US15/176,464 patent/US9694009B2/en not_active Expired - Lifetime
-
2017
- 2017-05-25 US US15/604,720 patent/US20170258788A1/en not_active Abandoned
-
2019
- 2019-01-08 US US16/242,315 patent/US20190151308A1/en not_active Abandoned
- 2019-10-28 US US16/664,984 patent/US20200289501A1/en not_active Abandoned
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