ZA200409425B - Secondary amino anilinic piperidines as MCH1 antagonists and uses thereof - Google Patents
Secondary amino anilinic piperidines as MCH1 antagonists and uses thereof Download PDFInfo
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- ZA200409425B ZA200409425B ZA200409425A ZA200409425A ZA200409425B ZA 200409425 B ZA200409425 B ZA 200409425B ZA 200409425 A ZA200409425 A ZA 200409425A ZA 200409425 A ZA200409425 A ZA 200409425A ZA 200409425 B ZA200409425 B ZA 200409425B
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Epidemiology (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Urology & Nephrology (AREA)
- Child & Adolescent Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US18914502A | 2002-07-03 | 2002-07-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200409425B true ZA200409425B (en) | 2006-04-26 |
Family
ID=30114020
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200409425A ZA200409425B (en) | 2002-07-03 | 2004-11-23 | Secondary amino anilinic piperidines as MCH1 antagonists and uses thereof |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US7473698B2 (ja) |
| EP (1) | EP1556351A4 (ja) |
| JP (1) | JP2005532399A (ja) |
| KR (1) | KR20050034710A (ja) |
| CN (1) | CN1319945C (ja) |
| AU (1) | AU2003259098A1 (ja) |
| BR (1) | BR0312257A (ja) |
| CA (1) | CA2485379A1 (ja) |
| EA (1) | EA008826B1 (ja) |
| HK (1) | HK1080471A1 (ja) |
| IL (1) | IL165730A0 (ja) |
| IS (1) | IS7560A (ja) |
| MX (1) | MXPA04012103A (ja) |
| NO (1) | NO20050113L (ja) |
| NZ (1) | NZ536329A (ja) |
| PL (1) | PL373621A1 (ja) |
| UA (1) | UA77536C2 (ja) |
| WO (1) | WO2004005257A1 (ja) |
| ZA (1) | ZA200409425B (ja) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7105544B2 (en) | 2001-07-05 | 2006-09-12 | Synaptic Pharmaceutical Corporation | Substituted alkyl amido piperidines |
| US7199135B2 (en) | 2001-07-05 | 2007-04-03 | H. Lundbeck A/S | Substituted alkyl amido piperidines |
| US20050154020A1 (en) * | 2004-01-14 | 2005-07-14 | Synaptic Pharmaceutical Corporation | 4-Aryl piperidines |
| US20050154022A1 (en) * | 2004-01-14 | 2005-07-14 | H. Lundbeck A/S | 4-aryl piperidines |
| WO2006015279A1 (en) * | 2004-07-28 | 2006-02-09 | Neurogen Corporation | Heterocyclic diamine compounds as ligands of the melanin concentrating hormone receptor useful for the treatment of obesity, diabetes, eating and sexual disorders |
| US20060079683A1 (en) * | 2004-10-08 | 2006-04-13 | Marzabadi Mohammad R | Arylthiobenzylpiperidine derivatives |
| US7329656B2 (en) | 2004-10-08 | 2008-02-12 | H. Lundbeck A/S | Arylthiobenzylpiperidine derivatives |
| US7446204B2 (en) | 2004-10-08 | 2008-11-04 | H. Lundbeck A/S | Amino substituted aryloxybenzylpiperidine derivatives |
| US9452980B2 (en) * | 2009-12-22 | 2016-09-27 | Hoffmann-La Roche Inc. | Substituted benzamides |
| EP3757102A1 (en) | 2016-03-17 | 2020-12-30 | F. Hoffmann-La Roche AG | 5-ethyl-4-methyl-pyrazole-3-carboxamide derivative having activity as agonist of taar |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0223403B1 (en) | 1985-10-25 | 1993-08-04 | Beecham Group Plc | Piperidine derivative, its preparation, and its use as medicament |
| FR2744448B1 (fr) | 1996-02-02 | 1998-04-24 | Pf Medicament | Nouvelles piperidines derivees d'aryl piperazine, ainsi que leur procede de preparation, les compositions pharmaceutiques et leur utilisation comme medicaments |
| TW548271B (en) * | 1996-12-20 | 2003-08-21 | Astra Pharma Inc | Novel piperidine derivatives having an exocyclic double bond with analgesic effects |
| ES2157148B1 (es) * | 1998-11-18 | 2002-03-01 | Faes Fabrica Espanola De Produ | Nuevas piperidinas 4-sustituidas. |
| US6326381B1 (en) * | 1998-12-17 | 2001-12-04 | American Home Products Corporation | Arylpiperidine and aryl-1,2,5,6-tetrahydropyidine amide derivates |
| US20030082623A1 (en) * | 1998-12-31 | 2003-05-01 | Beth Borowsky | DNA encoding a human melanin concentrating hormone receptor (MCH1) and uses thereof |
| EP1246847A2 (en) * | 2000-07-05 | 2002-10-09 | Synaptic Pharmaceutical Corporation | Dna encoding a human melanin concentrating hormone receptor (mch1) and uses thereof |
| JP2004504303A (ja) | 2000-07-05 | 2004-02-12 | シナプティック・ファーマスーティカル・コーポレーション | 選択的メラニン凝集ホルモン−１（ｍｃｈ１）受容体アンタゴニストおよびその使用 |
| JP2005515961A (ja) | 2001-05-22 | 2005-06-02 | ニューロジェン コーポレイション | メラニン凝集ホルモン受容体リガンド：置換１−ベンジル−４−アリールピペラジン類似体 |
| EA005934B1 (ru) | 2001-07-05 | 2005-08-25 | Х. Лундбекк А/С | Замещённые анилиновые пиперидины в качестве селективных антагонистов мсн |
-
2003
- 2003-03-07 UA UA20041210489A patent/UA77536C2/uk unknown
- 2003-07-03 MX MXPA04012103A patent/MXPA04012103A/es active IP Right Grant
- 2003-07-03 BR BR0312257-3A patent/BR0312257A/pt not_active IP Right Cessation
- 2003-07-03 PL PL03373621A patent/PL373621A1/xx not_active Application Discontinuation
- 2003-07-03 JP JP2004520047A patent/JP2005532399A/ja not_active Withdrawn
- 2003-07-03 US US10/518,675 patent/US7473698B2/en not_active Expired - Fee Related
- 2003-07-03 NZ NZ536329A patent/NZ536329A/en unknown
- 2003-07-03 CN CNB038157667A patent/CN1319945C/zh not_active Expired - Fee Related
- 2003-07-03 EP EP03763374A patent/EP1556351A4/en not_active Withdrawn
- 2003-07-03 KR KR1020057000078A patent/KR20050034710A/ko not_active Application Discontinuation
- 2003-07-03 IL IL16573003A patent/IL165730A0/xx unknown
- 2003-07-03 AU AU2003259098A patent/AU2003259098A1/en not_active Abandoned
- 2003-07-03 WO PCT/US2003/021391 patent/WO2004005257A1/en active Application Filing
- 2003-07-03 CA CA002485379A patent/CA2485379A1/en not_active Abandoned
- 2003-07-03 EA EA200500152A patent/EA008826B1/ru not_active IP Right Cessation
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2004
- 2004-11-23 ZA ZA200409425A patent/ZA200409425B/en unknown
- 2004-11-26 IS IS7560A patent/IS7560A/is unknown
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2005
- 2005-01-10 NO NO20050113A patent/NO20050113L/no not_active Application Discontinuation
-
2006
- 2006-01-09 HK HK06100334A patent/HK1080471A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| UA77536C2 (en) | 2006-12-15 |
| IL165730A0 (en) | 2006-01-15 |
| EA008826B1 (ru) | 2007-08-31 |
| WO2004005257A1 (en) | 2004-01-15 |
| CN1319945C (zh) | 2007-06-06 |
| EP1556351A4 (en) | 2007-07-25 |
| MXPA04012103A (es) | 2005-04-19 |
| US20050245743A1 (en) | 2005-11-03 |
| US7473698B2 (en) | 2009-01-06 |
| EP1556351A1 (en) | 2005-07-27 |
| BR0312257A (pt) | 2005-04-12 |
| EA200500152A1 (ru) | 2005-06-30 |
| NO20050113L (no) | 2005-01-10 |
| IS7560A (is) | 2004-11-26 |
| PL373621A1 (en) | 2005-09-05 |
| CN1665786A (zh) | 2005-09-07 |
| CA2485379A1 (en) | 2004-01-15 |
| KR20050034710A (ko) | 2005-04-14 |
| AU2003259098A1 (en) | 2004-01-23 |
| NZ536329A (en) | 2007-06-29 |
| JP2005532399A (ja) | 2005-10-27 |
| HK1080471A1 (en) | 2006-04-28 |
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