ZA200407461B - Carboxylic acid compounds and drugs containing the compounds as the active ingredient. - Google Patents
Carboxylic acid compounds and drugs containing the compounds as the active ingredient. Download PDFInfo
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- ZA200407461B ZA200407461B ZA200407461A ZA200407461A ZA200407461B ZA 200407461 B ZA200407461 B ZA 200407461B ZA 200407461 A ZA200407461 A ZA 200407461A ZA 200407461 A ZA200407461 A ZA 200407461A ZA 200407461 B ZA200407461 B ZA 200407461B
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- -1 Carboxylic acid compounds Chemical class 0.000 title claims abstract description 59
- 150000001875 compounds Chemical class 0.000 title claims abstract description 41
- 239000003814 drug Substances 0.000 title description 5
- 239000004480 active ingredient Substances 0.000 title description 4
- 229940079593 drug Drugs 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 claims abstract description 33
- 201000010099 disease Diseases 0.000 claims abstract description 21
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- 208000035475 disorder Diseases 0.000 claims abstract description 12
- 208000010668 atopic eczema Diseases 0.000 claims abstract description 11
- 206010012438 Dermatitis atopic Diseases 0.000 claims abstract description 9
- 206010039085 Rhinitis allergic Diseases 0.000 claims abstract description 9
- 208000024780 Urticaria Diseases 0.000 claims abstract description 9
- 201000010105 allergic rhinitis Diseases 0.000 claims abstract description 9
- 201000008937 atopic dermatitis Diseases 0.000 claims abstract description 9
- 206010010744 Conjunctivitis allergic Diseases 0.000 claims abstract description 8
- 206010061218 Inflammation Diseases 0.000 claims abstract description 8
- 208000002205 allergic conjunctivitis Diseases 0.000 claims abstract description 8
- 208000006673 asthma Diseases 0.000 claims abstract description 8
- 208000024998 atopic conjunctivitis Diseases 0.000 claims abstract description 8
- 230000004054 inflammatory process Effects 0.000 claims abstract description 8
- 208000030603 inherited susceptibility to asthma Diseases 0.000 claims abstract description 8
- 206010006482 Bronchospasm Diseases 0.000 claims abstract description 7
- 201000008736 Systemic mastocytosis Diseases 0.000 claims abstract description 7
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Classifications
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- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
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- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/12—Radicals substituted by oxygen atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
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- C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
- C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D307/80—Radicals substituted by oxygen atoms
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D327/00—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms
- C07D327/02—Heterocyclic compounds containing rings having oxygen and sulfur atoms as the only ring hetero atoms one oxygen atom and one sulfur atom
- C07D327/06—Six-membered rings
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
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- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Heart & Thoracic Surgery (AREA)
- Diabetes (AREA)
- Rheumatology (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Ophthalmology & Optometry (AREA)
- Hematology (AREA)
- Gastroenterology & Hepatology (AREA)
- Transplantation (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Toxicology (AREA)
- Otolaryngology (AREA)
- Anesthesiology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2002076456 | 2002-03-19 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200407461B true ZA200407461B (en) | 2005-07-01 |
Family
ID=28035445
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200407461A ZA200407461B (en) | 2002-03-19 | 2004-09-16 | Carboxylic acid compounds and drugs containing the compounds as the active ingredient. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US7351705B2 (fr) |
| EP (1) | EP1486491B1 (fr) |
| JP (2) | JP4547913B2 (fr) |
| KR (1) | KR20040095302A (fr) |
| CN (1) | CN100378083C (fr) |
| AT (1) | ATE516277T1 (fr) |
| AU (1) | AU2003221325A1 (fr) |
| BR (1) | BR0308518A (fr) |
| CA (1) | CA2479352A1 (fr) |
| ES (1) | ES2365985T3 (fr) |
| IL (1) | IL164094A0 (fr) |
| MX (1) | MXPA04009095A (fr) |
| NO (1) | NO20043894L (fr) |
| NZ (1) | NZ535309A (fr) |
| PL (1) | PL372466A1 (fr) |
| RU (1) | RU2329256C2 (fr) |
| WO (1) | WO2003078409A1 (fr) |
| ZA (1) | ZA200407461B (fr) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003297398B2 (en) | 2002-12-20 | 2009-09-24 | Amgen Inc. | Asthma and allergic inflammation modulators |
| AR041089A1 (es) | 2003-05-15 | 2005-05-04 | Merck & Co Inc | Procedimiento y composiciones farmaceutiicas para tratar aterosclerosis, dislipidemias y afecciones relacionadas |
| TWI341838B (en) * | 2003-09-17 | 2011-05-11 | Ono Pharmaceutical Co | Carboxylic acid compound and pharmaceutical composition containg same as active ingredient |
| PE20050483A1 (es) | 2003-10-31 | 2005-08-25 | Arena Pharm Inc | Derivados de tetrazol de formula (i), sus composiciones farmaceuticas y procesos para producir composiciones farmaceuticas |
| US20070244107A1 (en) * | 2004-08-25 | 2007-10-18 | Waters M Gerard | Method of Treating Atherosclerosis, Dyslipidemias and Related Conditions |
| CN101056635A (zh) * | 2004-11-04 | 2007-10-17 | 默克公司 | 烟酸受体激动剂、含有该化合物的组合物及治疗方法 |
| WO2006052798A2 (fr) * | 2004-11-08 | 2006-05-18 | Merck & Co., Inc. | Methode de traitement des rougeurs pathologiques |
| WO2006057922A2 (fr) * | 2004-11-23 | 2006-06-01 | Merck & Co., Inc. | Agonistes des recepteurs de la niacine, compositions contenant ces composes et methodes de traitement |
| PE20060949A1 (es) | 2004-12-23 | 2006-10-11 | Arena Pharm Inc | Derivados fusionados de pirazol como agonistas del receptor de niacina |
| WO2006068162A1 (fr) * | 2004-12-24 | 2006-06-29 | Shionogi & Co., Ltd. | Agent thérapeutique pour le traitement de la bronchopneumopathie chronique obstructive |
| CA2598273A1 (fr) * | 2005-02-17 | 2006-08-24 | Merck & Co., Inc. | Methode de traitement de l'atherosclerose, de dyslipidemies et de troubles lies |
| RU2405770C2 (ru) * | 2005-09-27 | 2010-12-10 | Сионоги Энд Ко., Лтд. | Производное сульфонамида, обладающее антагонистической активностью в отношении рецептора pgd2 |
| EP2037967B1 (fr) | 2006-06-16 | 2016-12-07 | The Trustees Of The University Of Pennsylvania | Antagonistes du récepteur de prostaglandine d2 pour le traitement de l'alopecie androgène |
| US20100260841A1 (en) * | 2007-02-08 | 2010-10-14 | Paolini John F | Method of Treating Atherosclerosis, Dyslipidemias and Related Conditions |
| TWI410410B (zh) * | 2007-08-10 | 2013-10-01 | Ono Pharmaceutical Co | Phenylacetic acid compounds |
| GB0721611D0 (en) * | 2007-11-02 | 2007-12-12 | Glaxo Group Ltd | Novel compounds |
| CN101903338A (zh) | 2007-12-19 | 2010-12-01 | 安姆根有限公司 | 用作炎症调节剂的苯基乙酸衍生物 |
| WO2010030360A1 (fr) * | 2008-09-11 | 2010-03-18 | Arena Pharmaceuticals, Inc. | Dérivés 3h-imidazo[4,5-b]pyridin-5-ol utiles dans le traitement de troubles du récepteur gpr81 |
| CA2776242C (fr) * | 2009-10-08 | 2014-09-02 | Sanofi | Derives de phenyloxadiazole en tant qu'inhibiteurs de pgds |
| SG11202102566YA (en) * | 2018-09-20 | 2021-04-29 | Ono Pharmaceutical Co | Dp antagonist |
| EP3960730A4 (fr) * | 2019-04-26 | 2023-02-08 | Nissan Chemical Corporation | Procédé de production d'un composé de type ester d'acide arylsulfonique |
| WO2021187547A1 (fr) * | 2020-03-19 | 2021-09-23 | 小野薬品工業株式会社 | Cristal de composé de phénylacétate |
| JP7047954B2 (ja) * | 2020-03-19 | 2022-04-05 | 小野薬品工業株式会社 | フェニル酢酸化合物を含有する医薬組成物 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0218728A1 (fr) * | 1985-04-03 | 1987-04-22 | Yamanouchi Pharmaceutical Co. Ltd. | Derives d'phenylene |
| BR9714016A (pt) * | 1996-12-13 | 2000-02-29 | Shionogi & Co | Derivados de benzotiofenocarboxamida e antagonistas a pgd2, que compreendem os mesmos |
| BR0109050A (pt) * | 2000-03-09 | 2004-04-27 | Ono Pharmaceutical Co | Derivados de indol, processo para prepapação e uso dos mesmos |
-
2003
- 2003-03-06 MX MXPA04009095A patent/MXPA04009095A/es active IP Right Grant
- 2003-03-06 ES ES03710260T patent/ES2365985T3/es not_active Expired - Lifetime
- 2003-03-06 IL IL16409403A patent/IL164094A0/xx unknown
- 2003-03-06 AU AU2003221325A patent/AU2003221325A1/en not_active Abandoned
- 2003-03-06 NZ NZ535309A patent/NZ535309A/en unknown
- 2003-03-06 BR BR0308518-0A patent/BR0308518A/pt not_active IP Right Cessation
- 2003-03-06 AT AT03710260T patent/ATE516277T1/de not_active IP Right Cessation
- 2003-03-06 WO PCT/JP2003/002635 patent/WO2003078409A1/fr active Application Filing
- 2003-03-06 JP JP2003576415A patent/JP4547913B2/ja not_active Expired - Fee Related
- 2003-03-06 US US10/507,885 patent/US7351705B2/en not_active Expired - Fee Related
- 2003-03-06 CN CNB03811495XA patent/CN100378083C/zh not_active Expired - Fee Related
- 2003-03-06 EP EP03710260A patent/EP1486491B1/fr not_active Expired - Lifetime
- 2003-03-06 KR KR10-2004-7014688A patent/KR20040095302A/ko not_active Application Discontinuation
- 2003-03-06 RU RU2004130837/04A patent/RU2329256C2/ru not_active IP Right Cessation
- 2003-03-06 CA CA002479352A patent/CA2479352A1/fr not_active Abandoned
- 2003-03-06 PL PL03372466A patent/PL372466A1/xx not_active Application Discontinuation
-
2004
- 2004-09-16 ZA ZA200407461A patent/ZA200407461B/en unknown
- 2004-09-17 NO NO20043894A patent/NO20043894L/no not_active Application Discontinuation
-
2010
- 2010-04-30 JP JP2010105565A patent/JP5168315B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| US7351705B2 (en) | 2008-04-01 |
| RU2004130837A (ru) | 2005-05-27 |
| EP1486491A4 (fr) | 2006-02-15 |
| CN100378083C (zh) | 2008-04-02 |
| JP4547913B2 (ja) | 2010-09-22 |
| WO2003078409A1 (fr) | 2003-09-25 |
| JP5168315B2 (ja) | 2013-03-21 |
| NZ535309A (en) | 2006-05-26 |
| EP1486491B1 (fr) | 2011-07-13 |
| AU2003221325A1 (en) | 2003-09-29 |
| RU2329256C2 (ru) | 2008-07-20 |
| KR20040095302A (ko) | 2004-11-12 |
| US20050222216A1 (en) | 2005-10-06 |
| MXPA04009095A (es) | 2004-12-06 |
| IL164094A0 (en) | 2005-12-18 |
| ES2365985T3 (es) | 2011-10-14 |
| ATE516277T1 (de) | 2011-07-15 |
| CA2479352A1 (fr) | 2003-09-25 |
| PL372466A1 (en) | 2005-07-25 |
| CN1656085A (zh) | 2005-08-17 |
| JPWO2003078409A1 (ja) | 2005-07-14 |
| JP2010189431A (ja) | 2010-09-02 |
| EP1486491A1 (fr) | 2004-12-15 |
| BR0308518A (pt) | 2005-02-22 |
| NO20043894L (no) | 2004-12-17 |
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