ZA200303203B - Antiinflammation agents. - Google Patents
Antiinflammation agents. Download PDFInfo
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- ZA200303203B ZA200303203B ZA200303203A ZA200303203A ZA200303203B ZA 200303203 B ZA200303203 B ZA 200303203B ZA 200303203 A ZA200303203 A ZA 200303203A ZA 200303203 A ZA200303203 A ZA 200303203A ZA 200303203 B ZA200303203 B ZA 200303203B
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Classifications
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- C07—ORGANIC CHEMISTRY
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- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
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- C07—ORGANIC CHEMISTRY
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Landscapes
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Applications Claiming Priority (1)
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Publications (1)
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| CA2427284A1 (en) | 2000-10-26 | 2002-05-30 | Tularik Inc. | Antiinflammation agents |
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| US7176314B2 (en) | 2001-12-05 | 2007-02-13 | Amgen, Inc. | Inflammation modulators |
| ME00355B (me) | 2002-06-06 | 2010-06-30 | Ptp Group Ltd | Kristalisan polietilen tereftalat, koji sadrži silicijum, i postupak za njegovo dobijanje |
| CA2502429A1 (en) | 2002-10-31 | 2004-05-21 | Amgen Inc. | Antiinflammation agents |
| WO2004060308A2 (en) | 2002-12-27 | 2004-07-22 | Chiron Corporation | Thiosemicarbazones as anti-virals and immunopotentiators |
| CA2534127A1 (en) | 2003-07-31 | 2005-02-10 | Boehringer Ingelheim Pharmaceuticals, Inc. | Substituted benzothiophene compounds and uses thereof |
| GB0400895D0 (en) * | 2004-01-15 | 2004-02-18 | Smithkline Beecham Corp | Chemical compounds |
| PE20060373A1 (es) * | 2004-06-24 | 2006-04-29 | Smithkline Beecham Corp | Derivados 3-piperidinil-7-carboxamida-indazol como inhibidores de la actividad cinasa de ikk2 |
| PE20060748A1 (es) | 2004-09-21 | 2006-10-01 | Smithkline Beecham Corp | Derivados de indolcarboxamida como inhibidores de quinasa ikk2 |
| JP5253159B2 (ja) * | 2005-06-24 | 2013-07-31 | デューク・ユニヴァーシティ | 熱応答性バイオポリマーに基づく直接的ドラッグデリバリーシステム |
| US8063071B2 (en) | 2007-10-31 | 2011-11-22 | GlaxoSmithKline, LLC | Chemical compounds |
| UA99699C2 (ru) | 2005-06-30 | 2012-09-25 | Смитклайн Бичам Корпорейшн | Производные индолкарбоксамида и фармацевтическая композиция, которая их содержит |
| EP1948187A4 (de) * | 2005-11-18 | 2010-11-03 | Glaxosmithkline Llc | Chemische verbindungen |
| GB0523576D0 (en) * | 2005-11-18 | 2005-12-28 | Theradeas Ltd | Drug composition and its use in therapy |
| US7592353B2 (en) | 2006-06-06 | 2009-09-22 | Boehringer Ingelheim International Gmbh | Substituted 3-amino-thieno[2,3-b]pyridine-2-carboxylic acid amide compounds and processes for preparing and their uses |
| DE102007012794B3 (de) * | 2007-03-16 | 2008-06-19 | Novaled Ag | Pyrido[3,2-h]chinazoline und/oder deren 5,6-Dihydroderivate, deren Herstellungsverfahren und diese enthaltendes dotiertes organisches Halbleitermaterial |
| PE20081889A1 (es) | 2007-03-23 | 2009-03-05 | Smithkline Beecham Corp | Indol carboxamidas como inhibidores de ikk2 |
| EP2154965A4 (de) * | 2007-05-29 | 2011-08-17 | Glaxosmithkline Llc | Naphthyridinderivate als p13-kinasehemmer |
| CA2721927C (en) | 2008-04-21 | 2014-01-28 | Otonomy, Inc. | Auris formulations for treating otic diseases and conditions |
| US11969501B2 (en) | 2008-04-21 | 2024-04-30 | Dompé Farmaceutici S.P.A. | Auris formulations for treating otic diseases and conditions |
| WO2010038465A1 (ja) * | 2008-10-02 | 2010-04-08 | 旭化成ファーマ株式会社 | ８位置換イソキノリン誘導体及びその用途 |
| JP2012520257A (ja) | 2009-03-10 | 2012-09-06 | グラクソ グループ リミテッド | Ｉｋｋ２阻害剤としてのインドール誘導体 |
| US9527829B2 (en) | 2013-03-14 | 2016-12-27 | Celgene Quanticel Research, Inc. | Histone demethylase inhibitors |
| CN107073006A (zh) | 2014-09-16 | 2017-08-18 | 赛尔基因昆蒂赛尔研究公司 | 组蛋白脱甲基酶抑制剂 |
| US9896436B2 (en) | 2014-09-16 | 2018-02-20 | Celgene Quanticel Research, Inc. | Histone demethylase inhibitors |
| US11192859B2 (en) * | 2016-04-18 | 2021-12-07 | New York University | Quinoline compounds as modulators of RAGE activity and uses thereof |
| CA3029281A1 (en) | 2016-06-29 | 2018-01-04 | Otonomy, Inc. | Triglyceride otic formulations and uses thereof |
| US20220274929A1 (en) * | 2019-02-25 | 2022-09-01 | The Regents Of The University Of California | Thiosemicarbazone compounds and uses thereof |
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| ATE289295T1 (de) * | 1997-04-22 | 2005-03-15 | Euro Celtique Sa | Die verwendung von durch carbozyklische und heterozyklische reste substituierte semicarbazonen und thiosemicarbazonen als natriumkanalblocker |
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| US6613942B1 (en) * | 1997-07-01 | 2003-09-02 | Novo Nordisk A/S | Glucagon antagonists/inverse agonists |
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| US6258822B1 (en) * | 1997-08-06 | 2001-07-10 | Abbott Laboratories | Urokinase inhibitors |
| BR0012450B1 (pt) | 1999-06-23 | 2011-08-23 | benzimidazóis substituìdos. | |
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| WO2001068648A1 (en) | 2000-03-15 | 2001-09-20 | Aventis Pharma Deutschland Gmbh | Substituted beta-carbolines with ikb-kinase inhibiting activity |
| JP4272338B2 (ja) | 2000-09-22 | 2009-06-03 | バイエル アクチェンゲゼルシャフト | ピリジン誘導体 |
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| CA2427284A1 (en) | 2000-10-26 | 2002-05-30 | Tularik Inc. | Antiinflammation agents |
| JP2002193938A (ja) | 2000-12-01 | 2002-07-10 | Bayer Ag | ４−アリールピリジン誘導体 |
| US7122544B2 (en) | 2000-12-06 | 2006-10-17 | Signal Pharmaceuticals, Llc | Anilinopyrimidine derivatives as IKK inhibitors and compositions and methods related thereto |
| CZ20032287A3 (cs) | 2001-02-01 | 2004-02-18 | Bristol-Myers Squibb Company | Způsoby léčení zánětlivých a imunitních nemocí za použití inhibitorů IkB kinázy (IKK) |
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- 2001-10-23 PL PL01366114A patent/PL366114A1/xx unknown
- 2001-10-23 MX MXPA03003599A patent/MXPA03003599A/es active IP Right Grant
- 2001-10-23 AU AU2002239806A patent/AU2002239806B2/en not_active Ceased
- 2001-10-23 AU AU3980602A patent/AU3980602A/xx active Pending
- 2001-10-23 EA EA200300508A patent/EA200300508A1/ru unknown
- 2001-10-23 CN CN01821344.8A patent/CN1503673A/zh active Pending
- 2001-10-23 NZ NZ525474A patent/NZ525474A/en unknown
- 2001-10-23 BR BR0114978-4A patent/BR0114978A/pt not_active IP Right Cessation
- 2001-10-23 JP JP2002544024A patent/JP4285602B2/ja not_active Expired - Fee Related
- 2001-10-23 ES ES01987605T patent/ES2305125T3/es not_active Expired - Lifetime
- 2001-10-23 AT AT01987605T patent/ATE392898T1/de not_active IP Right Cessation
- 2001-10-29 AR ARP010105038A patent/AR035499A1/es not_active Application Discontinuation
-
2003
- 2003-04-24 ZA ZA200303203A patent/ZA200303203B/en unknown
- 2003-04-25 NO NO20031869A patent/NO20031869L/no not_active Application Discontinuation
-
2004
- 2004-08-26 US US10/928,784 patent/US7186841B2/en not_active Expired - Fee Related
-
2007
- 2007-01-05 US US11/650,268 patent/US20070135464A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| AU2002239806B2 (en) | 2007-01-18 |
| JP4285602B2 (ja) | 2009-06-24 |
| EP1333834B1 (de) | 2008-04-23 |
| EP1333834A2 (de) | 2003-08-13 |
| NZ525474A (en) | 2005-10-28 |
| ES2305125T3 (es) | 2008-11-01 |
| WO2002041843A3 (en) | 2003-02-06 |
| DE60133758T2 (de) | 2009-07-02 |
| US6846834B2 (en) | 2005-01-25 |
| CA2427284A1 (en) | 2002-05-30 |
| KR20030064773A (ko) | 2003-08-02 |
| AU2002239806B8 (en) | 2002-06-03 |
| IL155519A0 (en) | 2003-11-23 |
| US7186841B2 (en) | 2007-03-06 |
| JP2004516252A (ja) | 2004-06-03 |
| CN1503673A (zh) | 2004-06-09 |
| MXPA03003599A (es) | 2003-08-01 |
| US20020161004A1 (en) | 2002-10-31 |
| NO20031869L (no) | 2003-06-26 |
| WO2002041843A2 (en) | 2002-05-30 |
| US20070135464A1 (en) | 2007-06-14 |
| EP1333834A4 (de) | 2007-01-17 |
| US20050043330A1 (en) | 2005-02-24 |
| PL366114A1 (en) | 2005-01-24 |
| ATE392898T1 (de) | 2008-05-15 |
| BR0114978A (pt) | 2004-04-20 |
| AR035499A1 (es) | 2004-06-02 |
| NO20031869D0 (no) | 2003-04-25 |
| EA200300508A1 (ru) | 2004-06-24 |
| DE60133758D1 (de) | 2008-06-05 |
| AU3980602A (en) | 2002-06-03 |
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