ZA200207413B - Compositions containing alpha-2-adrenergic agonist components. - Google Patents
Compositions containing alpha-2-adrenergic agonist components. Download PDFInfo
- Publication number
- ZA200207413B ZA200207413B ZA200207413A ZA200207413A ZA200207413B ZA 200207413 B ZA200207413 B ZA 200207413B ZA 200207413 A ZA200207413 A ZA 200207413A ZA 200207413 A ZA200207413 A ZA 200207413A ZA 200207413 B ZA200207413 B ZA 200207413B
- Authority
- ZA
- South Africa
- Prior art keywords
- composition
- component
- alpha
- solubility
- adrenergic agonist
- Prior art date
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- 239000000384 adrenergic alpha-2 receptor agonist Substances 0.000 title claims description 88
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- FEWJPZIEWOKRBE-JCYAYHJZSA-N Dextrotartaric acid Chemical compound OC(=O)[C@H](O)[C@@H](O)C(O)=O FEWJPZIEWOKRBE-JCYAYHJZSA-N 0.000 claims description 13
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Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/498—Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
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- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
- A61K31/716—Glucans
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K31/74—Synthetic polymeric materials
- A61K31/765—Polymers containing oxygen
- A61K31/78—Polymers containing oxygen of acrylic acid or derivatives thereof
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- A—HUMAN NECESSITIES
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- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
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- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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TW (1) | TWI287998B (hu) |
WO (1) | WO2002005853A2 (hu) |
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DE69909768T2 (de) | 1998-04-07 | 2004-06-17 | Alcon Manufacturing Ltd., Fort Worth | Xanthangummi enthaltende gelbildende ophthalmische zusammensetzungen |
WO2000012137A1 (en) * | 1998-09-02 | 2000-03-09 | Allergan Sales, Inc. | Preserved cyclodextrin-containing compositions |
ATE289804T1 (de) | 1998-10-08 | 2005-03-15 | Hampar L Karagoezian | Synergistische antimikrobielle. dermatologische und ophtahalmologische zubereitungen, die ein chlorit und wasserstoffperoxid enthalten |
IN185228B (hu) * | 1999-02-03 | 2000-12-09 | Bakulesh Mafatlal Dr Khamar | |
PT2153819E (pt) * | 2000-07-14 | 2012-11-14 | Allergan Inc | Utilização de um componente para aumento de solubilidade numa composição aquosa compreendendo tartarato de brimonidina |
NZ521185A (en) * | 2000-07-14 | 2005-02-25 | Allergan Inc | Compositions containing alpha-2-adrenergic agonist components |
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2001
- 2001-07-09 NZ NZ521185A patent/NZ521185A/en not_active IP Right Cessation
- 2001-07-09 KR KR1020027014270A patent/KR100757656B1/ko active IP Right Grant
- 2001-07-09 CN CNB018073395A patent/CN100569291C/zh not_active Expired - Lifetime
- 2001-07-09 CN CN200910247188.9A patent/CN101897704B/zh not_active Expired - Lifetime
- 2001-07-09 JP JP2002511784A patent/JP4927298B2/ja not_active Expired - Lifetime
- 2001-07-09 BR BR0109317-7A patent/BR0109317A/pt not_active Application Discontinuation
- 2001-07-09 RU RU2003101321/15A patent/RU2311928C2/ru active
- 2001-07-09 PL PL36070701A patent/PL360707A1/xx not_active Application Discontinuation
- 2001-07-09 HU HU0303197A patent/HUP0303197A3/hu not_active Application Discontinuation
- 2001-07-09 IL IL15153001A patent/IL151530A0/xx unknown
- 2001-07-09 MX MXPA02008930A patent/MXPA02008930A/es active IP Right Grant
- 2001-07-09 AU AU7326901A patent/AU7326901A/xx active Pending
- 2001-07-09 EP EP01952528A patent/EP1365811A2/en not_active Ceased
- 2001-07-09 WO PCT/US2001/021552 patent/WO2002005853A2/en active IP Right Grant
- 2001-07-09 AU AU2001273269A patent/AU2001273269B2/en not_active Expired
- 2001-07-09 CA CA002402405A patent/CA2402405C/en not_active Expired - Lifetime
- 2001-07-10 US US09/904,018 patent/US6627210B2/en not_active Expired - Lifetime
- 2001-07-13 TW TW090117220A patent/TWI287998B/zh not_active IP Right Cessation
- 2001-07-13 AR ARP010103344A patent/AR033539A1/es not_active Application Discontinuation
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2002
- 2002-08-28 IL IL151530A patent/IL151530A/en unknown
- 2002-09-04 NO NO20024221A patent/NO333367B1/no not_active IP Right Cessation
- 2002-09-06 US US10/236,566 patent/US6641834B2/en not_active Expired - Lifetime
- 2002-09-16 ZA ZA200207413A patent/ZA200207413B/en unknown
- 2002-11-19 US US10/299,386 patent/US6673337B2/en not_active Expired - Lifetime
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2003
- 2003-10-22 US US10/691,912 patent/US20040063689A1/en not_active Abandoned
-
2004
- 2004-05-18 HK HK04103520.9A patent/HK1060519A1/xx not_active IP Right Cessation
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2008
- 2008-06-02 JP JP2008144707A patent/JP2008231122A/ja active Pending
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2011
- 2011-12-27 JP JP2011286579A patent/JP2012067128A/ja active Pending
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