ZA200104620B - Benzoxazole derivatives and medicaments comprising said derivatives as active ingredient. - Google Patents

Benzoxazole derivatives and medicaments comprising said derivatives as active ingredient. Download PDF

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Publication number
ZA200104620B
ZA200104620B ZA200104620A ZA200104620A ZA200104620B ZA 200104620 B ZA200104620 B ZA 200104620B ZA 200104620 A ZA200104620 A ZA 200104620A ZA 200104620 A ZA200104620 A ZA 200104620A ZA 200104620 B ZA200104620 B ZA 200104620B
Authority
ZA
South Africa
Prior art keywords
group
homopiperazinyl
chloro
lower alkyl
alkyl group
Prior art date
Application number
ZA200104620A
Other languages
English (en)
Inventor
Sojiro Shiokawa
Yasuo Sato
Masaaki Izumi
Satoshi Yoshida
Hiroshi Murakami
Tomoko Ito
Tetsutaro Niisato
Original Assignee
Meiji Seika Kaisha
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Meiji Seika Kaisha filed Critical Meiji Seika Kaisha
Publication of ZA200104620B publication Critical patent/ZA200104620B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ZA200104620A 1998-11-20 2001-06-06 Benzoxazole derivatives and medicaments comprising said derivatives as active ingredient. ZA200104620B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP33127498 1998-11-20

Publications (1)

Publication Number Publication Date
ZA200104620B true ZA200104620B (en) 2002-02-04

Family

ID=18241866

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200104620A ZA200104620B (en) 1998-11-20 2001-06-06 Benzoxazole derivatives and medicaments comprising said derivatives as active ingredient.

Country Status (23)

Country Link
US (1) US7045516B1 (fr)
EP (1) EP1134220B1 (fr)
JP (1) JP4557112B2 (fr)
KR (1) KR100675033B1 (fr)
CN (1) CN1333771A (fr)
AT (1) ATE273974T1 (fr)
AU (1) AU753797B2 (fr)
BR (1) BR9916793A (fr)
CA (1) CA2351446A1 (fr)
CZ (1) CZ20011700A3 (fr)
DE (1) DE69919575T2 (fr)
ES (1) ES2222763T3 (fr)
HU (1) HUP0104238A3 (fr)
ID (1) ID30143A (fr)
IL (1) IL143178A0 (fr)
NO (1) NO20012443L (fr)
PL (1) PL348426A1 (fr)
RU (1) RU2204558C2 (fr)
SK (1) SK6772001A3 (fr)
TR (1) TR200101945T2 (fr)
TW (1) TW520370B (fr)
WO (1) WO2000031073A1 (fr)
ZA (1) ZA200104620B (fr)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6660858B2 (en) * 2001-03-28 2003-12-09 Lion Bioscience Ag 2-aminobenzoxazole derivatives and combinatorial libraries thereof
GB0203061D0 (en) * 2002-02-08 2002-03-27 Novartis Ag Organic compounds
AU2003252738A1 (en) * 2002-08-09 2004-02-25 Ajinomoto Co., Inc. Remedy for intestinal diseases and visceral pain
WO2007005780A2 (fr) * 2005-07-01 2007-01-11 Dynogen Pharmaceuticals, Inc. Compositions et procédés permettant de traite l'hypomotilité du système digestif et des troubles associés
AU2007229492B2 (en) * 2006-03-28 2011-11-03 High Point Pharmaceuticals, Llc Benzothiazoles having histamine H3 receptor activity
WO2010048514A1 (fr) * 2008-10-23 2010-04-29 Albany Molecular Research, Inc. Synthèse de composés de 2-amino-benzoxazole
KR101579688B1 (ko) 2014-07-08 2015-12-24 재단법인 전남생물산업진흥원 좁쌀풀 추출물을 유효성분으로 함유하는 과민성 대장증후군에 의한 내장 통증 억제예방 또는 치료용 약학 조성물
CA3182245A1 (fr) * 2020-06-12 2021-12-16 Jae Hee Cheon Composition pharmaceutique comprenant un compose derive de benzimidazole

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3193560B2 (ja) * 1993-04-16 2001-07-30 明治製菓株式会社 新規ベンゾオキサゾール誘導体
JP3520177B2 (ja) * 1996-05-09 2004-04-19 明治製菓株式会社 セロトニン5−ht3受容体部分活性薬

Also Published As

Publication number Publication date
PL348426A1 (en) 2002-05-20
DE69919575D1 (de) 2004-09-23
TR200101945T2 (tr) 2001-11-21
RU2204558C2 (ru) 2003-05-20
DE69919575T2 (de) 2005-09-29
KR20010086448A (ko) 2001-09-12
CZ20011700A3 (cs) 2001-10-17
TW520370B (en) 2003-02-11
KR100675033B1 (ko) 2007-01-29
CA2351446A1 (fr) 2000-06-02
HUP0104238A3 (en) 2003-05-28
EP1134220A4 (fr) 2001-12-19
WO2000031073A1 (fr) 2000-06-02
US7045516B1 (en) 2006-05-16
CN1333771A (zh) 2002-01-30
NO20012443D0 (no) 2001-05-18
BR9916793A (pt) 2001-11-13
ID30143A (id) 2001-11-08
JP4557112B2 (ja) 2010-10-06
NO20012443L (no) 2001-07-12
SK6772001A3 (en) 2001-12-03
AU753797B2 (en) 2002-10-31
AU1185000A (en) 2000-06-13
EP1134220B1 (fr) 2004-08-18
EP1134220A1 (fr) 2001-09-19
IL143178A0 (en) 2002-04-21
ES2222763T3 (es) 2005-02-01
HUP0104238A2 (en) 2002-08-28
ATE273974T1 (de) 2004-09-15

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