YU51701A - Postupak za dobijanje jedinjenja pirazola/4,3-d/ pirimidin-7-ona i njihovih derivata - Google Patents
Postupak za dobijanje jedinjenja pirazola/4,3-d/ pirimidin-7-ona i njihovih derivataInfo
- Publication number
- YU51701A YU51701A YU51701A YUP51701A YU51701A YU 51701 A YU51701 A YU 51701A YU 51701 A YU51701 A YU 51701A YU P51701 A YUP51701 A YU P51701A YU 51701 A YU51701 A YU 51701A
- Authority
- YU
- Yugoslavia
- Prior art keywords
- compounds
- pyrazolo
- pyrimidin
- intermediates
- preparation
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- 239000000543 intermediate Substances 0.000 title 1
- WAJNANMQOPCIPO-UHFFFAOYSA-N pyrazolo[4,3-d]pyrimidin-7-one Chemical class O=C1N=CN=C2C=NN=C12 WAJNANMQOPCIPO-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- XLYOFNOQVPJJNP-UHFFFAOYSA-M hydroxide Chemical compound [OH-] XLYOFNOQVPJJNP-UHFFFAOYSA-M 0.000 abstract 1
- 150000004679 hydroxides Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Gynecology & Obstetrics (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0018660A GB0018660D0 (en) | 2000-07-28 | 2000-07-28 | Pharmaceutically active compounds |
| GB0107526A GB0107526D0 (en) | 2001-03-26 | 2001-03-26 | Process for the preparation of pyrazolo [4,3-d] pyrimidin-7-one compounds and intermediates thereof |
| GB0110251A GB0110251D0 (en) | 2001-04-26 | 2001-04-26 | Process for the preparation of pyrazolo[4,4-d]Pyrimidin-7-one compounds and intermediates thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| YU51701A true YU51701A (sh) | 2003-12-31 |
Family
ID=27255823
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| YU51701A YU51701A (sh) | 2000-07-28 | 2001-07-17 | Postupak za dobijanje jedinjenja pirazola/4,3-d/ pirimidin-7-ona i njihovih derivata |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP1176147A1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP2002105076A (cg-RX-API-DMAC7.html) |
| KR (1) | KR20020010102A (cg-RX-API-DMAC7.html) |
| CN (1) | CN1335317A (cg-RX-API-DMAC7.html) |
| AR (1) | AR035650A1 (cg-RX-API-DMAC7.html) |
| AU (1) | AU754962B2 (cg-RX-API-DMAC7.html) |
| BR (1) | BR0103072A (cg-RX-API-DMAC7.html) |
| CA (1) | CA2354175A1 (cg-RX-API-DMAC7.html) |
| CZ (1) | CZ20012713A3 (cg-RX-API-DMAC7.html) |
| HK (1) | HK1040715A1 (cg-RX-API-DMAC7.html) |
| HU (1) | HUP0103075A3 (cg-RX-API-DMAC7.html) |
| IL (1) | IL144516A0 (cg-RX-API-DMAC7.html) |
| IN (1) | IN191315B (cg-RX-API-DMAC7.html) |
| MX (1) | MXPA01007676A (cg-RX-API-DMAC7.html) |
| PL (1) | PL348935A1 (cg-RX-API-DMAC7.html) |
| RU (1) | RU2224759C2 (cg-RX-API-DMAC7.html) |
| YU (1) | YU51701A (cg-RX-API-DMAC7.html) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0106631D0 (en) * | 2001-03-16 | 2001-05-09 | Pfizer Ltd | Pharmaceutically active compounds |
| US6831074B2 (en) | 2001-03-16 | 2004-12-14 | Pfizer Inc | Pharmaceutically active compounds |
| KR100824193B1 (ko) | 2003-04-29 | 2008-04-21 | 화이자 인코포레이티드 | 고혈압 치료에 유용한5,7-디아미노피라졸로[4,3-d]피리미딘 |
| JP2006219373A (ja) | 2003-06-13 | 2006-08-24 | Daiichi Asubio Pharma Co Ltd | Pde7阻害作用を有するピリジニルピラゾロピリミジノン誘導体 |
| US7572799B2 (en) | 2003-11-24 | 2009-08-11 | Pfizer Inc | Pyrazolo[4,3-d]pyrimidines as Phosphodiesterase Inhibitors |
| BRPI0509731A (pt) | 2004-04-07 | 2007-09-25 | Pfizer | pirazol[4,3-d]pirimidinas |
| JP5254029B2 (ja) * | 2005-11-16 | 2013-08-07 | エフ.ホフマン−ラ ロシュ アーゲー | Thocの新規製造方法 |
| CA2645893A1 (en) * | 2006-03-17 | 2007-09-27 | Cipla Limited | Synthesis of 4-[1-(4-cyano phenyl)-(1,2,4-tr1azol-1-yl)methyl] benzonitrile and 4-[1-(1h-1,2,4-triazol-1-yl)methylene benzonitrile intermediate |
| US7638541B2 (en) | 2006-12-28 | 2009-12-29 | Metabolex Inc. | 5-ethyl-2-{4-[4-(4-tetrazol-1-yl-phenoxymethyl)-thiazol-2-yl]-piperidin-1-yl}-pyrimidine |
| KR20100033419A (ko) | 2007-07-19 | 2010-03-29 | 메타볼렉스, 인코포레이티드 | 당뇨병 및 대사 장애의 치료를 위한 rup3 또는 gpr119 수용체의 작용제로서 n-아자시클릭 치환된 피롤, 피라졸, 이미다졸, 트리아졸 및 테트라졸 유도체 |
| CN102666553B (zh) | 2009-10-01 | 2015-05-06 | 赛马拜制药公司 | 取代的四唑-1-基-苯氧基甲基-噻唑-2-基-哌啶基-嘧啶盐 |
| ES2676209T3 (es) | 2010-06-23 | 2018-07-17 | Metabolex Inc. | Composiciones de 5-etil-2-{4-[4-(4-tetrazol-1-il-fenoximetil)-tiazol-2-il]-piperidin-1-il}-pirimidina |
| CN109862896A (zh) | 2016-08-03 | 2019-06-07 | 西玛贝医药公司 | 用于治疗炎症性胃肠疾病或胃肠病症的氧亚甲基芳基化合物 |
| CN119677737A (zh) | 2022-04-22 | 2025-03-21 | 沃泰克斯药物股份有限公司 | 用于治疗疼痛的杂芳基化合物 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2089971A (en) * | 1937-08-17 | Condensation products of | ||
| GB9013750D0 (en) * | 1990-06-20 | 1990-08-08 | Pfizer Ltd | Therapeutic agents |
| GB9114760D0 (en) * | 1991-07-09 | 1991-08-28 | Pfizer Ltd | Therapeutic agents |
| GB9612514D0 (en) * | 1996-06-14 | 1996-08-14 | Pfizer Ltd | Novel process |
| GB9822238D0 (en) * | 1998-10-12 | 1998-12-09 | Pfizer Ltd | Process for preparation of pyrazolo[4,3-D]pyrimidin-7-ones and intermediates thereof |
| GB9823101D0 (en) * | 1998-10-23 | 1998-12-16 | Pfizer Ltd | Pharmaceutically active compounds |
| CZ20021151A3 (cs) * | 1999-10-11 | 2003-03-12 | Pfizer Inc. | 5-(2-substituovaný-5-heterocyklylsulfonylpyrid-3-yl)-dihydropyrazolo[4,3-d]-pyrimidin-7-ony jako inhibitory fosfodiesterasy |
-
2001
- 2001-07-17 EP EP01306123A patent/EP1176147A1/en not_active Withdrawn
- 2001-07-17 YU YU51701A patent/YU51701A/sh unknown
- 2001-07-20 IN IN698MU2001 patent/IN191315B/en unknown
- 2001-07-23 IL IL14451601A patent/IL144516A0/xx unknown
- 2001-07-25 CZ CZ20012713A patent/CZ20012713A3/cs unknown
- 2001-07-26 PL PL01348935A patent/PL348935A1/xx not_active Application Discontinuation
- 2001-07-26 AR ARP010103577A patent/AR035650A1/es not_active Application Discontinuation
- 2001-07-26 AU AU57672/01A patent/AU754962B2/en not_active Ceased
- 2001-07-26 CA CA002354175A patent/CA2354175A1/en not_active Abandoned
- 2001-07-27 MX MXPA01007676A patent/MXPA01007676A/es unknown
- 2001-07-27 RU RU2001121162/04A patent/RU2224759C2/ru not_active IP Right Cessation
- 2001-07-27 KR KR1020010045414A patent/KR20020010102A/ko not_active Ceased
- 2001-07-27 CN CN01124351A patent/CN1335317A/zh active Pending
- 2001-07-27 HU HU0103075A patent/HUP0103075A3/hu unknown
- 2001-07-30 BR BR0103072-8A patent/BR0103072A/pt not_active IP Right Cessation
- 2001-07-30 JP JP2001229348A patent/JP2002105076A/ja active Pending
-
2002
- 2002-04-03 HK HK02102460.5A patent/HK1040715A1/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MXPA01007676A (es) | 2002-10-23 |
| EP1176147A1 (en) | 2002-01-30 |
| RU2224759C2 (ru) | 2004-02-27 |
| CA2354175A1 (en) | 2002-01-28 |
| CZ20012713A3 (cs) | 2002-04-17 |
| HK1040715A1 (zh) | 2002-06-21 |
| HUP0103075A2 (hu) | 2002-07-29 |
| CN1335317A (zh) | 2002-02-13 |
| AR035650A1 (es) | 2004-06-23 |
| PL348935A1 (en) | 2002-02-11 |
| HU0103075D0 (en) | 2001-10-28 |
| JP2002105076A (ja) | 2002-04-10 |
| KR20020010102A (ko) | 2002-02-02 |
| IN191315B (cg-RX-API-DMAC7.html) | 2003-11-22 |
| AU754962B2 (en) | 2002-11-28 |
| HUP0103075A3 (en) | 2003-04-28 |
| AU5767201A (en) | 2002-01-31 |
| IL144516A0 (en) | 2002-05-23 |
| BR0103072A (pt) | 2002-04-09 |
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