YU39155B - Process for obtaining 2-(4-aroylpiperazine-1-yl)-4-amino-6,7-dimethoxy quinazolines - Google Patents

Process for obtaining 2-(4-aroylpiperazine-1-yl)-4-amino-6,7-dimethoxy quinazolines

Info

Publication number
YU39155B
YU39155B YU02096/77A YU209677A YU39155B YU 39155 B YU39155 B YU 39155B YU 02096/77 A YU02096/77 A YU 02096/77A YU 209677 A YU209677 A YU 209677A YU 39155 B YU39155 B YU 39155B
Authority
YU
Yugoslavia
Prior art keywords
aroylpiperazine
amino
obtaining
quinazolines
dimethoxy
Prior art date
Application number
YU02096/77A
Other languages
English (en)
Other versions
YU209677A (en
Inventor
P D Hammen
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of YU209677A publication Critical patent/YU209677A/xx
Publication of YU39155B publication Critical patent/YU39155B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
YU02096/77A 1976-09-20 1977-09-02 Process for obtaining 2-(4-aroylpiperazine-1-yl)-4-amino-6,7-dimethoxy quinazolines YU39155B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/724,707 US4062844A (en) 1976-09-20 1976-09-20 Process for preparing hypotensive 2-(4-aroylpiperazin-1-yl)-amino-6,7-dimethoxyquinazolines

Publications (2)

Publication Number Publication Date
YU209677A YU209677A (en) 1982-06-30
YU39155B true YU39155B (en) 1984-06-30

Family

ID=24911552

Family Applications (1)

Application Number Title Priority Date Filing Date
YU02096/77A YU39155B (en) 1976-09-20 1977-09-02 Process for obtaining 2-(4-aroylpiperazine-1-yl)-4-amino-6,7-dimethoxy quinazolines

Country Status (32)

Country Link
US (1) US4062844A (ru)
JP (1) JPS5337676A (ru)
AR (1) AR213659A1 (ru)
AT (1) AT357542B (ru)
AU (1) AU500908B2 (ru)
BE (1) BE858844A (ru)
BG (1) BG28054A3 (ru)
CA (1) CA1068699A (ru)
CH (1) CH632507A5 (ru)
CS (1) CS203172B2 (ru)
DD (1) DD132661A5 (ru)
DE (1) DE2740331C3 (ru)
DK (1) DK143340C (ru)
ES (1) ES462146A1 (ru)
FI (1) FI66610C (ru)
FR (1) FR2364918A1 (ru)
GB (1) GB1543668A (ru)
GR (1) GR69792B (ru)
HK (1) HK31181A (ru)
HU (1) HU180041B (ru)
IE (1) IE45966B1 (ru)
LU (1) LU78149A1 (ru)
MY (1) MY8100266A (ru)
NL (1) NL189132C (ru)
NO (1) NO147423C (ru)
PL (1) PL105830B1 (ru)
PT (1) PT67006B (ru)
RO (1) RO73051A (ru)
SE (1) SE435381B (ru)
SU (1) SU847919A3 (ru)
YU (1) YU39155B (ru)
ZA (1) ZA775098B (ru)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0022481A1 (en) * 1979-06-21 1981-01-21 Mitsubishi Yuka Pharmaceutical Co., Ltd. 5,6-Alkylenepyrimidine derivatives, processes for preparing the same and pharmaceutical compositions
US4607034A (en) * 1979-10-29 1986-08-19 Mitsubishi Yuka Pharmaceutical Co., Ltd. Quinazoline derivatives and pharmaceutical composition thereof
JPS5793977A (en) * 1980-11-26 1982-06-11 Sankyo Co Ltd Acylaminoquinazoline derivative and its preparation
FI70411C (fi) * 1980-12-29 1986-09-19 Pfizer Foerfarande foer framstaellning av nya antihypertensiva 4-amino-6,7-dimetoxi-2-piperazinokinazolin derivat
US4625012A (en) * 1985-08-26 1986-11-25 Essex Specialty Products, Inc. Moisture curable polyurethane polymers
IT1270993B (it) * 1994-03-18 1997-05-26 Recordati Chem Pharm Derivati chinzolilamminici attivi come alfa-antagonisti
GB9708917D0 (en) * 1997-05-01 1997-06-25 Pfizer Ltd Compounds useful in therapy
US6313294B1 (en) 1998-02-04 2001-11-06 Development Center For Biotechnology Process for preparing amides

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3511836A (en) * 1967-12-13 1970-05-12 Pfizer & Co C 2,4,6,7-tetra substituted quinazolines
US3935213A (en) * 1973-12-05 1976-01-27 Pfizer Inc. Process for hypotensive 4-amino-2-(piperazin-1-yl) quinazoline derivatives

Also Published As

Publication number Publication date
SU847919A3 (ru) 1981-07-15
BE858844A (fr) 1978-03-20
US4062844A (en) 1977-12-13
PT67006B (en) 1979-02-12
AU2822177A (en) 1979-03-01
DE2740331C3 (de) 1981-03-12
DE2740331B2 (de) 1980-06-19
ZA775098B (en) 1978-07-26
CA1068699A (en) 1979-12-25
RO73051A (ro) 1981-09-24
NL189132B (nl) 1992-08-17
FI772629A (fi) 1978-03-21
ATA636877A (de) 1979-12-15
ES462146A1 (es) 1978-06-16
DK395877A (da) 1978-03-21
CS203172B2 (en) 1981-02-27
DD132661A5 (de) 1978-10-18
AR213659A1 (es) 1979-02-28
NL189132C (nl) 1993-01-18
NL7709736A (nl) 1978-03-22
IE45966B1 (en) 1983-01-12
IE45966L (en) 1978-03-20
JPS5337676A (en) 1978-04-06
DK143340C (da) 1981-12-14
MY8100266A (en) 1981-12-31
PT67006A (en) 1977-10-01
SE7708942L (sv) 1978-03-21
GB1543668A (en) 1979-04-04
YU209677A (en) 1982-06-30
NO147423C (no) 1983-04-06
FI66610B (fi) 1984-07-31
GR69792B (ru) 1982-07-07
SE435381B (sv) 1984-09-24
HK31181A (en) 1981-07-10
PL105830B1 (pl) 1979-11-30
AU500908B2 (en) 1979-06-07
NO773073L (no) 1978-03-21
NO147423B (no) 1982-12-27
AT357542B (de) 1980-07-10
BG28054A3 (en) 1980-02-25
FR2364918A1 (fr) 1978-04-14
HU180041B (en) 1983-01-28
DE2740331A1 (de) 1978-03-23
PL200710A1 (pl) 1978-05-22
LU78149A1 (fr) 1979-05-25
FR2364918B1 (ru) 1981-11-20
CH632507A5 (de) 1982-10-15
DK143340B (da) 1981-08-10
FI66610C (fi) 1984-11-12

Similar Documents

Publication Publication Date Title
YU165282A (en) Process for producing 2-piperazinyl-6,7-dimethoxy-quinazoline
YU198482A (en) Process for obtaining quinazoline compounds
YU211479A (en) Process for obtaining 1-phenyl-2-azolyl-4,4-dimeethyl-1-pentene-3-ole
YU312781A (en) Process for obtaining 4-amino-6,7-dimethoxy-2-piperazine quinazoline
YU163577A (en) Process for obtaining 6a,10a-transhexahydro-dibenzo-(b,d)-pyrane-9-one
YU41294B (en) Process for obtaining the crystalline alpha-from of 2-(4(2-furoy)-piperazione-1-yl)-4-amino-6,7-dimethoxy quinazoline hydroclorides
YU211582A (en) Process for obtaining cardiostimulating quinazolines
YU39155B (en) Process for obtaining 2-(4-aroylpiperazine-1-yl)-4-amino-6,7-dimethoxy quinazolines
YU38683A (en) Process for obtaining antihypertensive quinazolines
HU177883B (en) Process for preparing 2-/4-/2-furoyl/-piperazin-1-yl/-4-amino-6,7-dimethoxy-quinazoline
YU40698B (en) Process for preparing 2-(2,2,2-trihaloethy)-4-halocyclobutane-l-ones
YU22980A (en) Process for obtaining quinazolines
BG29871A3 (en) Method for obtaining of 6, 7- dimethoxy- 1, 2, 3, 4- tetrahydro- 1- isohinolylacetamids
YU233278A (en) Process for obtaining quinazoline
YU132777A (en) Process for obtaining quinoxaline-carbazate-1,4-dioxide
YU39397B (en) Process for the manufacture of 2-(4-(2-furoyl)-piperazine-1-yl)-4-amino-6,7-dimethoxy-quinazoline
YU263878A (en) Process for obtaining antihypertensive quinazolines
IT7848092A0 (it) Procedimento per produrre 2,5-diossotetraidrofurano 3-sostituito
PL197861A1 (pl) Sposob wytwarzania 1,3-dwualkilo-5-/2/1,5,5,-trojalkilopirolidynylideno/etylideno/-2-tiohydantoin
NZ183626A (en) 2-(2-(2-aminopyrimid-4-yl)-ehten-1-yl)-quinoxaline-1,4-dioxides
YU41676A (en) Process for obtaining new 6-amino-5-beta, 19-cycloandrostane derivatives
YU113180A (en) Process for obtaining quinazolines
ZA783438B (en) Improved process for preparing quinazolinone oxides