YU34891B - Process for preparing novel racemic or optically active piperazine derivatives and acid addition salts thereof - Google Patents

Process for preparing novel racemic or optically active piperazine derivatives and acid addition salts thereof

Info

Publication number
YU34891B
YU34891B YU60078A YU60078A YU34891B YU 34891 B YU34891 B YU 34891B YU 60078 A YU60078 A YU 60078A YU 60078 A YU60078 A YU 60078A YU 34891 B YU34891 B YU 34891B
Authority
YU
Yugoslavia
Prior art keywords
acid addition
addition salts
optically active
piperazine derivatives
preparing novel
Prior art date
Application number
YU60078A
Other languages
English (en)
Other versions
YU60078A (en
Inventor
Renth Otto Ernst
Otto Ernst Renth
Mentrup Rolf
Rolf Mentrup
Schromm Kurt
Kurt Schromm
Giesemann Rolf
Rolf Giesemann
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Publication of YU60078A publication Critical patent/YU60078A/xx
Publication of YU34891B publication Critical patent/YU34891B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/02—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements
    • C07D295/027—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements containing only one hetero ring
    • C07D295/03—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms containing only hydrogen and carbon atoms in addition to the ring hetero elements containing only one hetero ring with the ring nitrogen atoms directly attached to acyclic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/58—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring other than with oxygen or sulphur atoms in position 2 or 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/56—Radicals substituted by sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/58—Radicals substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D319/00—Heterocyclic compounds containing six-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D319/10—1,4-Dioxanes; Hydrogenated 1,4-dioxanes
    • C07D319/14—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems
    • C07D319/16—1,4-Dioxanes; Hydrogenated 1,4-dioxanes condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D319/18—Ethylenedioxybenzenes, not substituted on the hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
YU60078A 1970-07-30 1978-03-13 Process for preparing novel racemic or optically active piperazine derivatives and acid addition salts thereof YU34891B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2037852A DE2037852C3 (de) 1970-07-30 1970-07-30 Neue Piperazinderivate und Verfahren zu ihrer Herstellung

Publications (2)

Publication Number Publication Date
YU60078A YU60078A (en) 1979-10-31
YU34891B true YU34891B (en) 1980-04-30

Family

ID=5778382

Family Applications (7)

Application Number Title Priority Date Filing Date
YU1986/71A YU34530B (en) 1970-07-30 1971-07-29 Process for preparing novel or optically active piperazine derivatives
YU60078A YU34891B (en) 1970-07-30 1978-03-13 Process for preparing novel racemic or optically active piperazine derivatives and acid addition salts thereof
YU598/78A YU34889B (en) 1970-07-30 1978-03-13 Process for preparing novel racemic or optically active piperazine derivatives and acid addition salts thereof
YU599/78A YU34890B (en) 1970-07-30 1978-03-13 Process for preparing novel racemic or optically active piperazine derivatives and acid addition salts thereof
YU596/78A YU34888B (en) 1970-07-30 1978-03-13 Process for preparing novel racemic or optically active piperazine derivatives and acid addition salts thereof
YU597/78A YU35248B (en) 1970-07-30 1978-03-13 Process for preparing novel racemic or optically active piperazine derivatives
YU01388/78A YU138878A (en) 1970-07-30 1978-06-12 Process for preparing new racemic or optically active piperazine derivatives and acid addition salts thereof

Family Applications Before (1)

Application Number Title Priority Date Filing Date
YU1986/71A YU34530B (en) 1970-07-30 1971-07-29 Process for preparing novel or optically active piperazine derivatives

Family Applications After (5)

Application Number Title Priority Date Filing Date
YU598/78A YU34889B (en) 1970-07-30 1978-03-13 Process for preparing novel racemic or optically active piperazine derivatives and acid addition salts thereof
YU599/78A YU34890B (en) 1970-07-30 1978-03-13 Process for preparing novel racemic or optically active piperazine derivatives and acid addition salts thereof
YU596/78A YU34888B (en) 1970-07-30 1978-03-13 Process for preparing novel racemic or optically active piperazine derivatives and acid addition salts thereof
YU597/78A YU35248B (en) 1970-07-30 1978-03-13 Process for preparing novel racemic or optically active piperazine derivatives
YU01388/78A YU138878A (en) 1970-07-30 1978-06-12 Process for preparing new racemic or optically active piperazine derivatives and acid addition salts thereof

Country Status (19)

Country Link
US (1) US3808212A (xx)
JP (1) JPS5716989B1 (xx)
AT (6) AT311976B (xx)
AU (1) AU463957B2 (xx)
BE (1) BE770800A (xx)
BG (5) BG20370A3 (xx)
CH (6) CH565781A5 (xx)
CS (1) CS172929B2 (xx)
DE (1) DE2037852C3 (xx)
DK (1) DK137990C (xx)
ES (6) ES393738A1 (xx)
FR (1) FR2100972B1 (xx)
GB (1) GB1344720A (xx)
NL (1) NL173643C (xx)
PL (6) PL84349B1 (xx)
RO (6) RO59997A (xx)
SE (2) SE375308B (xx)
SU (4) SU437292A3 (xx)
YU (7) YU34530B (xx)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3940396A (en) * 1973-02-28 1976-02-24 Uniroyal Inc. 1,2,3,4,4A,5,7,7A-Octahydrothieno[3,4-b]pyrazines 6,6-dioxides
US3991036A (en) * 1973-02-28 1976-11-09 Uniroyal Inc. Preparation of polyurethane using 1,2,3,4,4a,5,7,7a-Octahydrothieno[3,4-b]py
GB1407552A (en) * 1973-04-02 1975-09-24 Science Union & Cie Disubstituted piperazines processes for their preparation and pharmaceutical compositions containing them
GB1432660A (en) * 1973-10-30 1976-04-22 Science Union & Cie Piperazine derivatives processes for their preparation and and pharamacueitcal compositions containing them
US3960863A (en) * 1974-06-25 1976-06-01 Sankyo Company Limited Pyrido[1,2-a]pyrimidinone derivatives
DE2604838A1 (de) * 1976-02-07 1977-08-11 Knoll Ag Alkylendioxypiperazinderivate
DE3476196D1 (en) * 1983-01-21 1989-02-23 Fisons Plc Aromatic amines
DE3571436D1 (en) * 1984-12-21 1989-08-17 Duphar Int Res New pharmaceutical compositions having anti-psychotic properties
FR2692264B1 (fr) * 1992-06-12 1994-08-05 Adir Nouvelles piperazines 1,4-disubstituees, leur procede de preparation et les compositions pharmaceutiques les contenant.
FR2734819B1 (fr) * 1995-05-31 1997-07-04 Adir Nouveaux composes de la piperazine, de la piperidine et de la 1,2,5,6-tetrahydropyridine, leur procede de preparation et les compositions pharmaceutiques les contenant
US6002005A (en) * 1995-06-02 1999-12-14 Neurogen Corporation Certain 1-substituted aminomethyl imidazole and pyrrole derivatives: novel dopamine receptor subtype specific ligands
FR2737724B1 (fr) * 1995-08-09 1997-09-05 Synthelabo Derives de 1-[2-(2,3-dihydro-1h-inden-1-yl)ethyl]-4- (naphtalen-1-yl) piperazine, leur preparation et leur application en therapeutique
JPH09124643A (ja) * 1995-08-14 1997-05-13 Bristol Myers Squibb Co 抗うつ作用を有する１−アリールアルキル−４−（アルコキシピリジニル）−又は４−（アルコキシピリミジニル）ピペラジン誘導体
US6040448A (en) * 1997-10-24 2000-03-21 Neurogen Corporation Certain 1-(2-naphthyl) and 1-(2-azanaphthyl)-4-(1-phenylmethyl) piperazines, dopamine receptor subtype specific ligands
MA41169A (fr) * 2014-12-17 2017-10-24 Acraf Composés antibactériens à large spectre d'activité

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL132357C (xx) * 1966-09-03

Also Published As

Publication number Publication date
AU3177271A (en) 1973-02-01
BE770800A (fr) 1972-01-31
ES396215A1 (es) 1974-04-16
YU34888B (en) 1980-04-30
DE2037852B2 (de) 1979-10-11
CH575412A5 (xx) 1976-05-14
AT311986B (de) 1973-12-10
ES396213A1 (es) 1974-04-16
SU437291A3 (ru) 1974-07-25
YU35248B (en) 1980-10-31
BG21029A3 (bg) 1976-01-20
FR2100972B1 (xx) 1974-11-15
ES396212A1 (es) 1974-04-16
SU416945A3 (ru) 1974-02-25
BG19598A3 (xx) 1975-06-25
SE7408533L (xx) 1974-06-27
SU437289A3 (ru) 1974-07-25
BG20370A3 (bg) 1975-11-05
AT311988B (de) 1973-12-10
YU34890B (en) 1980-04-30
PL84348B1 (xx) 1976-03-31
PL84664B1 (xx) 1976-04-30
YU60078A (en) 1979-10-31
ES396216A1 (es) 1974-04-16
PL84349B1 (xx) 1976-03-31
BG20594A3 (xx) 1975-12-05
RO60596A (xx) 1976-08-15
CH565781A5 (xx) 1975-08-29
SU437293A3 (ru) 1974-07-25
YU138878A (en) 1982-10-31
DK137990C (da) 1978-11-13
DE2037852A1 (de) 1972-02-03
DK137990B (da) 1978-06-19
SU440840A3 (xx) 1974-08-25
YU59778A (en) 1980-04-30
RO59997A (xx) 1976-06-15
AU463957B2 (en) 1975-08-14
CH565165A5 (xx) 1975-08-15
CS172929B2 (xx) 1977-01-28
AT311984B (de) 1973-12-10
NL7110538A (xx) 1972-02-01
YU59978A (en) 1979-10-31
SU437290A3 (ru) 1974-07-25
AT311985B (de) 1973-12-10
YU34889B (en) 1980-04-30
ES393738A1 (es) 1974-07-01
NL173643C (nl) 1984-02-16
RO60597A (xx) 1976-08-15
SU437292A3 (ru) 1974-07-25
SE403288B (sv) 1978-08-07
GB1344720A (en) 1974-01-23
CH565166A5 (xx) 1975-08-15
FR2100972A1 (xx) 1972-03-24
YU59878A (en) 1979-10-31
YU59678A (en) 1979-10-31
PL84347B1 (xx) 1976-03-31
DE2037852C3 (de) 1980-06-26
NL173643B (nl) 1983-09-16
AT311987B (de) 1973-12-10
SE375308B (xx) 1975-04-14
US3808212A (en) 1974-04-30
RO61040A (xx) 1976-08-15
CH565167A5 (xx) 1975-08-15
PL84610B1 (xx) 1976-04-30
RO60599A (xx) 1976-08-15
CH565780A5 (xx) 1975-08-29
PL91965B1 (xx) 1977-03-31
ES396214A1 (es) 1974-04-16
JPS5716989B1 (xx) 1982-04-08
YU34530B (en) 1979-09-10
RO60598A (xx) 1976-07-15
AT311976B (de) 1973-12-10
BG20369A3 (bg) 1975-11-05
YU198671A (en) 1979-02-28

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