YU183181A - Process for obtaining a stabilized aqueous ivermection containing formulation - Google Patents

Process for obtaining a stabilized aqueous ivermection containing formulation

Info

Publication number
YU183181A
YU183181A YU01831/81A YU183181A YU183181A YU 183181 A YU183181 A YU 183181A YU 01831/81 A YU01831/81 A YU 01831/81A YU 183181 A YU183181 A YU 183181A YU 183181 A YU183181 A YU 183181A
Authority
YU
Yugoslavia
Prior art keywords
ivermection
obtaining
containing formulation
stabilized aqueous
stabilized
Prior art date
Application number
YU01831/81A
Other languages
English (en)
Inventor
P K A Lo
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of YU183181A publication Critical patent/YU183181A/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Dispersion Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
YU01831/81A 1980-08-04 1981-07-23 Process for obtaining a stabilized aqueous ivermection containing formulation YU183181A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17495780A 1980-08-04 1980-08-04

Publications (1)

Publication Number Publication Date
YU183181A true YU183181A (en) 1984-02-29

Family

ID=22638223

Family Applications (1)

Application Number Title Priority Date Filing Date
YU01831/81A YU183181A (en) 1980-08-04 1981-07-23 Process for obtaining a stabilized aqueous ivermection containing formulation

Country Status (17)

Country Link
EP (1) EP0045655B1 (cg-RX-API-DMAC7.html)
JP (1) JPS5765330A (cg-RX-API-DMAC7.html)
KR (1) KR860001503B1 (cg-RX-API-DMAC7.html)
AR (1) AR229354A1 (cg-RX-API-DMAC7.html)
AT (1) ATE12179T1 (cg-RX-API-DMAC7.html)
AU (1) AU551280B2 (cg-RX-API-DMAC7.html)
CA (1) CA1162857A (cg-RX-API-DMAC7.html)
DE (1) DE3169381D1 (cg-RX-API-DMAC7.html)
DK (1) DK163637C (cg-RX-API-DMAC7.html)
ES (1) ES8607721A1 (cg-RX-API-DMAC7.html)
GR (1) GR74604B (cg-RX-API-DMAC7.html)
IE (1) IE51460B1 (cg-RX-API-DMAC7.html)
NZ (1) NZ197796A (cg-RX-API-DMAC7.html)
OA (1) OA06863A (cg-RX-API-DMAC7.html)
PT (1) PT73471B (cg-RX-API-DMAC7.html)
YU (1) YU183181A (cg-RX-API-DMAC7.html)
ZA (1) ZA815317B (cg-RX-API-DMAC7.html)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
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US4485099A (en) * 1983-06-15 1984-11-27 Merck & Co., Inc. Renin inhibitors containing a C-terminal amide cycle
US4477440A (en) * 1983-09-14 1984-10-16 Merck & Co., Inc. Renin inhibitors containing an n-terminal disulfide cycle
NZ210505A (en) * 1983-12-22 1988-06-30 Merck & Co Inc Parasiticidal compositions containing avermectin or milbemycin derivatives
ZA89552B (en) * 1988-01-29 1989-10-25 Merrell Dow Pharma Pharmaceutical composition for 4-aroylimidazol-2-ones
GB8803836D0 (en) * 1988-02-18 1988-03-16 Glaxo Group Ltd Compositions
JP2680614B2 (ja) * 1988-08-01 1997-11-19 日清製粉株式会社 ダナゾール組成物
NZ335166A (en) 1999-04-14 2001-11-30 Ashmont Holdings Ltd Anthelmintic composition containing triclabendazole in at least one solvent
US5419897A (en) * 1993-04-09 1995-05-30 Buckman Laboratories International, Inc. Ionene polymers as anthelmintics in animals
US5602107A (en) * 1993-05-10 1997-02-11 Merck & Co., Inc. Pour-on formulations consisting of gylcols, glycerides and avermectin compounds
PL174488B1 (pl) * 1993-05-10 1998-08-31 Merck & Co Inc Preparat do zwalczania pasożytów zwierząt oraz sposób wytwarzania preparatu do zwalczania pasożytów zwierząt
DE69432982T2 (de) * 1993-05-10 2004-04-15 Merck & Co., Inc. Pour-on formulierung enthaltend polymerische material, glykole und glyzeriden
JP2855181B2 (ja) 1993-12-10 1999-02-10 敏雄 鈴木 松類の枯損防止用組成物及び防止方法
DE19613972A1 (de) * 1996-04-09 1997-10-16 Bayer Ag Injektionsformulierungen von Avermectinen und Milbemycinen auf Basis von Rizinusöl
DE19638045A1 (de) * 1996-09-18 1998-03-19 Bayer Ag Injektionsformulierungen von Avermectinen und Milbemycinen
MXPA01007486A (es) * 1999-01-25 2003-06-24 Optime Therapeutics Inc Formulaciones de liposomas.
US6780885B1 (en) * 2000-01-14 2004-08-24 Idexx Laboratories, Inc. Formulations and methods for administration of pharmacologically or biologically active compounds
RU2162699C1 (ru) * 2000-02-14 2001-02-10 Закрытое Акционерное Общество "Нита-Фарм" Водно-дисперсная лекарственная форма ивермектина для лечения экто- и эндопаразитозов
BG64140B1 (bg) * 2000-12-21 2004-02-27 "Биовет" Ад Състав за растителна защита с инсектицидно и акарицидно действие
GB2386066A (en) 2002-02-28 2003-09-10 Norbrook Lab Ltd Long-acting parasiticidal composition with improved bioavailability comprising a salicylanilide, a further anti-parasitic compound & a polymeric species
AU2002952597A0 (en) * 2002-11-11 2002-11-28 Schering-Plough Pty. Limited Topical parasiticide formulations and methods of treatment
DE10331253B4 (de) * 2003-01-28 2007-03-08 Alpha-Biocare Gmbh Therapeutika gegen Parasiten von Fischen
FR2854074B1 (fr) 2003-04-24 2007-11-23 Galderma Res & Dev Utilisation de l'ivermectine pour le traitement de desordres dermatologiques
GB0316377D0 (en) 2003-07-12 2003-08-13 Norbrook Lab Ltd Parasiticidal composition
US20080125480A1 (en) * 2004-12-30 2008-05-29 Cheminova A/S Oil-In-Water Formulation Of Avermectins
FR2894823B1 (fr) 2005-12-20 2008-02-29 Galderma Sa Composition de type emulsion inverse comprenant de l'ivermectine, et ses utilisations en cosmetique et en dermatologie
RU2493825C2 (ru) 2008-10-08 2013-09-27 ВАЙЕТ ЭлЭлСи Бензимидазольные антигельминтные композиции
BRPI0804639A2 (pt) * 2008-10-23 2010-07-20 Formil Veterinaria Ltda processo para preparação de formulação de suspensão veterinária para administração de medicamento insolúvel em água, por meio de sistemas de distribuição de água e respectiva formulação de suspensão veterinária para administração de medicamento insolúvel em água
MX2011004442A (es) 2008-10-29 2011-10-14 Topaz Pharmaceuticals Inc Sistema conservante para formulaciones topicas terapeuticas basadas en emulsion.
JP5717034B2 (ja) * 2012-08-27 2015-05-13 丸和バイオケミカル株式会社 マクロライド系化合物を含有する土壌線虫防除用薬剤
EP2966116A4 (en) 2013-03-06 2016-10-19 Sekisui Chemical Co Ltd RESIN COMPOSITE MANUFACTURING METHOD AND RESIN COMPOSITE MATERIAL
US9233117B2 (en) 2013-07-08 2016-01-12 Galderma S. A. Treatment of inflammatory lesions of rosacea with ivermectin
FR3042412A1 (fr) * 2015-10-14 2017-04-21 Biotopic Pharmaceuticals Formulation pharmaceutique stabilisee et prete a l'emploi d'ivermectine dans le traitement des parasitoses humaines et animales
CN107802599A (zh) * 2017-12-08 2018-03-16 宁夏大学 一种驼用饮水型驱虫溶液的研制和使用方法
PT110634B (pt) 2018-03-19 2021-03-17 Hovione Farmaciencia Sa Ivermectina amorfa e processo para a sua produção
CN109966438A (zh) * 2019-05-17 2019-07-05 石家庄九鼎动物药业有限公司 一种兽用抗寄生虫药物伊维菌素注射液及其制备方法
US11077134B1 (en) 2020-11-10 2021-08-03 Mountain Valley Md Inc Water dissolvable macrocyclic lactone cyclodextrin complexes
US11638714B2 (en) 2020-11-10 2023-05-02 Mountain Valley Md Inc Water dissolvable macrocyclic lactone cyclodextrin complexes

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB784659A (en) * 1954-11-26 1957-10-16 Upjohn Co Therapeutic compositions and aqueous suspensions thereof
CH420490A (de) * 1961-10-16 1966-09-15 Hoffmann La Roche Wässriges Verdünnungsmittel zur Herstellung von parenteralen Injektionslösungen und Verfahren zu dessen Herstellung
GB1225979A (cg-RX-API-DMAC7.html) * 1967-03-23 1971-03-24
US4199569A (en) * 1977-10-03 1980-04-22 Merck & Co., Inc. Selective hydrogenation products of C-076 compounds and derivatives thereof

Also Published As

Publication number Publication date
AU551280B2 (en) 1986-04-24
ZA815317B (en) 1983-03-30
ES8607721A1 (es) 1986-06-01
EP0045655A2 (en) 1982-02-10
AU7361281A (en) 1982-02-11
IE51460B1 (en) 1986-12-24
PT73471A (en) 1981-09-01
DE3169381D1 (en) 1985-04-25
KR830005849A (ko) 1983-09-14
EP0045655B1 (en) 1985-03-20
DK163637B (da) 1992-03-23
ATE12179T1 (de) 1985-04-15
NZ197796A (en) 1984-11-09
JPS5765330A (en) 1982-04-20
PT73471B (en) 1983-07-06
DK345081A (da) 1982-02-05
JPH057371B2 (cg-RX-API-DMAC7.html) 1993-01-28
CA1162857A (en) 1984-02-28
GR74604B (cg-RX-API-DMAC7.html) 1984-06-29
DK163637C (da) 1992-08-17
AR229354A1 (es) 1983-07-29
KR860001503B1 (ko) 1986-09-30
IE811751L (en) 1982-02-04
OA06863A (fr) 1983-02-28
EP0045655A3 (en) 1982-10-06
ES504513A0 (es) 1986-06-01

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