YU171880A - Process for obtaining new indolizine derivatives - Google Patents

Process for obtaining new indolizine derivatives

Info

Publication number
YU171880A
YU171880A YU01718/80A YU171880A YU171880A YU 171880 A YU171880 A YU 171880A YU 01718/80 A YU01718/80 A YU 01718/80A YU 171880 A YU171880 A YU 171880A YU 171880 A YU171880 A YU 171880A
Authority
YU
Yugoslavia
Prior art keywords
obtaining new
indolizine derivatives
new indolizine
derivatives
obtaining
Prior art date
Application number
YU01718/80A
Other languages
English (en)
Inventor
G Rosseels
P Nokin
Original Assignee
Labaz Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Labaz Nv filed Critical Labaz Nv
Publication of YU171880A publication Critical patent/YU171880A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
YU01718/80A 1979-07-06 1980-07-01 Process for obtaining new indolizine derivatives YU171880A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7923599 1979-07-06

Publications (1)

Publication Number Publication Date
YU171880A true YU171880A (en) 1983-10-31

Family

ID=10506339

Family Applications (1)

Application Number Title Priority Date Filing Date
YU01718/80A YU171880A (en) 1979-07-06 1980-07-01 Process for obtaining new indolizine derivatives

Country Status (24)

Country Link
US (1) US4400387A (cs)
EP (1) EP0022762B1 (cs)
JP (1) JPS5618979A (cs)
AR (1) AR225314A1 (cs)
AT (1) AT375078B (cs)
AU (1) AU529725B2 (cs)
CA (1) CA1153379A (cs)
DD (1) DD151940A5 (cs)
DE (1) DE3060097D1 (cs)
DK (1) DK146962C (cs)
ES (1) ES493139A0 (cs)
FI (1) FI67217C (cs)
GR (1) GR69280B (cs)
HU (1) HU182151B (cs)
IE (1) IE49994B1 (cs)
IN (1) IN151594B (cs)
NO (1) NO153496C (cs)
NZ (1) NZ193926A (cs)
OA (1) OA06563A (cs)
PL (1) PL125597B1 (cs)
PT (1) PT71424A (cs)
SU (1) SU993817A3 (cs)
YU (1) YU171880A (cs)
ZA (1) ZA803434B (cs)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6103702A (en) * 1999-05-24 2000-08-15 Board Of Trustees Of The University Of Illinois Use of adenosine deaminase inhibitors to treat systemic inflammatory response syndrome
EP1200102A1 (en) * 1999-07-22 2002-05-02 Supergen, Inc. Methods for treating autoimmune diseases
FR2805460A1 (fr) 2000-02-25 2001-08-31 Oreal Compositions de teinture des fibres keratiniques contenant des derives d'indolizine cationiques et procede de teinture
FR2838123B1 (fr) * 2002-04-04 2005-06-10 Sanofi Synthelabo Nouveaux derives d'indolozine-1,2,3 substituee, inhibiteurs selectifs du b-fgf
JP4048166B2 (ja) * 2002-11-18 2008-02-13 三井製糖株式会社 血糖値上昇抑制剤及び体脂肪蓄積抑制剤並びに食用材料
FR2859997B1 (fr) * 2003-09-18 2006-02-03 Sanofi Synthelabo Nouveaux derives d'indolizine 1,2,3,6,7,8 substituee, inhibiteurs des fgfs, leur procede de preparation et les compositions pharmaceutiques les contenant.
AR051780A1 (es) * 2004-11-29 2007-02-07 Japan Tobacco Inc Compuestos en anillo fusionados que contienen nitrogeno y utilizacion de los mismos
FR2896247B1 (fr) 2006-01-13 2008-02-29 Sanofi Aventis Sa Composes dimeres agonistes des recepteurs des fgfs (fgfrs), leur procede de preparation et leur application en therapeutique
WO2010113942A1 (ja) * 2009-03-31 2010-10-07 キッセイ薬品工業株式会社 インドリジン誘導体及びその医薬用途
US20100261666A1 (en) * 2009-04-14 2010-10-14 The Board Of Trustees Of The University Of Illinois Compositions and methods for the treatment of myocardial dysfunction associated with sirs or sepsis
ES2549926T3 (es) * 2010-09-29 2015-11-03 Kissei Pharmaceutical Co., Ltd. Derivados (aza)indolizínicos como inhibidores de la xantina-oxidasa
DK3348557T3 (da) * 2015-09-10 2020-07-20 Jiangsu Atom Bioscience And Pharmaceutical Co Ltd Imidazo[1,2-a]pyridiner til behandling eller forebyggelse af hyperurekæmi eller gigt
CN108084186B (zh) 2016-11-16 2021-06-25 江苏新元素医药科技有限公司 Urat1抑制剂及其应用
WO2018090921A1 (zh) 2016-11-16 2018-05-24 江苏新元素医药科技有限公司 Urat1抑制剂及其应用
CN108727267B (zh) * 2017-05-26 2022-05-13 江苏新元素医药科技有限公司 一类urat1抑制剂及其应用
EP3632904B1 (en) * 2017-05-26 2022-04-20 Jiangsu Atom Bioscience and Pharmaceutical Co., Ltd. Urat1 inhibitors for promoting uric acid excretion
KR102750849B1 (ko) * 2018-01-19 2025-01-08 쑤저우 시노벤트 파마슈티칼즈 씨오., 엘티디. 헤테로시클릭 화합물, 제조 방법 및 의약품에서의 이의 용도
CN110283167A (zh) * 2018-11-14 2019-09-27 贵州省中国科学院天然产物化学重点实验室 一种抗心率失常药物布托普洛嗪的制备方法
WO2022169974A1 (en) 2021-02-05 2022-08-11 Nexys Therapeutics, Inc. Inhibitors of urat1 and pharmaceutical uses thereof
WO2023221078A1 (en) * 2022-05-20 2023-11-23 Jiangsu Atom Bioscience And Pharmaceutical Co., Ltd. Solid forms of a compound for treating or preventing hyperuricemia or gout
WO2025237171A1 (zh) * 2024-05-11 2025-11-20 广州市联瑞制药有限公司 嘧啶并五元氮杂环酚类化合物及其应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SU430639A1 (ru) 1972-06-05 1978-02-28 Московский Ордена Ленина И Ордена Трудового Красного Знамени Государственный Университет Им.М.В.Ломоносова Способ получени 1-пиридилиндолизинов
FI61030C (fi) * 1976-02-19 1982-05-10 Sanofi Sa Foerfarande foer framstaellning av terapeutiskt verkande 2-substituerade-1- eller 3-benzoyl-indolizinderivat
GB1518443A (en) * 1976-02-19 1978-07-19 Labaz Indolizine derivatives and process for preparing the same

Also Published As

Publication number Publication date
IE801349L (en) 1981-01-06
EP0022762B1 (fr) 1981-11-25
EP0022762A1 (fr) 1981-01-21
PL225479A1 (cs) 1981-10-30
DK291180A (da) 1981-01-07
DD151940A5 (de) 1981-11-11
IN151594B (cs) 1983-06-04
US4400387A (en) 1983-08-23
AR225314A1 (es) 1982-03-15
DK146962C (da) 1984-08-06
ES8105710A1 (es) 1981-06-16
NZ193926A (en) 1984-05-31
OA06563A (fr) 1981-07-31
CA1153379A (en) 1983-09-06
ZA803434B (en) 1981-05-27
ATA354380A (de) 1983-11-15
DK146962B (da) 1984-02-27
AT375078B (de) 1984-06-25
AU529725B2 (en) 1983-06-16
ES493139A0 (es) 1981-06-16
DE3060097D1 (en) 1982-01-28
JPS5618979A (en) 1981-02-23
FI67217B (fi) 1984-10-31
HU182151B (en) 1983-12-28
AU5948780A (en) 1981-01-15
GR69280B (cs) 1982-05-13
NO802015L (no) 1981-01-07
FI802165A7 (fi) 1981-01-07
PT71424A (en) 1980-07-01
NO153496B (no) 1985-12-23
FI67217C (fi) 1985-02-11
SU993817A3 (ru) 1983-01-30
NO153496C (no) 1986-05-14
IE49994B1 (en) 1986-01-22
PL125597B1 (en) 1983-05-31

Similar Documents

Publication Publication Date Title
YU42064B (en) Process for obtaining new glycevol derivatives
YU11380A (en) Process for obtaining n-benzyl-imidazole
YU171880A (en) Process for obtaining new indolizine derivatives
YU42658B (en) Process for preparing new pleuromutiline derivatives
YU42877A (en) Process for obtaining new indolizine derivatives
YU65680A (en) Process for obtaining 9-amino-alkylfluorene
YU145480A (en) Process for obtaining new hydroxyamino-eburnane derivatives
YU116380A (en) Process for obtaining thiazolylidene-oxo-propionitrile
YU43305B (en) Process for obtaining 2-amino-3-benzoyl-phenylacetamides
PT71812B (en) Process for preparing pyridazopyridazine derivatives
YU13180A (en) Process for obtaining spiro-quinolyl-hydantoin
YU108580A (en) Process for obtaining alkoxyalkylidene hydrazinopyridazine
HU178523B (en) Process for preparing new pyrazolo-quinazoline derivatives
YU236180A (en) Process for obtaining 15-sulfonamido-prostaglandin derivatives
YU188180A (en) Process for obtaining new nitroalkanol derivatives
YU100280A (en) Process for obtaining new aminoisoquinazoline derivatives
HU182184B (en) Process for preparing nitroso-carbamide derivatives
YU239680A (en) Process for obtaiing new decahydroquinolinone derivatives
YU204080A (en) Process for preparing 3-amino-2-oxozalidine derivatives
YU42127B (en) Process for obtaining new indoysine derivatives
HU178004B (en) Process for preparing new encephaline derivatives
YU297780A (en) Process for obtaining glucoso-isomerase
YU96779A (en) Process for obtaining nitrofurane derivatives
YU290679A (en) Process for obtaining furfurol-acetone derivatives
YU41658B (en) Process for obtaining guaridine derivatives