WO1999010351A1 - Derives d'acide pyridonecarboxylique et intermediaires aux fins de leur preparation - Google Patents

Derives d'acide pyridonecarboxylique et intermediaires aux fins de leur preparation Download PDF

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Publication number
WO1999010351A1
WO1999010351A1 PCT/JP1997/002918 JP9702918W WO9910351A1 WO 1999010351 A1 WO1999010351 A1 WO 1999010351A1 JP 9702918 W JP9702918 W JP 9702918W WO 9910351 A1 WO9910351 A1 WO 9910351A1
Authority
WO
WIPO (PCT)
Prior art keywords
group
compound
hydrogen atom
lower alkyl
amino
Prior art date
Application number
PCT/JP1997/002918
Other languages
English (en)
Japanese (ja)
Inventor
Nobuhiko Horiuchi
Takenori Yonezawa
Katsumi Chiba
Hiroaki Yoshida
Original Assignee
Dainippon Pharmaceutical Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dainippon Pharmaceutical Co., Ltd. filed Critical Dainippon Pharmaceutical Co., Ltd.
Priority to AU39523/97A priority Critical patent/AU3952397A/en
Priority to PCT/JP1997/002918 priority patent/WO1999010351A1/fr
Publication of WO1999010351A1 publication Critical patent/WO1999010351A1/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

L'invention a trait à des dérivés d'acide pyridonecarboxylique de la formule générale (I), à leurs sels et à leurs esters, à des médicaments les contenant ainsi qu'à des composés bicycliques amine, intermédiaires directs de ces dérivés d'acide pyridonecarboxylique. Dans la formule générale (I), R représente un cycloalkyle éventuellement halogéné ou analogue, X représente un hydrogène, un alkyle de faible poids moléculaire, un hydroxy ou un amino, Y représente un hydrogène ou un halogéno, A représente un azote ou un groupe de C-Z (où Z représente un alcoxy de faible poids moléculaire éventuellement halogéné ou analogue), R1 et R2 représentent, chacun de manière indépendante un hydrogène ou analogue, R3 représente un hydrogène ou un alkyle de faible poids moléculaire, R4, R5, R6, R7, R8 et R9 représentent, chacun de manière indépendante, un hydrogène ou un halogéno ou un alkyle de faible poids moléculaire, m vaut 0 ou 1 et n et p valent, chacun de manière indépendante 0 ou 1.
PCT/JP1997/002918 1997-08-22 1997-08-22 Derives d'acide pyridonecarboxylique et intermediaires aux fins de leur preparation WO1999010351A1 (fr)

Priority Applications (2)

Application Number Priority Date Filing Date Title
AU39523/97A AU3952397A (en) 1997-08-22 1997-08-22 Pyridonecarboxylic acid derivatives and intermediates for the preparation thereof
PCT/JP1997/002918 WO1999010351A1 (fr) 1997-08-22 1997-08-22 Derives d'acide pyridonecarboxylique et intermediaires aux fins de leur preparation

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/JP1997/002918 WO1999010351A1 (fr) 1997-08-22 1997-08-22 Derives d'acide pyridonecarboxylique et intermediaires aux fins de leur preparation

Publications (1)

Publication Number Publication Date
WO1999010351A1 true WO1999010351A1 (fr) 1999-03-04

Family

ID=14181007

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP1997/002918 WO1999010351A1 (fr) 1997-08-22 1997-08-22 Derives d'acide pyridonecarboxylique et intermediaires aux fins de leur preparation

Country Status (2)

Country Link
AU (1) AU3952397A (fr)
WO (1) WO1999010351A1 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007501819A (ja) * 2003-08-13 2007-02-01 バイエル・ヘルスケア・アクチェンゲゼルシャフト キノロン抗生物質の新規使用

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0352889A (ja) * 1989-07-19 1991-03-07 Taisho Pharmaceut Co Ltd ピロリジン化合物
WO1997031919A1 (fr) * 1996-02-27 1997-09-04 Dainippon Pharmaceutical Co., Ltd. Derives d'acide pyridonecarboxylique et leur intermediaires de synthese

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0352889A (ja) * 1989-07-19 1991-03-07 Taisho Pharmaceut Co Ltd ピロリジン化合物
WO1997031919A1 (fr) * 1996-02-27 1997-09-04 Dainippon Pharmaceutical Co., Ltd. Derives d'acide pyridonecarboxylique et leur intermediaires de synthese

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2007501819A (ja) * 2003-08-13 2007-02-01 バイエル・ヘルスケア・アクチェンゲゼルシャフト キノロン抗生物質の新規使用

Also Published As

Publication number Publication date
AU3952397A (en) 1999-03-16

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