UY36037A - Derivados de indazol y 2-metil-pirazol-piridina sustituidos como inhibidores de la tirosina quinasa (syk) del bazo y composiciones farmacéuticas que las contienen - Google Patents

Derivados de indazol y 2-metil-pirazol-piridina sustituidos como inhibidores de la tirosina quinasa (syk) del bazo y composiciones farmacéuticas que las contienen

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Publication number
UY36037A
UY36037A UY0001036037A UY36037A UY36037A UY 36037 A UY36037 A UY 36037A UY 0001036037 A UY0001036037 A UY 0001036037A UY 36037 A UY36037 A UY 36037A UY 36037 A UY36037 A UY 36037A
Authority
UY
Uruguay
Prior art keywords
typosine
bazo
pirazol
syk
indazol
Prior art date
Application number
UY0001036037A
Other languages
English (en)
Spanish (es)
Inventor
Dahmann Georg
Hoffmann Matthias
Klicic Jasna
David James Lamb
Mccarthy Clive
Napier Spencer
Parrish Karen
Scott John
Jennifer L Swantek Fitzgerald
Walker Edward
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of UY36037A publication Critical patent/UY36037A/es

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4162—1,2-Diazoles condensed with heterocyclic ring systems
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CY1121937T1 (el) 2020-10-14
HUE046061T2 (hu) 2020-02-28
US20170008896A1 (en) 2017-01-12
WO2015140054A1 (en) 2015-09-24
AU2015233654B2 (en) 2018-12-06
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CN110713489A (zh) 2020-01-21
US20160244446A1 (en) 2016-08-25
JP6535022B2 (ja) 2019-06-26
AP2016009373A0 (en) 2016-08-31
ES2738416T3 (es) 2020-01-22
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TW201623285A (zh) 2016-07-01
JP6599884B2 (ja) 2019-10-30
CN110713489B (zh) 2022-05-31
WO2015140051A1 (en) 2015-09-24
CL2016001963A1 (es) 2016-12-23
EP3119772B1 (en) 2019-05-22
MX2016011784A (es) 2016-12-02
PH12016501796A1 (en) 2016-11-21
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