UY34972A - Proceso para la preparación de inhibidores de quinasa c-FMS - Google Patents

Proceso para la preparación de inhibidores de quinasa c-FMS

Info

Publication number
UY34972A
UY34972A UY0001034972A UY34972A UY34972A UY 34972 A UY34972 A UY 34972A UY 0001034972 A UY0001034972 A UY 0001034972A UY 34972 A UY34972 A UY 34972A UY 34972 A UY34972 A UY 34972A
Authority
UY
Uruguay
Prior art keywords
kinase inhibitors
preparation
fms kinase
fms
present
Prior art date
Application number
UY0001034972A
Other languages
English (en)
Spanish (es)
Inventor
Kolodziejczyk Krzysztof
Alfred Elisabeth Stappers
Christopher A Teleha
Koen Johan Herman Weerts
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of UY34972A publication Critical patent/UY34972A/es

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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P13/08—Drugs for disorders of the urinary system of the prostate
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    • C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/30—Oxygen atoms, e.g. delta-lactones
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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
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    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/10—Compounds having one or more C—Si linkages containing nitrogen having a Si-N linkage

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UY0001034972A 2012-08-07 2013-08-07 Proceso para la preparación de inhibidores de quinasa c-FMS UY34972A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261680446P 2012-08-07 2012-08-07

Publications (1)

Publication Number Publication Date
UY34972A true UY34972A (es) 2014-02-28

Family

ID=48980367

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001034972A UY34972A (es) 2012-08-07 2013-08-07 Proceso para la preparación de inhibidores de quinasa c-FMS

Country Status (12)

Country Link
US (2) US9029352B2 (cg-RX-API-DMAC7.html)
EP (2) EP3091006B1 (cg-RX-API-DMAC7.html)
JP (1) JP6290884B2 (cg-RX-API-DMAC7.html)
CN (2) CN104520295B (cg-RX-API-DMAC7.html)
AR (2) AR092070A1 (cg-RX-API-DMAC7.html)
AU (2) AU2013299926B2 (cg-RX-API-DMAC7.html)
ES (2) ES2607807T3 (cg-RX-API-DMAC7.html)
IN (1) IN2015DN00660A (cg-RX-API-DMAC7.html)
JO (2) JOP20180012A1 (cg-RX-API-DMAC7.html)
TW (2) TWI608004B (cg-RX-API-DMAC7.html)
UY (1) UY34972A (cg-RX-API-DMAC7.html)
WO (1) WO2014025679A1 (cg-RX-API-DMAC7.html)

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WO2015125710A1 (ja) * 2014-02-18 2015-08-27 第一三共株式会社 活性化血液凝固第Ｘ因子（ＦＸａ）の阻害薬の製造方法
TW201811326A (zh) 2016-07-18 2018-04-01 比利時商健生藥品公司 ４－氰基－ｎ－（２－（４，４－二甲基環己－１－烯－１－基）－６－（２，２，６，６－四甲基四氫－２ｈ－哌喃－４－基）吡啶－３－基）－１ｈ－咪唑－２－甲醯胺之鹽形式
TWI752980B (zh) 2016-07-18 2022-01-21 比利時商健生藥品公司 4-氰基-n-(2-(4,4-二甲基環己-1-烯-1-基)-6-(2,2,6,6-四甲基四氫-2h-哌喃-4-基)吡啶-3-基)-1h-咪唑-2-甲醯胺之晶型
JP6831558B2 (ja) * 2016-08-23 2021-02-17 株式会社Ｈｂｃフナト 脳機能改善組成物
JP2020510673A (ja) * 2017-03-03 2020-04-09 ヤンセン バイオテツク，インコーポレーテツド がんの治療のための低分子ｃｓｆ−１ｒ阻害剤とｃｄ４０に特異的に結合するアゴニスト抗体とを含む併用療法
WO2020222109A1 (en) 2019-05-02 2020-11-05 Janssen Biotech, Inc. Csf-1/csf-1r gene set

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