UY32976A - Derivados de azaindol - Google Patents

Derivados de azaindol

Info

Publication number
UY32976A
UY32976A UY0001032976A UY32976A UY32976A UY 32976 A UY32976 A UY 32976A UY 0001032976 A UY0001032976 A UY 0001032976A UY 32976 A UY32976 A UY 32976A UY 32976 A UY32976 A UY 32976A
Authority
UY
Uruguay
Prior art keywords
compounds
azaindol
derivatives
copd
asthma
Prior art date
Application number
UY0001032976A
Other languages
English (en)
Inventor
David Michael Evans
Christine Elizabeth Allan
Original Assignee
Vantia Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vantia Ltd filed Critical Vantia Ltd
Publication of UY32976A publication Critical patent/UY32976A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pulmonology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La presente invención proporciona compuestos de fórmula (I), composiciones que comprenden dichos compuestos; el uso de dichos compuestos en terapia (tal como asma o EPOC); y métodos para tratar pacientes con tales compuestos; en donde R1 a R20 y A1 son tal como se definen en la presente.
UY0001032976A 2009-10-28 2010-10-27 Derivados de azaindol UY32976A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25561009P 2009-10-28 2009-10-28
GBGB0918924.2A GB0918924D0 (en) 2009-10-28 2009-10-28 Azaindole derivatives

Publications (1)

Publication Number Publication Date
UY32976A true UY32976A (es) 2011-05-31

Family

ID=41434816

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032976A UY32976A (es) 2009-10-28 2010-10-27 Derivados de azaindol

Country Status (5)

Country Link
AR (1) AR078818A1 (es)
GB (1) GB0918924D0 (es)
TW (1) TW201120038A (es)
UY (1) UY32976A (es)
WO (1) WO2011051672A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9290485B2 (en) 2010-08-04 2016-03-22 Novartis Ag N-((6-amino-pyridin-3-yl)methyl)-heteroaryl-carboxamides
CN114269431A (zh) * 2019-08-21 2022-04-01 卡尔维斯塔制药有限公司 酶抑制剂

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Also Published As

Publication number Publication date
WO2011051672A1 (en) 2011-05-05
AR078818A1 (es) 2011-12-07
TW201120038A (en) 2011-06-16
GB0918924D0 (en) 2009-12-16

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Effective date: 20121113