UA85087C2 - Monocyclic heterocycles as kinase inhibitors - Google Patents
Monocyclic heterocycles as kinase inhibitorsInfo
- Publication number
- UA85087C2 UA85087C2 UAA200612282A UAA200612282A UA85087C2 UA 85087 C2 UA85087 C2 UA 85087C2 UA A200612282 A UAA200612282 A UA A200612282A UA A200612282 A UAA200612282 A UA A200612282A UA 85087 C2 UA85087 C2 UA 85087C2
- Authority
- UA
- Ukraine
- Prior art keywords
- kinase inhibitors
- monocyclic heterocycles
- heterocycles
- monocyclic
- cancer
- Prior art date
Links
Abstract
Даний винахід спрямований на сполуки, які мають формулу [І + II], та способи їх застосування для лікування раку..
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US56484204P | 2004-04-23 | 2004-04-23 |
Publications (1)
Publication Number | Publication Date |
---|---|
UA85087C2 true UA85087C2 (en) | 2008-12-25 |
Family
ID=39095986
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UAA200612282A UA85087C2 (en) | 2004-04-23 | 2005-04-22 | Monocyclic heterocycles as kinase inhibitors |
Country Status (4)
Country | Link |
---|---|
CN (1) | CN101128199B (uk) |
ES (1) | ES2359836T3 (uk) |
UA (1) | UA85087C2 (uk) |
ZA (1) | ZA200608775B (uk) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EA201170627A1 (ru) * | 2008-10-29 | 2011-10-31 | ДЕСИФЕРА ФАРМАСЬЮТИКАЛЗ, ЭлЭлСи | Циклопропанамиды и аналоги, проявляющие противораковые и антипролиферативные активности |
AR076332A1 (es) * | 2009-04-21 | 2011-06-01 | Boehringer Ingelheim Int | Derivados heterociclicos de 5-alquinil-piridinas, composiciones farmaceuticas que los comprenden y uso de los mismos para el tratamiento y/o prevencion del cancer, procesos inflamatorios, autoinmunes, y/o infecciones. |
CN102285914B (zh) * | 2010-06-18 | 2013-12-25 | 上海药明康德新药开发有限公司 | 2-(1-甲基-6-羰基-1,6-二氢-吡啶)-乙酸的合成方法 |
CN102816175B (zh) * | 2011-06-09 | 2015-12-16 | 上海汇伦生命科技有限公司 | 一种杂环并吡啶酮类化合物,其中间体、制备方法和用途 |
TWI570116B (zh) * | 2012-08-03 | 2017-02-11 | 習寧 | 取代的吡唑酮化合物及其使用方法 |
CN102875455A (zh) * | 2012-10-23 | 2013-01-16 | 西华大学 | 一种3,6-二氯-2-氨基吡啶的合成工艺 |
WO2014209841A2 (en) * | 2013-06-25 | 2014-12-31 | F. Hoffmann-La Roche Ag | Compounds for treating spinal muscular atrophy |
WO2019080723A1 (zh) * | 2017-10-26 | 2019-05-02 | 北京越之康泰生物医药科技有限公司 | 多取代吡啶酮类衍生物、其制备方法及其医药用途 |
KR20210066820A (ko) * | 2018-08-27 | 2021-06-07 | 베이징 위에즈캉타이 바이오메디슨스 컴퍼니, 리미티드 | 다중-치환된 피리돈 유도체 및 이의 의학적 용도 |
CN113999205B (zh) * | 2021-12-13 | 2023-09-15 | 辽宁大学 | 含三氮唑酮酰胺和咪唑酰胺结构的吡啶类化合物及其应用 |
CN117486860A (zh) * | 2022-07-25 | 2024-02-02 | 上海博悦生物科技有限公司 | Axl&c-Met双重抑制剂、制备方法以及用途 |
CN116870968B (zh) * | 2023-09-08 | 2023-11-10 | 烟台大学 | 铱配合物功能化纳米石墨烯催化剂、其制备方法与应用 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ATE443047T1 (de) * | 2001-06-22 | 2009-10-15 | Kirin Pharma Kk | Chinolinderivat und chinazolinderivat, die die selbstphosphorylierung des hepatocytus- proliferator-rezeptors hemmen, und diese enthaltende medizinische zusammensetzung |
WO2005005389A2 (en) * | 2003-07-07 | 2005-01-20 | Merck Patent Gmbh | Malonamide derivatives |
-
2005
- 2005-04-22 ES ES05779444T patent/ES2359836T3/es active Active
- 2005-04-22 UA UAA200612282A patent/UA85087C2/ru unknown
- 2005-04-22 CN CN200580020112.2A patent/CN101128199B/zh active Active
-
2006
- 2006-10-20 ZA ZA200608775A patent/ZA200608775B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
CN101128199B (zh) | 2013-07-24 |
ZA200608775B (en) | 2008-06-25 |
CN101128199A (zh) | 2008-02-20 |
ES2359836T3 (es) | 2011-05-27 |
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