UA85087C2 - Monocyclic heterocycles as kinase inhibitors - Google Patents

Monocyclic heterocycles as kinase inhibitors

Info

Publication number
UA85087C2
UA85087C2 UAA200612282A UAA200612282A UA85087C2 UA 85087 C2 UA85087 C2 UA 85087C2 UA A200612282 A UAA200612282 A UA A200612282A UA A200612282 A UAA200612282 A UA A200612282A UA 85087 C2 UA85087 C2 UA 85087C2
Authority
UA
Ukraine
Prior art keywords
kinase inhibitors
monocyclic heterocycles
heterocycles
monocyclic
cancer
Prior art date
Application number
UAA200612282A
Other languages
English (en)
Russian (ru)
Inventor
Роберт М. Борзиллери
Линдон А.М. Корнелиус
Роберт Дж. ШМИДТ
Гретхен М. Шредер
Кьянг С. Ким
Original Assignee
Бристол-Майэрс Сквибб Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Бристол-Майэрс Сквибб Компани filed Critical Бристол-Майэрс Сквибб Компани
Publication of UA85087C2 publication Critical patent/UA85087C2/ru

Links

Abstract

Даний винахід спрямований на сполуки, які мають формулу [І + II], та способи їх застосування для лікування раку..
UAA200612282A 2004-04-23 2005-04-22 Monocyclic heterocycles as kinase inhibitors UA85087C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US56484204P 2004-04-23 2004-04-23

Publications (1)

Publication Number Publication Date
UA85087C2 true UA85087C2 (en) 2008-12-25

Family

ID=39095986

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200612282A UA85087C2 (en) 2004-04-23 2005-04-22 Monocyclic heterocycles as kinase inhibitors

Country Status (4)

Country Link
CN (1) CN101128199B (uk)
ES (1) ES2359836T3 (uk)
UA (1) UA85087C2 (uk)
ZA (1) ZA200608775B (uk)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA201170627A1 (ru) * 2008-10-29 2011-10-31 ДЕСИФЕРА ФАРМАСЬЮТИКАЛЗ, ЭлЭлСи Циклопропанамиды и аналоги, проявляющие противораковые и антипролиферативные активности
AR076332A1 (es) * 2009-04-21 2011-06-01 Boehringer Ingelheim Int Derivados heterociclicos de 5-alquinil-piridinas, composiciones farmaceuticas que los comprenden y uso de los mismos para el tratamiento y/o prevencion del cancer, procesos inflamatorios, autoinmunes, y/o infecciones.
CN102285914B (zh) * 2010-06-18 2013-12-25 上海药明康德新药开发有限公司 2-(1-甲基-6-羰基-1,6-二氢-吡啶)-乙酸的合成方法
CN102816175B (zh) * 2011-06-09 2015-12-16 上海汇伦生命科技有限公司 一种杂环并吡啶酮类化合物,其中间体、制备方法和用途
TWI570116B (zh) * 2012-08-03 2017-02-11 習寧 取代的吡唑酮化合物及其使用方法
CN102875455A (zh) * 2012-10-23 2013-01-16 西华大学 一种3,6-二氯-2-氨基吡啶的合成工艺
WO2014209841A2 (en) * 2013-06-25 2014-12-31 F. Hoffmann-La Roche Ag Compounds for treating spinal muscular atrophy
WO2019080723A1 (zh) * 2017-10-26 2019-05-02 北京越之康泰生物医药科技有限公司 多取代吡啶酮类衍生物、其制备方法及其医药用途
KR20210066820A (ko) * 2018-08-27 2021-06-07 베이징 위에즈캉타이 바이오메디슨스 컴퍼니, 리미티드 다중-치환된 피리돈 유도체 및 이의 의학적 용도
CN113999205B (zh) * 2021-12-13 2023-09-15 辽宁大学 含三氮唑酮酰胺和咪唑酰胺结构的吡啶类化合物及其应用
CN117486860A (zh) * 2022-07-25 2024-02-02 上海博悦生物科技有限公司 Axl&c-Met双重抑制剂、制备方法以及用途
CN116870968B (zh) * 2023-09-08 2023-11-10 烟台大学 铱配合物功能化纳米石墨烯催化剂、其制备方法与应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE443047T1 (de) * 2001-06-22 2009-10-15 Kirin Pharma Kk Chinolinderivat und chinazolinderivat, die die selbstphosphorylierung des hepatocytus- proliferator-rezeptors hemmen, und diese enthaltende medizinische zusammensetzung
WO2005005389A2 (en) * 2003-07-07 2005-01-20 Merck Patent Gmbh Malonamide derivatives

Also Published As

Publication number Publication date
CN101128199B (zh) 2013-07-24
ZA200608775B (en) 2008-06-25
CN101128199A (zh) 2008-02-20
ES2359836T3 (es) 2011-05-27

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