ZA200608775B - Monocyclic heterocycles as kinase inhibitors - Google Patents

Monocyclic heterocycles as kinase inhibitors

Info

Publication number
ZA200608775B
ZA200608775B ZA200608775A ZA200608775A ZA200608775B ZA 200608775 B ZA200608775 B ZA 200608775B ZA 200608775 A ZA200608775 A ZA 200608775A ZA 200608775 A ZA200608775 A ZA 200608775A ZA 200608775 B ZA200608775 B ZA 200608775B
Authority
ZA
South Africa
Prior art keywords
kinase inhibitors
monocyclic heterocycles
heterocycles
monocyclic
kinase
Prior art date
Application number
ZA200608775A
Other languages
English (en)
Inventor
Robert M Borzilleri
Robert J Schmidt
Kyoung S Kim
Lyndon A M Cornelius
Gretchen M Schroeder
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of ZA200608775B publication Critical patent/ZA200608775B/xx

Links

ZA200608775A 2004-04-23 2006-10-20 Monocyclic heterocycles as kinase inhibitors ZA200608775B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US56484204P 2004-04-23 2004-04-23

Publications (1)

Publication Number Publication Date
ZA200608775B true ZA200608775B (en) 2008-06-25

Family

ID=39095986

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200608775A ZA200608775B (en) 2004-04-23 2006-10-20 Monocyclic heterocycles as kinase inhibitors

Country Status (4)

Country Link
CN (1) CN101128199B (xx)
ES (1) ES2359836T3 (xx)
UA (1) UA85087C2 (xx)
ZA (1) ZA200608775B (xx)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI0920765A2 (pt) * 2008-10-29 2015-08-18 Deciphera Pharmaceuticals Llc Amidas de cilopropano e análogos que exibem atividades anticâncer e antiproliferativas
AR076332A1 (es) * 2009-04-21 2011-06-01 Boehringer Ingelheim Int Derivados heterociclicos de 5-alquinil-piridinas, composiciones farmaceuticas que los comprenden y uso de los mismos para el tratamiento y/o prevencion del cancer, procesos inflamatorios, autoinmunes, y/o infecciones.
CN102285914B (zh) * 2010-06-18 2013-12-25 上海药明康德新药开发有限公司 2-(1-甲基-6-羰基-1,6-二氢-吡啶)-乙酸的合成方法
CN102816175B (zh) * 2011-06-09 2015-12-16 上海汇伦生命科技有限公司 一种杂环并吡啶酮类化合物,其中间体、制备方法和用途
TWI565702B (zh) * 2012-08-03 2017-01-11 習寧 取代的吡唑酮化合物及其使用方法
CN102875455A (zh) * 2012-10-23 2013-01-16 西华大学 一种3,6-二氯-2-氨基吡啶的合成工艺
KR102314290B1 (ko) * 2013-06-25 2021-10-21 에프. 호프만-라 로슈 아게 척수성 근위축증을 치료하기 위한 화합물
WO2019080723A1 (zh) * 2017-10-26 2019-05-02 北京越之康泰生物医药科技有限公司 多取代吡啶酮类衍生物、其制备方法及其医药用途
EP3845527A4 (en) * 2018-08-27 2022-06-08 Beijing Yuezhikangtai Biomedicines Co., Ltd. MULTISUBSTITUTED PYRIDONE DERIVATIVES AND THEIR MEDICAL USE
CN113999205B (zh) * 2021-12-13 2023-09-15 辽宁大学 含三氮唑酮酰胺和咪唑酰胺结构的吡啶类化合物及其应用
CN117486860A (zh) * 2022-07-25 2024-02-02 上海博悦生物科技有限公司 Axl&c-Met双重抑制剂、制备方法以及用途
CN116870968B (zh) * 2023-09-08 2023-11-10 烟台大学 铱配合物功能化纳米石墨烯催化剂、其制备方法与应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003000660A1 (en) * 2001-06-22 2003-01-03 Kirin Beer Kabushiki Kaisha Quinoline derivative and quinazoline derivative inhibiting self-phosphorylation of hepatocytus proliferator receptor, and medicinal composition containing the same
AU2004255566B2 (en) * 2003-07-07 2010-07-08 Merk Patent Gmbh Malonamide derivatives

Also Published As

Publication number Publication date
CN101128199A (zh) 2008-02-20
UA85087C2 (xx) 2008-12-25
CN101128199B (zh) 2013-07-24
ES2359836T3 (es) 2011-05-27

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