UA82782C2 - Антимикобактериальной фармакологическая композиция и способ ее получения - Google Patents
Антимикобактериальной фармакологическая композиция и способ ее получения Download PDFInfo
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- UA82782C2 UA82782C2 UAA200612258A UAA200612258A UA82782C2 UA 82782 C2 UA82782 C2 UA 82782C2 UA A200612258 A UAA200612258 A UA A200612258A UA A200612258 A UAA200612258 A UA A200612258A UA 82782 C2 UA82782 C2 UA 82782C2
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Landscapes
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Abstract
Изобретение относится к фармацевтике, в частности к антимикобактериальной комбинации для лечения туберкулёза. Используемыми соединениями являются N-(3-[[4-(3-трифторметилфенил)пиперазинил]метил]-2-метил-5-фенил-пирролил)-4-пиридилкарбоксамид формули (І) или его фармацевтически приемлемая нетоксическая сольи один или несколько антитуберкулёзных лекарственных средств первого ряда. Изобретение также относится к способу получения этой комбинации.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US10/844,992 US7491721B2 (en) | 2004-05-12 | 2004-05-12 | Antimycobacterial pharmaceutical composition |
PCT/IN2004/000266 WO2005107809A2 (en) | 2004-05-12 | 2004-08-27 | Antimycobacterial pharmaceutical composition comprising an antitubercular drug |
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UA82782C2 true UA82782C2 (ru) | 2008-05-12 |
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UAA200612258A UA82782C2 (ru) | 2004-05-12 | 2004-08-27 | Антимикобактериальной фармакологическая композиция и способ ее получения |
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US20090118509A1 (en) * | 2005-04-11 | 2009-05-07 | Lupin Limited | Preparation of [2-methyl-5-phenyl-3-(piperazin-1-ylmethyl)] pyrrole derivatives |
JP5339840B2 (ja) * | 2008-10-02 | 2013-11-13 | 公益財団法人微生物化学研究会 | 抗xdr−tb薬、抗mdr−tb薬、及び併用抗結核薬 |
US9198913B2 (en) * | 2009-07-31 | 2015-12-01 | Global Alliance For Tb Drug Development | Nitroimidazooxazines and their uses in anti-tubercular therapy |
JP2013504591A (ja) * | 2009-09-11 | 2013-02-07 | バーテックス ファーマシューティカルズ インコーポレイテッド | N−ベンジル−3−(4−クロロフェニル)−2−[メチル−[2−オキソ−2−(3,4,5−トリメトキシフェニル)アセチル]アミノ]−n−[3−(4−ピリジル)−1−[2−(4−ピリジル)エチル]プロピル]プロパンアミドの組成物およびその使用 |
HUP1000033A2 (en) * | 2010-01-21 | 2011-07-28 | Uratim Kft | Piperazine derivatives useful against mycobacteriums |
KR102462751B1 (ko) * | 2021-10-20 | 2022-11-03 | 순천향대학교 산학협력단 | 신규한 페디오코커스 균주 및 이를 포함하는 결핵 예방, 치료, 또는 개선용 조성물 |
US11977085B1 (en) | 2023-09-05 | 2024-05-07 | Elan Ehrlich | Date rape drug detection device and method of using same |
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US5227383A (en) * | 1991-06-14 | 1993-07-13 | The University Of Mississippi | Compounds and compositions useful as antifungal and antimycobacterial agents |
JP2006503837A (ja) * | 2002-09-20 | 2006-02-02 | ルピン・リミテッド | 新規の抗マイコバクテリア化合物 |
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