UA72890C2 - A crystalline form of osanetant (variants), a method for the preparation thereof (variants) and a pharmaceutical composition - Google Patents
A crystalline form of osanetant (variants), a method for the preparation thereof (variants) and a pharmaceutical compositionInfo
- Publication number
- UA72890C2 UA72890C2 UA2001010591A UA2001010591A UA72890C2 UA 72890 C2 UA72890 C2 UA 72890C2 UA 2001010591 A UA2001010591 A UA 2001010591A UA 2001010591 A UA2001010591 A UA 2001010591A UA 72890 C2 UA72890 C2 UA 72890C2
- Authority
- UA
- Ukraine
- Prior art keywords
- variants
- osanetant
- preparation
- pharmaceutical composition
- crystalline form
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9810107A FR2782082B3 (fr) | 1998-08-05 | 1998-08-05 | Formes cristallines de (r)-(+)-n-[[3-[1-benzoyl-3-(3,4- dichlorophenyl)piperidin-3-yl]prop-1-yl]-4-phenylpiperidin-4 -yl]-n-methylacetamide (osanetant) et procede pour la preparation dudit compose |
| PCT/FR1999/001914 WO2000007987A1 (fr) | 1998-08-05 | 1999-08-03 | Formes cristallines du osanetant |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA72890C2 true UA72890C2 (en) | 2005-05-16 |
Family
ID=9529458
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UA2001010591A UA72890C2 (en) | 1998-08-05 | 1999-08-03 | A crystalline form of osanetant (variants), a method for the preparation thereof (variants) and a pharmaceutical composition |
Country Status (32)
| Country | Link |
|---|---|
| US (1) | US7041679B2 (de) |
| EP (1) | EP1102747B1 (de) |
| JP (1) | JP3807938B2 (de) |
| KR (1) | KR100571944B1 (de) |
| CN (1) | CN1114592C (de) |
| AR (1) | AR019953A1 (de) |
| AT (1) | ATE243197T1 (de) |
| AU (1) | AU748177B2 (de) |
| BR (1) | BR9913357A (de) |
| CA (1) | CA2339007A1 (de) |
| CO (1) | CO5070576A1 (de) |
| DE (1) | DE69908951T2 (de) |
| DK (1) | DK1102747T3 (de) |
| DZ (1) | DZ3074A1 (de) |
| EA (1) | EA003205B1 (de) |
| EE (1) | EE04274B1 (de) |
| ES (1) | ES2200535T3 (de) |
| FR (1) | FR2782082B3 (de) |
| HK (1) | HK1035535A1 (de) |
| HU (1) | HUP0103134A3 (de) |
| IS (1) | IS5821A (de) |
| MY (1) | MY121447A (de) |
| NO (1) | NO320645B1 (de) |
| NZ (1) | NZ509561A (de) |
| PL (1) | PL345999A1 (de) |
| PT (1) | PT1102747E (de) |
| SK (1) | SK1742001A3 (de) |
| TR (1) | TR200100261T2 (de) |
| TW (1) | TW527354B (de) |
| UA (1) | UA72890C2 (de) |
| WO (1) | WO2000007987A1 (de) |
| YU (1) | YU8601A (de) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0100902D0 (sv) * | 2001-03-15 | 2001-03-15 | Astrazeneca Ab | Compounds |
| SE0202539D0 (sv) | 2002-08-27 | 2002-08-27 | Astrazeneca Ab | Compounds |
| SE0401762D0 (sv) * | 2004-07-05 | 2004-07-05 | Astrazeneca Ab | Novel compounds |
| US7648992B2 (en) * | 2004-07-05 | 2010-01-19 | Astrazeneca Ab | Hydantoin derivatives for the treatment of obstructive airway diseases |
| SE0403086D0 (sv) * | 2004-12-17 | 2004-12-17 | Astrazeneca Ab | Compounds |
| SE0403085D0 (sv) * | 2004-12-17 | 2004-12-17 | Astrazeneca Ab | Novel componds |
| TW200800954A (en) * | 2006-03-16 | 2008-01-01 | Astrazeneca Ab | Novel crystal modifications |
| TW200831488A (en) * | 2006-11-29 | 2008-08-01 | Astrazeneca Ab | Novel compounds |
| WO2023278843A2 (en) * | 2021-07-02 | 2023-01-05 | Acer Therapeutics, Inc. | Solid forms of osanetant |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2719311B1 (fr) | 1994-03-18 | 1998-06-26 | Sanofi Sa | Composés antagonistes sélectifs du récepteur NK3 humain et leur utilisation comme médicaments et outils de diagnostic. |
| JPH1053576A (ja) * | 1996-06-07 | 1998-02-24 | Eisai Co Ltd | 塩酸ドネペジルの多形結晶およびその製造法 |
| WO1998005640A2 (en) * | 1996-08-05 | 1998-02-12 | Smithkline Beecham S.P.A. | Process for the preparation of 3,3-disubstituted piperidines |
| US6040316A (en) * | 1996-09-16 | 2000-03-21 | Warner-Lambert Company | 3-alkyl-3-phenyl-piperidines |
| FR2757543B1 (fr) * | 1996-12-23 | 1999-04-02 | Sanofi Sa | Procede pour la cristallisation d'un derive de tetrahydropyridine et formes cristallines ainsi obtenues |
-
1998
- 1998-08-05 FR FR9810107A patent/FR2782082B3/fr not_active Expired - Lifetime
-
1999
- 1999-07-25 DZ DZ990156A patent/DZ3074A1/xx active
- 1999-07-28 AR ARP990103741A patent/AR019953A1/es unknown
- 1999-08-03 DK DK99936672T patent/DK1102747T3/da active
- 1999-08-03 TR TR2001/00261T patent/TR200100261T2/xx unknown
- 1999-08-03 CA CA002339007A patent/CA2339007A1/en not_active Abandoned
- 1999-08-03 PL PL99345999A patent/PL345999A1/xx not_active Application Discontinuation
- 1999-08-03 PT PT99936672T patent/PT1102747E/pt unknown
- 1999-08-03 MY MYPI99003297A patent/MY121447A/en unknown
- 1999-08-03 ES ES99936672T patent/ES2200535T3/es not_active Expired - Lifetime
- 1999-08-03 KR KR1020017001460A patent/KR100571944B1/ko not_active IP Right Cessation
- 1999-08-03 EE EEP200100070A patent/EE04274B1/xx not_active IP Right Cessation
- 1999-08-03 CN CN99810182A patent/CN1114592C/zh not_active Expired - Fee Related
- 1999-08-03 EP EP99936672A patent/EP1102747B1/de not_active Expired - Lifetime
- 1999-08-03 UA UA2001010591A patent/UA72890C2/xx unknown
- 1999-08-03 NZ NZ509561A patent/NZ509561A/xx unknown
- 1999-08-03 EA EA200100096A patent/EA003205B1/ru not_active IP Right Cessation
- 1999-08-03 AU AU51685/99A patent/AU748177B2/en not_active Ceased
- 1999-08-03 DE DE69908951T patent/DE69908951T2/de not_active Expired - Fee Related
- 1999-08-03 HU HU0103134A patent/HUP0103134A3/hu unknown
- 1999-08-03 AT AT99936672T patent/ATE243197T1/de not_active IP Right Cessation
- 1999-08-03 WO PCT/FR1999/001914 patent/WO2000007987A1/fr not_active Application Discontinuation
- 1999-08-03 SK SK174-2001A patent/SK1742001A3/sk unknown
- 1999-08-03 BR BR9913357-1A patent/BR9913357A/pt not_active IP Right Cessation
- 1999-08-03 YU YU8601A patent/YU8601A/sh unknown
- 1999-08-03 JP JP2000563621A patent/JP3807938B2/ja not_active Expired - Fee Related
- 1999-08-04 CO CO99049286A patent/CO5070576A1/es unknown
- 1999-08-04 TW TW088113235A patent/TW527354B/zh not_active IP Right Cessation
-
2001
- 2001-01-23 IS IS5821A patent/IS5821A/is unknown
- 2001-02-01 NO NO20010553A patent/NO320645B1/no unknown
- 2001-09-04 HK HK01106232A patent/HK1035535A1/xx not_active IP Right Cessation
-
2003
- 2003-08-28 US US10/651,313 patent/US7041679B2/en not_active Expired - Fee Related
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