UA128161C2 - ПОХІДНІ БЕНЗІМІДАЗОЛУ ЯК МОДУЛЯТОРИ РЕТИНОЇД-СПОРІДНЕНОГО ОРФАННОГО РЕЦЕПТОРА ГАММА (ROR<font face="Symbol">g</font>) ТА ЇХ ФАРМАЦЕВТИЧНЕ ЗАСТОСУВАННЯ - Google Patents

ПОХІДНІ БЕНЗІМІДАЗОЛУ ЯК МОДУЛЯТОРИ РЕТИНОЇД-СПОРІДНЕНОГО ОРФАННОГО РЕЦЕПТОРА ГАММА (ROR<font face="Symbol">g</font>) ТА ЇХ ФАРМАЦЕВТИЧНЕ ЗАСТОСУВАННЯ Download PDF

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UA128161C2
UA128161C2 UAA202007544A UAA202007544A UA128161C2 UA 128161 C2 UA128161 C2 UA 128161C2 UA A202007544 A UAA202007544 A UA A202007544A UA A202007544 A UAA202007544 A UA A202007544A UA 128161 C2 UA128161 C2 UA 128161C2
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Ukraine
Prior art keywords
alkyl
cycloalkyl
group
heterocyclyl
heteroaryl
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UAA202007544A
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English (en)
Ukrainian (uk)
Inventor
Іньфа Янь
Иньфа ЯНЬ
Міньшен Жанг
Миньшен Жанг
Донг Ліу
Донг Лиу
Феньци Жанг
Сусин Ліу
Сусин Лу
Румін Жанг
Румин Жанг
Фенг ХЕ
Вейкан Тао
Original Assignee
Джянгсу Хенгруй Медісін Ко., Лтд.
Джянгсу Хенгруй Медисин Ко., Лтд.
Шанхай Хенгруй Фармасьютікал Ко., Лтд.
Шанхай Хенгруй Фармасьютикал Ко., Лтд.
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Publication of UA128161C2 publication Critical patent/UA128161C2/uk

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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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UAA202007544A 2018-05-03 2019-05-03 ПОХІДНІ БЕНЗІМІДАЗОЛУ ЯК МОДУЛЯТОРИ РЕТИНОЇД-СПОРІДНЕНОГО ОРФАННОГО РЕЦЕПТОРА ГАММА (ROR<font face="Symbol">g</font>) ТА ЇХ ФАРМАЦЕВТИЧНЕ ЗАСТОСУВАННЯ UA128161C2 (uk)

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US201862666312P 2018-05-03 2018-05-03
PCT/US2019/030526 WO2019213470A1 (en) 2018-05-03 2019-05-03 Benzimidazole derivatives as modulators of retinoid-related orphan receptor gamma (rorϒ) and pharmaceutical uses thereof

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UA128161C2 true UA128161C2 (uk) 2024-04-24

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