UA121473C2 - Поліморфна форма [5-фтор-3-({2-[(4-фторбензол)сульфоніл]піридин-3-іл}метил)-2-метиліндол-1-іл]-оцтової кислоти - Google Patents
Поліморфна форма [5-фтор-3-({2-[(4-фторбензол)сульфоніл]піридин-3-іл}метил)-2-метиліндол-1-іл]-оцтової кислоти Download PDFInfo
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- UA121473C2 UA121473C2 UAA201611544A UAA201611544A UA121473C2 UA 121473 C2 UA121473 C2 UA 121473C2 UA A201611544 A UAA201611544 A UA A201611544A UA A201611544 A UAA201611544 A UA A201611544A UA 121473 C2 UA121473 C2 UA 121473C2
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- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
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- Ophthalmology & Optometry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| GBGB1407807.5A GB201407807D0 (en) | 2014-05-02 | 2014-05-02 | Polymorphic form |
| PCT/GB2015/051289 WO2015166274A1 (en) | 2014-05-02 | 2015-05-01 | Polymorphic form of [5-fluoro-3-({2-[(4-fluorobenzene) sulfonyl]pyridin-3-yl}methyl)-2-methylindol-1-yl]-acetic acid |
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| UA121473C2 true UA121473C2 (uk) | 2020-06-10 |
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| EP3555061B1 (en) | 2016-12-13 | 2023-06-07 | Watson Laboratories Inc. | Solid state forms of apalutamide |
| CN108658858B (zh) * | 2017-06-27 | 2022-02-25 | 上海中西三维药业有限公司 | 一种羟氯喹的制备和精制方法及其硫酸盐的制备方法 |
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| BE790679A (fr) | 1971-11-03 | 1973-04-27 | Ici Ltd | Derives de l'indole |
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| DE3514696A1 (de) | 1985-04-24 | 1986-11-06 | Bayer Ag, 5090 Leverkusen | N-indolylethyl-sulfonsaeureamide, verfahren zu ihrer herstellung und ihre verwendung |
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| SE0201635D0 (sv) | 2002-05-30 | 2002-05-30 | Astrazeneca Ab | Novel compounds |
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| GB0324763D0 (en) | 2003-10-23 | 2003-11-26 | Oxagen Ltd | Use of compounds in therapy |
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| GB2422831A (en) | 2005-02-04 | 2006-08-09 | Oxagen Ltd | Pyrrolopyridines and their use in the treatment of diseases mediated by PGD2 at the CRTH2 receptor |
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| GB0614066D0 (en) | 2006-07-14 | 2006-08-23 | Glaxo Group Ltd | Compounds |
| GB0614068D0 (en) | 2006-07-14 | 2006-08-23 | Glaxo Group Ltd | Compounds |
| EP2492268A1 (en) | 2006-07-22 | 2012-08-29 | Oxagen Limited | Compounds having CRTH2 antagonist activity |
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| GB201103837D0 (en) | 2011-03-07 | 2011-04-20 | Oxagen Ltd | Amorphous (5-Fluoro-2-Methyl-3-Quinolin-2-Ylmethyl-Indol-1-Yl)-acetic acid |
| GB201121557D0 (en) * | 2011-12-15 | 2012-01-25 | Oxagen Ltd | Process |
| MX2014007239A (es) | 2011-12-16 | 2014-08-08 | Atopix Therapeutics Ltd | Combinacion de un antagonista crth2 y un inhibidor de bomba de proton para el tratamiento de esofagitis eosinofilica. |
| GB201322273D0 (en) | 2013-12-17 | 2014-01-29 | Atopix Therapeutics Ltd | Process |
| GB201407813D0 (en) | 2014-05-02 | 2014-06-18 | Atopix Therapeutics Ltd | Polymorphic form |
| GB201407820D0 (en) * | 2014-05-02 | 2014-06-18 | Atopix Therapeutics Ltd | Polymorphic form |
-
2014
- 2014-05-02 GB GBGB1407807.5A patent/GB201407807D0/en not_active Ceased
-
2015
- 2015-05-01 US US15/308,288 patent/US10011584B2/en active Active
- 2015-05-01 EP EP15721029.5A patent/EP3137452B1/en active Active
- 2015-05-01 WO PCT/GB2015/051289 patent/WO2015166274A1/en not_active Ceased
- 2015-05-01 JP JP2016565467A patent/JP2017514842A/ja active Pending
- 2015-05-01 RU RU2016141463A patent/RU2751319C2/ru active
- 2015-05-01 UA UAA201611544A patent/UA121473C2/uk unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US10011584B2 (en) | 2018-07-03 |
| RU2751319C2 (ru) | 2021-07-13 |
| WO2015166274A1 (en) | 2015-11-05 |
| GB201407807D0 (en) | 2014-06-18 |
| JP2017514842A (ja) | 2017-06-08 |
| EP3137452A1 (en) | 2017-03-08 |
| EP3137452B1 (en) | 2019-12-25 |
| US20170057944A1 (en) | 2017-03-02 |
| RU2016141463A (ru) | 2018-06-05 |
| RU2016141463A3 (cg-RX-API-DMAC7.html) | 2018-11-06 |
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