TWI842681B - 用於醫學治療的索馬谷如肽 - Google Patents

用於醫學治療的索馬谷如肽 Download PDF

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Publication number
TWI842681B
TWI842681B TW107136028A TW107136028A TWI842681B TW I842681 B TWI842681 B TW I842681B TW 107136028 A TW107136028 A TW 107136028A TW 107136028 A TW107136028 A TW 107136028A TW I842681 B TWI842681 B TW I842681B
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TW
Taiwan
Prior art keywords
peptide
somagro
somaglutinol
composition
weight
Prior art date
Application number
TW107136028A
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English (en)
Chinese (zh)
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TW201914611A (zh
Inventor
瑪麗亞 凱比史契
湯瑪士 漢聲
Original Assignee
丹麥商諾佛 儂迪克股份有限公司
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=60083831&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TWI842681(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 丹麥商諾佛 儂迪克股份有限公司 filed Critical 丹麥商諾佛 儂迪克股份有限公司
Publication of TW201914611A publication Critical patent/TW201914611A/zh
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/26Glucagons
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Obesity (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Endocrinology (AREA)
  • Zoology (AREA)
  • Diabetes (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Hematology (AREA)
  • Dispersion Chemistry (AREA)
  • Dermatology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
TW107136028A 2017-10-12 2018-10-12 用於醫學治療的索馬谷如肽 TWI842681B (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP17196254.1 2017-10-12
EP17196254 2017-10-12

Publications (2)

Publication Number Publication Date
TW201914611A TW201914611A (zh) 2019-04-16
TWI842681B true TWI842681B (zh) 2024-05-21

Family

ID=60083831

Family Applications (1)

Application Number Title Priority Date Filing Date
TW107136028A TWI842681B (zh) 2017-10-12 2018-10-12 用於醫學治療的索馬谷如肽

Country Status (18)

Country Link
US (4) US12029779B2 (OSRAM)
EP (1) EP3694538A1 (OSRAM)
JP (2) JP7148605B2 (OSRAM)
KR (1) KR20200069316A (OSRAM)
CN (4) CN119838000A (OSRAM)
AU (2) AU2018348929B2 (OSRAM)
BR (1) BR112020006246A2 (OSRAM)
CA (1) CA3078652A1 (OSRAM)
CL (1) CL2020000812A1 (OSRAM)
IL (3) IL322968A (OSRAM)
MA (1) MA50358A (OSRAM)
MX (3) MX2020003049A (OSRAM)
MY (1) MY204827A (OSRAM)
PH (1) PH12020550185A1 (OSRAM)
SG (1) SG11202002841PA (OSRAM)
TW (1) TWI842681B (OSRAM)
WO (1) WO2019072941A1 (OSRAM)
ZA (3) ZA202503387B (OSRAM)

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Publication number Priority date Publication date Assignee Title
MA50358A (fr) * 2017-10-12 2020-08-19 Novo Nordisk As Sémaglutide en thérapie médicale
AU2021208601B2 (en) * 2020-02-18 2025-06-05 Novo Nordisk A/S Glp-1 compositions and uses thereof
US11478533B2 (en) * 2020-04-27 2022-10-25 Novo Nordisk A/S Semaglutide for use in medicine
US20240197700A1 (en) * 2021-03-29 2024-06-20 Sanford Health Methods and Compositions for Treating Lysosomal Storage Disorders
AU2023285400A1 (en) * 2022-06-08 2024-12-05 Zydus Lifesciences Limited Reusable multi-dose, variable dose, single pen injector for type 2 diabetes and weight management
WO2024249659A2 (en) * 2023-05-30 2024-12-05 The Medical College Of Wisconsin, Inc. Methods for weight loss and/or reducing weight gain
WO2024252134A1 (en) * 2023-06-05 2024-12-12 Closed Loop Medicine Ltd Dosing of incretin pathway drugs

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US6268343B1 (en) 1996-08-30 2001-07-31 Novo Nordisk A/S Derivatives of GLP-1 analogs
DK1412384T3 (da) 2001-06-28 2008-04-28 Novo Nordisk As Stabil formulering af modificeret GLP-1
KR101241862B1 (ko) 2003-09-19 2013-03-13 노보 노르디스크 에이/에스 신규 glp-1 유도체
CN102784386A (zh) 2003-11-20 2012-11-21 诺沃挪第克公司 对于生产和用于注射装置中是最佳的含有丙二醇的肽制剂
JP5175103B2 (ja) 2004-11-12 2013-04-03 ノヴォ ノルディスク アー/エス 安定なペプチド製剤
TWI372629B (en) 2005-03-18 2012-09-21 Novo Nordisk As Acylated glp-1 compounds
KR101384456B1 (ko) 2005-09-14 2014-04-10 맨카인드 코포레이션 활성제에 대한 결정질 미립자 표면의 친화력의 증가를 기반으로 하는 약물 제제화의 방법
MX2008013216A (es) 2006-04-14 2008-10-27 Mannkind Corp Formulaciones farmaceuticas de peptido-1 tipo glucagon (glp-1).
EP2121897A4 (en) 2007-03-20 2010-03-31 Nippon Kayaku Kk METHOD FOR MONITORING THE DRUG EFFECT ON DIABETES PATIENTS USING AN ASSAY FOR 1,5-ANHYDRO-D-GLUCITOL
EP2190873B1 (en) 2007-09-05 2015-07-22 Novo Nordisk A/S Truncated glp-1 derivatives and their therapeutical use
LT2373681T (lt) 2008-12-10 2017-04-10 Glaxosmithkline Llc Albiglutido farmacinės kompozicijos
NZ594044A (en) 2009-02-13 2014-08-29 Boehringer Ingelheim Int Antidiabetic medications comprising a dpp-4 inhibitor (linagliptin) optionally in combination with other antidiabetics
JP2013514322A (ja) 2009-12-16 2013-04-25 ノヴォ ノルディスク アー/エス 修飾されたn末端を有するglp−1受容体アゴニスト化合物
KR101819609B1 (ko) 2010-05-05 2018-01-17 베링거 인겔하임 인터내셔날 게엠베하 체중 감소 치료에 후속하는 dpp-4 억제제에 의한 순차적 병용 요법
WO2012016419A1 (zh) 2010-08-06 2012-02-09 浙江贝达药业有限公司 Glp-1衍生物及其应用
PL3326620T3 (pl) 2010-12-16 2020-08-24 Novo Nordisk A/S Kompozycje stałe zawierające agonistę glp-1 i sól kwasu n-(8-(2- hydroksybenzoilo)amino)kaprylowego
AR084558A1 (es) 2010-12-22 2013-05-22 Marcadia Biotech Metodos para tratar trastornos metabolicos y obesidad con peptidos basados en glucagon activos para el receptor de peptido insulinotropico dependiente de glucosa (gip)/peptido-1 similar al glucagon (glp-1)
US20130035281A1 (en) 2011-02-09 2013-02-07 Boehringer Ingelheim International Gmbh Pharmaceutical composition, methods for treating and uses thereof
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UA116189C2 (uk) 2011-05-02 2018-02-26 Мілленніум Фармасьютікалз, Інк. КОМПОЗИЦІЯ АНТИ-α4β7 АНТИТІЛА
CN102229668A (zh) 2011-06-03 2011-11-02 浙江贝达药业有限公司 一种glp-1衍生物及其应用
JP2014520159A (ja) 2011-06-24 2014-08-21 アミリン・ファーマシューティカルズ,リミテッド・ライアビリティ・カンパニー Glp−1受容体アゴニストの徐放性製剤による糖尿病の治療方法
JP6250034B2 (ja) * 2012-05-08 2017-12-20 ノヴォ ノルディスク アー/エス 二重アシル化されたglp−1誘導体
DK2866825T3 (da) * 2012-07-01 2020-06-08 Novo Nordisk As Anvendelse af langstidsvirkende glp-1-peptider
PT2991671T (pt) * 2013-05-02 2018-11-05 Novo Nordisk As Dosagem oral de compostos de glp-1
MY197023A (en) 2015-12-23 2023-05-22 Amgen Inc Method of treating or ameliorating metabolic disorders using binding proteins for gastric inhibitory peptide receptor (gipr) in combination with glp-1 agonists
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MA50358A (fr) * 2017-10-12 2020-08-19 Novo Nordisk As Sémaglutide en thérapie médicale

Also Published As

Publication number Publication date
WO2019072941A1 (en) 2019-04-18
MX2020003049A (es) 2020-07-27
AU2025203535A1 (en) 2025-06-05
CL2020000812A1 (es) 2020-08-14
JP7475398B2 (ja) 2024-04-26
JP2022132414A (ja) 2022-09-08
JP2020536854A (ja) 2020-12-17
ZA202503388B (en) 2025-09-25
ZA202503387B (en) 2025-09-25
RU2020114960A3 (OSRAM) 2022-02-11
IL273470A (en) 2020-05-31
US12029779B2 (en) 2024-07-09
IL322969A (en) 2025-10-01
US12295988B2 (en) 2025-05-13
TW201914611A (zh) 2019-04-16
MX2025002189A (es) 2025-04-02
JP7148605B2 (ja) 2022-10-05
IL322968A (en) 2025-10-01
AU2018348929A1 (en) 2020-05-07
EP3694538A1 (en) 2020-08-19
BR112020006246A2 (pt) 2021-03-30
CN111212657A (zh) 2020-05-29
US20240316159A1 (en) 2024-09-26
ZA202503350B (en) 2025-09-25
CA3078652A1 (en) 2019-04-18
CN119950682A (zh) 2025-05-09
US20240415935A1 (en) 2024-12-19
US20200237876A1 (en) 2020-07-30
MX2025002188A (es) 2025-04-02
MA50358A (fr) 2020-08-19
AU2018348929B2 (en) 2025-02-27
CN119838000A (zh) 2025-04-18
MY204827A (en) 2024-09-18
CN120241968A (zh) 2025-07-04
KR20200069316A (ko) 2020-06-16
US20250235511A1 (en) 2025-07-24
SG11202002841PA (en) 2020-04-29
RU2020114960A (ru) 2021-10-28
PH12020550185A1 (en) 2021-03-01

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