TWI767937B - 外核苷酸酶抑制劑及其使用方法 - Google Patents
外核苷酸酶抑制劑及其使用方法 Download PDFInfo
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- TWI767937B TWI767937B TW106130807A TW106130807A TWI767937B TW I767937 B TWI767937 B TW I767937B TW 106130807 A TW106130807 A TW 106130807A TW 106130807 A TW106130807 A TW 106130807A TW I767937 B TWI767937 B TW I767937B
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| TW202014182A (zh) * | 2018-04-30 | 2020-04-16 | 美商歐瑞克製藥公司 | Cd73抑制劑 |
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| CN112888696B (zh) * | 2018-06-21 | 2024-04-16 | 德琪医疗有限公司 | 外核苷酸酶抑制剂及其使用方法 |
| US11332492B2 (en) | 2018-08-28 | 2022-05-17 | Jiangsu Hengrui Medicine Co., Ltd. | CD73 inhibitors and therapeutic uses thereof |
| MX2021002878A (es) | 2018-09-11 | 2021-08-16 | Risen Suzhou Pharma Tech Co Ltd | Inhibidores de cd73 y usos farmaceuticos de los mismos. |
| US11530234B2 (en) | 2018-09-11 | 2022-12-20 | Risen (Suzhou) Pharma Tech Co., Ltd. | CD73 inhibitors and pharmaceutical uses thereof |
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| EP3939988A4 (en) * | 2019-03-20 | 2022-08-24 | Korea Research Institute of Chemical Technology | Pharmaceutical composition comprising novel azolopyrimidine heterocyclic compound as active ingredient |
| CN113905743B (zh) * | 2019-03-29 | 2024-04-16 | 江苏恒瑞医药股份有限公司 | Cd73抑制剂及其治疗用途 |
| WO2020210938A1 (en) * | 2019-04-15 | 2020-10-22 | Bioardis Llc | Quinazoline derivatives as cd73 inhibitors |
| KR20220024629A (ko) * | 2019-06-20 | 2022-03-03 | 칼리테라 바이오사이언시즈, 인코포레이티드 | 엑토뉴클레오티다제 억제제 및 이의 사용 방법 |
| MX2022005256A (es) * | 2019-10-30 | 2022-08-25 | Oric Pharmaceuticals Inc | Inhibidores de cd73. |
| WO2022052886A1 (zh) * | 2020-09-08 | 2022-03-17 | 贝达药业股份有限公司 | Cd73抑制剂及其在医药上的应用 |
| CN114099698B (zh) * | 2021-11-26 | 2024-02-09 | 山东大学齐鲁医院 | 一种pH敏感脂质体及其制备方法与应用 |
| AU2023252914A1 (en) | 2022-04-13 | 2024-10-17 | Arcus Biosciences, Inc. | Combination therapy for treating trop-2 expressing cancers |
| CN117430651A (zh) * | 2022-07-21 | 2024-01-23 | 武汉精准智药科技有限公司 | 单磷酸核苷类化合物及其制备方法 |
| CN115611954A (zh) * | 2022-12-19 | 2023-01-17 | 天津奥瑞芙生物医药有限公司 | 一种5′-o-(4,4′-二甲氧基三苯甲基)-核苷的制备方法 |
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| WO2025162964A1 (en) | 2024-01-30 | 2025-08-07 | Institut National de la Santé et de la Recherche Médicale | Methods for the treatment of endometriosis |
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| WO2004096233A2 (en) * | 2003-04-25 | 2004-11-11 | Gilead Sciences, Inc. | Nucleoside phosphonate conjugates |
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| JP2019530669A (ja) | 2019-10-24 |
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| US20180072742A1 (en) | 2018-03-15 |
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