TWI661835B - 選擇性ｐｙｙ化合物及其用途 - Google Patents
選擇性ｐｙｙ化合物及其用途 Download PDFInfo
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- TWI661835B TWI661835B TW103139321A TW103139321A TWI661835B TW I661835 B TWI661835 B TW I661835B TW 103139321 A TW103139321 A TW 103139321A TW 103139321 A TW103139321 A TW 103139321A TW I661835 B TWI661835 B TW I661835B
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- 230000014616 translation Effects 0.000 description 1
- ZGYICYBLPGRURT-UHFFFAOYSA-N tri(propan-2-yl)silicon Chemical compound CC(C)[Si](C(C)C)C(C)C ZGYICYBLPGRURT-UHFFFAOYSA-N 0.000 description 1
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Classifications
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- A61K38/1703—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
- A61K38/1709—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates from mammals
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- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
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Landscapes
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| IL302745A (en) * | 2020-11-09 | 2023-07-01 | Embark Biotech Aps | Compounds and their use in the treatment of tachykinin receptor mediated disorders |
| JP2025526148A (ja) | 2022-08-18 | 2025-08-07 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 長時間作用型ｇｌｐ－１／グルカゴン受容体アゴニスト及びｎｐｙ２受容体アゴニストを含む組合せ治療 |
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| EP2992008B1 (en) | 2013-05-02 | 2019-04-10 | GlaxoSmithKline Intellectual Property Development Limited | Therapeutic peptides |
| WO2015071355A1 (en) | 2013-11-15 | 2015-05-21 | Novo Nordisk A/S | Selective pyy compounds and uses thereof |
| US10583172B2 (en) | 2013-11-15 | 2020-03-10 | Novo Nordisk A/S | HPYY(1-36) having a beta-homoarginine substitution at position 35 |
| MX392572B (es) * | 2015-06-12 | 2025-03-24 | Novo Nordisk As | Compuestos del péptido yy (pyy) selectivos y sus usos. |
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| CN102573888A (zh) * | 2009-09-18 | 2012-07-11 | 诺和诺德公司 | 长效y2 受体激动剂 |
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| PL3068421T3 (pl) | 2019-11-29 |
| AU2014350197A1 (en) | 2016-05-05 |
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| IL245045A0 (en) | 2016-05-31 |
| CN105722526A (zh) | 2016-06-29 |
| BR112016010383A2 (pt) | 2017-12-05 |
| EP3068421B1 (en) | 2019-04-17 |
| AU2014350197B2 (en) | 2018-10-04 |
| SI3068421T1 (sl) | 2019-08-30 |
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| US10246497B2 (en) | 2019-04-02 |
| EP3068421A1 (en) | 2016-09-21 |
| US20150152150A1 (en) | 2015-06-04 |
| KR20160075819A (ko) | 2016-06-29 |
| MX369818B (es) | 2019-11-22 |
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