TWI542590B - １，２-雙取代雜環化合物 - Google Patents

１，２-雙取代雜環化合物 Download PDF

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TWI542590B
TWI542590B TW103127120A TW103127120A TWI542590B TW I542590 B TWI542590 B TW I542590B TW 103127120 A TW103127120 A TW 103127120A TW 103127120 A TW103127120 A TW 103127120A TW I542590 B TWI542590 B TW I542590B
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Taiwan
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etoac
phenyl
group
mmol
water
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TW103127120A
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Chinese (zh)
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TW201506028A (zh
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愛咪 瑞普卡
吉登 莎普羅
理查 雀斯沃斯
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福倫製藥股份有限公司
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
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    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/47—Quinolines; Isoquinolines
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    • A61K31/50—Pyridazines; Hydrogenated pyridazines
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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  • Orthopedic Medicine & Surgery (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
TW103127120A 2008-06-25 2009-06-25 １，２-雙取代雜環化合物 TWI542590B (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US7559408P 2008-06-25 2008-06-25
US10916208P 2008-10-28 2008-10-28
US13886608P 2008-12-18 2008-12-18
US17641309P 2009-05-07 2009-05-07

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TW201506028A TW201506028A (zh) 2015-02-16
TWI542590B true TWI542590B (zh) 2016-07-21

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US (7) US8071595B2 (enExample)
EP (2) EP2297133B1 (enExample)
JP (4) JP5658664B2 (enExample)
KR (2) KR20110031355A (enExample)
CN (2) CN102131801B (enExample)
AU (2) AU2009262241B2 (enExample)
BR (2) BRPI0914772A2 (enExample)
CA (2) CA2729259A1 (enExample)
MX (2) MX2011000175A (enExample)
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PL2617420T3 (pl) * 2009-05-07 2016-04-29 Forum Pharmaceuticals Inc Heterocykliczne związki fenoksymetylu
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JP5785548B2 (ja) 2010-08-04 2015-09-30 武田薬品工業株式会社 縮合複素環化合物
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US9029399B2 (en) 2011-04-28 2015-05-12 Novartis Ag 17α-hydroxylase/C17,20-lyase inhibitors
WO2013047411A1 (ja) * 2011-09-29 2013-04-04 富士フイルム株式会社 新規なトリアジン誘導体、紫外線吸収剤
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