TW201823235A - 西克里維羅（ｃｅｎｉｃｒｉｖｉｒｏｃ）甲磺酸鹽之固體型式和製造西克里維羅甲磺酸鹽之固體型式的方法 - Google Patents
西克里維羅（ｃｅｎｉｃｒｉｖｉｒｏｃ）甲磺酸鹽之固體型式和製造西克里維羅甲磺酸鹽之固體型式的方法 Download PDFInfo
- Publication number
- TW201823235A TW201823235A TW106129555A TW106129555A TW201823235A TW 201823235 A TW201823235 A TW 201823235A TW 106129555 A TW106129555 A TW 106129555A TW 106129555 A TW106129555 A TW 106129555A TW 201823235 A TW201823235 A TW 201823235A
- Authority
- TW
- Taiwan
- Prior art keywords
- crystalline form
- msoh
- compound
- patent application
- scope
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
- C07C309/01—Sulfonic acids
- C07C309/02—Sulfonic acids having sulfo groups bound to acyclic carbon atoms
- C07C309/03—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C309/04—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton containing only one sulfo group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Gastroenterology & Hepatology (AREA)
- Epidemiology (AREA)
- Urology & Nephrology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201662382153P | 2016-08-31 | 2016-08-31 | |
| US62/382,153 | 2016-08-31 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW201823235A true TW201823235A (zh) | 2018-07-01 |
Family
ID=61241572
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW106129555A TW201823235A (zh) | 2016-08-31 | 2017-08-30 | 西克里維羅（ｃｅｎｉｃｒｉｖｉｒｏｃ）甲磺酸鹽之固體型式和製造西克里維羅甲磺酸鹽之固體型式的方法 |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US10301287B2 (enExample) |
| EP (1) | EP3506896A4 (enExample) |
| JP (2) | JP2019526628A (enExample) |
| KR (1) | KR20190057066A (enExample) |
| CN (1) | CN110167550A (enExample) |
| AU (1) | AU2017321594A1 (enExample) |
| BR (1) | BR112019003987A2 (enExample) |
| CA (1) | CA3034606A1 (enExample) |
| MX (1) | MX2019002057A (enExample) |
| RU (1) | RU2019109019A (enExample) |
| SG (1) | SG11201901438VA (enExample) |
| TW (1) | TW201823235A (enExample) |
| WO (1) | WO2018045043A1 (enExample) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2019238041A1 (zh) * | 2018-06-12 | 2019-12-19 | 南京明德新药研发有限公司 | 一种丙烯酰胺类化合物的晶型及其制备方法 |
| WO2019245517A1 (en) * | 2018-06-18 | 2019-12-26 | Hewlett-Packard Development Company, L.P. | Three-dimensional printing |
| US11613670B2 (en) | 2018-06-18 | 2023-03-28 | Hewlett-Packard Development Company, L.P. | Three-dimensional printing |
| US11591486B2 (en) | 2018-06-19 | 2023-02-28 | Hewlett-Packard Development Company, L.P. | Three-dimensional printing |
| WO2019245589A1 (en) | 2018-06-19 | 2019-12-26 | Hewlett-Packard Development Company, L.P. | Three-dimensional printing |
| WO2019245534A1 (en) * | 2018-06-19 | 2019-12-26 | Hewlett-Packard Development Company, L.P. | Three-dimensional printing |
| KR20210053921A (ko) * | 2018-08-31 | 2021-05-12 | 에보니크 오퍼레이션즈 게엠베하 | 중합체 분말을 제조하는 방법 |
| WO2021133811A1 (en) | 2019-12-26 | 2021-07-01 | Teva Pharmaceuticals International Gmbh | Solid state forms of cenicriviroc and process for preparation thereof |
| EP4159730A4 (en) | 2020-05-22 | 2024-05-01 | Medshine Discovery Inc. | PYRIDINE DERIVATIVE AND APPLICATION THEREOF |
| US20240124690A1 (en) * | 2021-02-22 | 2024-04-18 | Asahi Kasei Kabushiki Kaisha | Composition Containing Cellulose Nanofibers |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS62265270A (ja) | 1986-05-13 | 1987-11-18 | Zeria Shinyaku Kogyo Kk | 新規イミダゾ−ル誘導体およびそれらを有効成分とする抗潰瘍剤 |
| AU2808495A (en) | 1994-07-04 | 1996-01-25 | Takeda Chemical Industries Ltd. | Phosphonic acid compounds, their production and use |
| WO1999032100A2 (en) | 1997-12-19 | 1999-07-01 | Takeda Chemical Industries, Ltd. | Pharmaceutical composition for antagonizing ccr5 comprising anilide derivative |
| EP1104416A2 (en) | 1998-08-20 | 2001-06-06 | Takeda Chemical Industries, Ltd. | Quaternary ammonium salts and their use as anti-hiv agents |
| CA2384145A1 (en) | 1999-09-06 | 2001-03-15 | Takeda Chemical Industries, Ltd. | Process for the preparation of 2,3-dihydroazepine compounds |
| US7371772B2 (en) | 2001-08-08 | 2008-05-13 | Takeda Pharmaceutical Company Limited | Bicyclic compound, production and use thereof |
| JP2004123694A (ja) * | 2002-03-12 | 2004-04-22 | Takeda Chem Ind Ltd | 光学活性スルホキシド誘導体の製造法 |
| EP1728504B1 (en) | 2004-03-24 | 2013-07-31 | Takeda Pharmaceutical Company Limited | Emulsion stabilizer |
| JP2007269628A (ja) * | 2004-05-28 | 2007-10-18 | Takeda Chem Ind Ltd | 医薬化合物の結晶 |
| GT200600148A (es) | 2005-04-14 | 2006-11-22 | Metodos para el tratamiento y la prevencion de fibrosis | |
| CA2818308A1 (en) | 2010-11-18 | 2012-05-24 | Yale University | Bifunctional molecules with antibody-recruiting and entry inhibitory activity against the human immunodeficiency virus |
| AU2013257951A1 (en) | 2012-05-11 | 2015-01-22 | Akron Molecules Ag | Use of compounds for the treatment of pain |
| KR20160013068A (ko) | 2013-05-15 | 2016-02-03 | 토비라 쎄라퓨틱스, 인크. | 세니크리비록 조성물 및 이들을 만들고 이용하는 방법 |
| CA2941411A1 (en) * | 2014-03-21 | 2015-09-24 | Tobira Therapeutics, Inc. | Cenicriviroc for the treatment of fibrosis |
| WO2015187663A1 (en) * | 2014-06-02 | 2015-12-10 | Tobira Therapeutics, Inc. | Cenicriviroc for the treatment of hiv-2 infection |
| SG11201704837VA (en) | 2014-12-23 | 2017-07-28 | Tobira Therapeutics Inc | Process of making cenicriviroc and related analogs |
-
2017
- 2017-08-30 JP JP2019531594A patent/JP2019526628A/ja active Pending
- 2017-08-30 CA CA3034606A patent/CA3034606A1/en not_active Abandoned
- 2017-08-30 KR KR1020197008786A patent/KR20190057066A/ko not_active Withdrawn
- 2017-08-30 EP EP17847477.1A patent/EP3506896A4/en not_active Withdrawn
- 2017-08-30 MX MX2019002057A patent/MX2019002057A/es unknown
- 2017-08-30 AU AU2017321594A patent/AU2017321594A1/en not_active Abandoned
- 2017-08-30 BR BR112019003987A patent/BR112019003987A2/pt not_active Application Discontinuation
- 2017-08-30 US US15/691,191 patent/US10301287B2/en active Active
- 2017-08-30 WO PCT/US2017/049400 patent/WO2018045043A1/en not_active Ceased
- 2017-08-30 CN CN201780061529.6A patent/CN110167550A/zh active Pending
- 2017-08-30 RU RU2019109019A patent/RU2019109019A/ru not_active Application Discontinuation
- 2017-08-30 SG SG11201901438VA patent/SG11201901438VA/en unknown
- 2017-08-30 TW TW106129555A patent/TW201823235A/zh unknown
-
2022
- 2022-07-14 JP JP2022113230A patent/JP2022137223A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| JP2019526628A (ja) | 2019-09-19 |
| JP2022137223A (ja) | 2022-09-21 |
| RU2019109019A3 (enExample) | 2021-08-23 |
| WO2018045043A1 (en) | 2018-03-08 |
| RU2019109019A (ru) | 2020-10-01 |
| US20180057481A1 (en) | 2018-03-01 |
| SG11201901438VA (en) | 2019-03-28 |
| CN110167550A (zh) | 2019-08-23 |
| KR20190057066A (ko) | 2019-05-27 |
| AU2017321594A1 (en) | 2019-04-18 |
| US10301287B2 (en) | 2019-05-28 |
| BR112019003987A2 (pt) | 2019-05-28 |
| EP3506896A1 (en) | 2019-07-10 |
| MX2019002057A (es) | 2019-11-18 |
| EP3506896A4 (en) | 2020-08-26 |
| CA3034606A1 (en) | 2018-03-08 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| US10301287B2 (en) | Solid forms of cenicriviroc mesylate and processes of making solid forms of cenicriviroc mesylate | |
| JP6081763B2 (ja) | ダサチニブ多形体およびその調製プロセス | |
| US11149017B2 (en) | Solid state forms of apalutamide | |
| EA034409B1 (ru) | Способы получения кристаллического фенилацетата l-орнитина | |
| RU2704795C2 (ru) | Кристаллическая форма бисульфата ингибитора jak и способ ее получения | |
| WO2011095059A1 (zh) | 达沙替尼多晶型物及其制备方法和药物组合物 | |
| JP2021181446A (ja) | （ｓ）−２−（（２−（（ｓ）−４−（ジフルオロメチル）−２−オキソオキサゾリジン−３−イル）−５，６−ジヒドロベンゾ［ｆ］イミダゾ［１，２−ｄ］［１，４］オキサゼピン−９−イル）アミノ）プロパンアミドの多形体及び固体形態と、生産方法 | |
| WO2021143841A1 (zh) | 三并环类pde3/pde4双重抑制剂化合物的药物组合物 | |
| US12209073B2 (en) | Polymorphs of a dihydroorotate dehydrogenase (DHOD) inhibitor | |
| JP2005298424A (ja) | エパルレスタット結晶の製造方法 | |
| TW202545917A (zh) | Ｎ－［（１ｓ，２ｅ）－１－環丙基－３－（甲磺醯基）丙－２－烯－１－基］－２－（１，１－二氟乙基）－４－苯氧基嘧啶－５－甲醯胺的新固體形式 | |
| TW202434600A (zh) | 磺醯胺衍生物結晶形式及其製備方法 | |
| WO2025002335A1 (zh) | Baxdrostat的晶型及其制备方法和用途 | |
| EP4486458A1 (en) | Crystalline forms of trilaciclib and trilaciclib salts | |
| KR20190029601A (ko) | 고체 형태의 ttk 억제제 | |
| US20140073791A1 (en) | Novel salts of sitagliptin, process for the preparation and pharmaceutical composition thereof | |
| US7655800B2 (en) | Crystalline 1H-imidazo[4,5-b]pyridin-5-amine, 7-[5-[(cyclohexylmethylamino)-methyl]-1H-indol-2-yl]-2-methyl, sulfate (1:1), trihydrate and its pharmaceutical uses | |
| EP4477652A1 (en) | Polymorph as thyroid hormone receptor agonists and use thereof | |
| WO2019233328A1 (zh) | 4-苯基噻唑衍生物的晶型及其制备方法 | |
| WO2019086008A1 (zh) | 一种苯并三氮唑衍生物的晶型及其制备方法和用途 | |
| WO2024179558A1 (zh) | Pirtobrutinib的晶型及其制备方法和用途 | |
| TW202543633A (zh) | 喹唑啉酮衍生物的晶型及其製備方法和應用 | |
| TW202606690A (zh) | 吡啶并吡唑衍生物的晶型物、藥物組合物及其用途 | |
| KR20260032991A (ko) | (3r)-n-[2-시아노-4-플루오로-3-(3-메틸-4-옥소-퀴나졸린-6-일)옥시-페닐]-3-플루오로-피롤리딘-1-설폰아미드의신규 고체 형태 | |
| TW202333694A (zh) | 稠環衍生物的晶型、其製備方法及其應用 |