TW201536284A - 使用黃嘌呤氧化酶抑制劑之治療方法與組成物 - Google Patents
使用黃嘌呤氧化酶抑制劑之治療方法與組成物 Download PDFInfo
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- TW201536284A TW201536284A TW103119057A TW103119057A TW201536284A TW 201536284 A TW201536284 A TW 201536284A TW 103119057 A TW103119057 A TW 103119057A TW 103119057 A TW103119057 A TW 103119057A TW 201536284 A TW201536284 A TW 201536284A
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
- A61K9/1676—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface having a drug-free core with discrete complete coating layer containing drug
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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- A61P13/12—Drugs for disorders of the urinary system of the kidneys
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
Landscapes
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
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- Chemical & Material Sciences (AREA)
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- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Immunology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US201361839609P | 2013-06-26 | 2013-06-26 |
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| TW201536284A true TW201536284A (zh) | 2015-10-01 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| MX2018005345A (es) * | 2015-10-28 | 2018-08-14 | Sun Pharmaceutical Ind Ltd | Composiciones farmaceuticas de dimetil fumarato. |
| CN105769766B (zh) * | 2016-03-24 | 2018-07-06 | 长沙佰顺生物科技有限公司 | 一种托匹司他纳米乳及其制备方法 |
| JP7108384B2 (ja) * | 2016-07-13 | 2022-07-28 | 日本ケミファ株式会社 | ２－［３－シアノ－４－（２－メチルプロポキシ）フェニル］－４－メチルチアゾール－５－カルボン酸の口腔内崩壊錠 |
| DK3484862T3 (da) * | 2016-07-18 | 2021-11-08 | Arthrosi Therapeutics Inc | Forbindelser, sammensætninger og fremgangsmåder til behandling eller forebyggelse af et symptom, der er forbundet med gigt eller hyperurikæmi |
| US12419854B2 (en) | 2018-12-06 | 2025-09-23 | Arthrosi Therapeutics, Inc. | Methods for treating or preventing gout or hyperuricemia |
| SG11202105745UA (en) | 2018-12-06 | 2021-06-29 | Arthrosi Therapeutics Inc | Crystalline forms of a compound for treating or preventing gout or hyperuricemia |
| CN113924145A (zh) * | 2019-06-04 | 2022-01-11 | 日本化学药品株式会社 | 痛风或高尿酸血症的治疗药 |
| PE20240242A1 (es) * | 2021-06-15 | 2024-02-16 | Lg Chemical Ltd | Una composicion farmaceutica que comprende acido 1-(3-ciano-1-isopropil-indol-5-il)pirazol-4-carboxilico |
| CN115252567A (zh) * | 2022-07-08 | 2022-11-01 | 广西纯正堂制药有限公司 | 非布司他渗透泵缓释片及其制备方法 |
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| GB1478759A (en) | 1974-11-18 | 1977-07-06 | Alza Corp | Process for forming outlet passageways in pills using a laser |
| US4200098A (en) | 1978-10-23 | 1980-04-29 | Alza Corporation | Osmotic system with distribution zone for dispensing beneficial agent |
| US5286497A (en) | 1991-05-20 | 1994-02-15 | Carderm Capital L.P. | Diltiazem formulation |
| US5573776A (en) | 1992-12-02 | 1996-11-12 | Alza Corporation | Oral osmotic device with hydrogel driving member |
| US5544163A (en) | 1994-03-08 | 1996-08-06 | Excel, Inc. | Expandable telecommunications system |
| DK1488790T3 (da) | 2002-03-28 | 2014-10-13 | Teijin Pharma Ltd | Fast præparat indeholdende en enkeltkrystalform A af etthiazolcarboxylsyrederivat |
| PL1757610T3 (pl) | 2004-06-14 | 2011-10-31 | Nippon Chemiphar Co | Skondensowana pochodna pirymidyny oraz inhibitor oksydazy ksantynowej |
| WO2007043457A1 (ja) | 2005-10-07 | 2007-04-19 | Astellas Pharma Inc. | トリアリールカルボン酸誘導体 |
| CN101646440A (zh) * | 2007-01-19 | 2010-02-10 | 武田制药北美公司 | 使用黄嘌呤氧化还原酶抑制剂和抗炎剂预防痛风突发或减少痛风突发次数的方法 |
| KR101772963B1 (ko) | 2009-03-31 | 2017-08-31 | 깃세이 야쿠힌 고교 가부시키가이샤 | 인돌리진 유도체 및 그 의약용도 |
| CN101773498B (zh) * | 2009-12-30 | 2012-06-20 | 青岛黄海制药有限责任公司 | 一种含有非布司他的口服缓控释制剂的制备方法 |
| JP5865904B2 (ja) * | 2010-06-16 | 2016-02-17 | タケダ ファーマシューティカルズ ユー．エス．エー． インコーポレイティド | キサンチンオキシドレダクターゼ阻害剤またはキサンチンオキシダーゼ阻害剤の新規の調節放出剤形 |
| MX339452B (es) | 2010-06-16 | 2016-05-27 | Teijin Pharma Ltd | Tableta con nucleo recubierto de liberacion controlada. |
| CN102641255A (zh) * | 2012-05-08 | 2012-08-22 | 南方医科大学 | 一种治疗痛风的非布索坦渗透泵控释片及其制备方法 |
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2014
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- 2014-05-30 TW TW103119057A patent/TW201536284A/zh unknown
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- 2014-05-30 JP JP2016517049A patent/JP2016520133A/ja active Pending
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2017
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2019
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Also Published As
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| CN105579037A (zh) | 2016-05-11 |
| JP2016520133A (ja) | 2016-07-11 |
| WO2014194226A3 (en) | 2015-05-14 |
| SG11201509738RA (en) | 2015-12-30 |
| MX2015016494A (es) | 2016-11-18 |
| US20140357683A1 (en) | 2014-12-04 |
| SG10201709955PA (en) | 2018-01-30 |
| WO2014194226A2 (en) | 2014-12-04 |
| PH12015502679A1 (en) | 2016-03-07 |
| JP2019108356A (ja) | 2019-07-04 |
| CA2913755A1 (en) | 2014-12-04 |
| US20180311217A1 (en) | 2018-11-01 |
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