TW201414735A - 三環喹啉及喹噁啉衍生物 - Google Patents

三環喹啉及喹噁啉衍生物 Download PDF

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Publication number
TW201414735A
TW201414735A TW102133403A TW102133403A TW201414735A TW 201414735 A TW201414735 A TW 201414735A TW 102133403 A TW102133403 A TW 102133403A TW 102133403 A TW102133403 A TW 102133403A TW 201414735 A TW201414735 A TW 201414735A
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TW
Taiwan
Prior art keywords
fluorinated
group
alkyl
ring
alkoxy
Prior art date
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TW102133403A
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English (en)
Chinese (zh)
Inventor
Hannes Koolman
Wilfried Braje
Helmut Mack
Andreas Haupt
Ana Lucia Relo
Karla Drescher
Margaretha Henrica Maria Bakker
Viktor Lakics
Carolin Hoft
Ru-Xu Xu
xiao-na Zhao
Original Assignee
Abbvie Deutschland
Abbvie Inc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50275085&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TW201414735(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from CN201310410951.1A external-priority patent/CN104418862A/zh
Application filed by Abbvie Deutschland, Abbvie Inc filed Critical Abbvie Deutschland
Publication of TW201414735A publication Critical patent/TW201414735A/zh

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06Peri-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P13/00Drugs for disorders of the urinary system
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    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
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    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
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    • A61P17/00Drugs for dermatological disorders
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    • A61P17/00Drugs for dermatological disorders
    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P17/06Antipsoriatics
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/06Peri-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/16Peri-condensed systems

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Pain & Pain Management (AREA)
  • Hematology (AREA)
  • Dermatology (AREA)
  • Reproductive Health (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Rheumatology (AREA)
  • Anesthesiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Emergency Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
TW102133403A 2012-09-14 2013-09-14 三環喹啉及喹噁啉衍生物 TW201414735A (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201261701531P 2012-09-14 2012-09-14
US201261701514P 2012-09-14 2012-09-14
US201361793033P 2013-03-15 2013-03-15
CN201310410951.1A CN104418862A (zh) 2013-09-11 2013-09-11 三环喹啉和喹喔啉衍生物

Publications (1)

Publication Number Publication Date
TW201414735A true TW201414735A (zh) 2014-04-16

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Family Applications (1)

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TW102133403A TW201414735A (zh) 2012-09-14 2013-09-14 三環喹啉及喹噁啉衍生物

Country Status (26)

Country Link
US (3) US10118926B2 (en:Method)
EP (1) EP2895485A1 (en:Method)
JP (1) JP6290217B2 (en:Method)
KR (1) KR20150056608A (en:Method)
CN (1) CN104995191A (en:Method)
AR (1) AR092568A1 (en:Method)
AU (2) AU2013314279B2 (en:Method)
BR (1) BR112015005743A2 (en:Method)
CA (1) CA2884548A1 (en:Method)
CL (1) CL2015000628A1 (en:Method)
CR (1) CR20150186A (en:Method)
DO (1) DOP2015000058A (en:Method)
EC (1) ECSP15012766A (en:Method)
HK (1) HK1212684A1 (en:Method)
IL (1) IL237726A0 (en:Method)
IN (1) IN2015DN02070A (en:Method)
MX (1) MX2015003364A (en:Method)
NZ (1) NZ631187A (en:Method)
PE (1) PE20150777A1 (en:Method)
PH (1) PH12015500551A1 (en:Method)
RU (1) RU2015113558A (en:Method)
SG (1) SG11201501894VA (en:Method)
TW (1) TW201414735A (en:Method)
UA (1) UA116216C2 (en:Method)
UY (1) UY35029A (en:Method)
WO (1) WO2014041131A1 (en:Method)

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KR20210104785A (ko) 2018-12-17 2021-08-25 인트라-셀룰라 써래피스, 인코퍼레이티드. 유기 화합물
EP3897621A4 (en) 2018-12-21 2022-09-07 Intra-Cellular Therapies, Inc. Organic compounds
JP7377871B2 (ja) 2018-12-21 2023-11-10 イントラ-セルラー・セラピーズ・インコーポレイテッド 有機化合物
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