TW201326194A - Ｇｌｐ－１胃泌素受體促效劑肽結合物 - Google Patents

Ｇｌｐ－１胃泌素受體促效劑肽結合物 Download PDF

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Publication number
TW201326194A
TW201326194A TW101140873A TW101140873A TW201326194A TW 201326194 A TW201326194 A TW 201326194A TW 101140873 A TW101140873 A TW 101140873A TW 101140873 A TW101140873 A TW 101140873A TW 201326194 A TW201326194 A TW 201326194A
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TW
Taiwan
Prior art keywords
8ado
pharmaceutically acceptable
glu
solvate
disease
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TW101140873A
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English (en)
Chinese (zh)
Inventor
Trine Skovlund Neerup
Jakob Lind Tolborg
Keld Fosgerau
Torben Oesterlund
Dorthe Lennert Almholt
Lone Larsen
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Zealand Pharma As
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Publication of TW201326194A publication Critical patent/TW201326194A/zh

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    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
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    • A61K47/62—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being a protein, peptide or polyamino acid
    • A61K47/64—Drug-peptide, drug-protein or drug-polyamino acid conjugates, i.e. the modifying agent being a peptide, protein or polyamino acid which is covalently bonded or complexed to a therapeutically active agent
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  • Proteomics, Peptides & Aminoacids (AREA)
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  • Endocrinology (AREA)
  • Immunology (AREA)
  • Zoology (AREA)
  • Biophysics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
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  • Urology & Nephrology (AREA)
  • Genetics & Genomics (AREA)
  • Vascular Medicine (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Ophthalmology & Optometry (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
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TW101140873A 2011-11-03 2012-11-02 Ｇｌｐ－１胃泌素受體促效劑肽結合物 TW201326194A (zh)

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US201161555435P 2011-11-03 2011-11-03

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US (2) US9259477B2 (enExample)
EP (1) EP2773377B1 (enExample)
JP (1) JP6359972B2 (enExample)
KR (1) KR20140100947A (enExample)
CN (1) CN104144704B (enExample)
AR (1) AR088636A1 (enExample)
AU (1) AU2012331053A1 (enExample)
BR (1) BR112014010780A2 (enExample)
CA (1) CA2853884A1 (enExample)
EA (1) EA028951B9 (enExample)
MX (1) MX2014005351A (enExample)
TW (1) TW201326194A (enExample)
WO (1) WO2013064669A1 (enExample)

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MX2014005351A (es) 2011-11-03 2014-05-28 Zealand Pharma As Conjugados de gastrina peptidicos de agonistas de receptor glp-1.
EA035466B9 (ru) 2013-11-06 2020-08-17 Зилэнд Фарма А/С Соединения и способы на основе двойного агониста гип и гпп-1
EP3066117B1 (en) 2013-11-06 2019-01-02 Zealand Pharma A/S Glucagon-glp-1-gip triple agonist compounds
CA2965732A1 (en) 2014-10-29 2016-05-06 Zealand Pharma A/S Gip agonist compounds and methods
WO2016168388A2 (en) 2015-04-14 2016-10-20 Palatin Technologies, Inc. Therapies for obesity, diabetes and related indications
US10829527B2 (en) * 2016-03-10 2020-11-10 Shenzhen Hightide Biopharmaceutical, Ltd. Conjugates of islet neogenesis peptides and analogs, and methods thereof
SG10201911851VA (en) 2016-12-09 2020-02-27 Zealand Pharma As Acylated glp-1/glp-2 dual agonists
CN111051338B (zh) * 2017-06-29 2024-12-03 乌雷卡有限公司 具有改进的药物学性能的前药肽
CN109248323B (zh) * 2017-07-14 2023-09-08 杭州先为达生物科技有限公司 酰化的glp-1衍生物
CN109331173B (zh) * 2018-12-17 2021-05-07 中国医学科学院医学实验动物研究所 胃泌素-二氧化硅微球及其用途
CN112759640B (zh) * 2020-12-09 2023-09-08 江苏师范大学 一类glp-1/胃泌素受体双重激动剂及其应用
GB202308304D0 (en) * 2023-06-02 2023-07-19 Univ Ulster A fusion peptide for activation of the apj and/or glp-1 receptors

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US9259477B2 (en) 2016-02-16
AU2012331053A1 (en) 2014-05-29
BR112014010780A2 (pt) 2017-04-25
WO2013064669A1 (en) 2013-05-10
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EA028951B1 (ru) 2018-01-31
US20160082118A1 (en) 2016-03-24
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AR088636A1 (es) 2014-06-25
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CA2853884A1 (en) 2013-05-10
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